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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
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NF-κB
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Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
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Piperidines
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Pyrimidines
Quinolines
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Cas号索引 1
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Cas号索引 1
1305267-37-1 | Roginolisib
(Catalog# : 25068)
Roginolisib, also known as MSC2360844 and IOA-244, is a potent, orally active and sel
1496510-51-0 | Relacorilant
(Catalog# : 25035)
Relacorilant is discontinued.
1494684-33-1 | Risovalisib mesylate
(Catalog# : 24078)
CYH33 (CYH-33) is a novel potent, PI3Kα-selective inhibitor with IC50 of 5.9 nM/598
1423719-27-0 | (R,S)-BI 1015550
(Catalog# : 230403)
BI 1015550 is a novel PDE4 inhibitor showing a preferential enzymatic inhibition of P
139339-45-0 | Ro 24-7429
(Catalog# : 2320201)
Ro24-7429是一种有效的口服活性HIV-1 反式激活蛋白Tat 拮抗剂和一种
1239729-06-6 | 布瑞拉沙秦(Brilaroxazine)
(Catalog# : 822224)
RP-5063(Brilaroxazine) 是一种多模式的血清素和多巴胺受体调节剂,
1859053-21-6 | Rucaparib Camsylate
(Catalog# : 20316)
Rucaparib camsylate is a potent, orally available inhibitor of poly ADP-ribose polyme
1281870-42-5 | Rhosin hydrochloride
(Catalog# : 21235)
1831116-75-6 | (R,Z)-1-(4-((3-chloro-4-((3-fluorobenzyl)oxy)phenyl)amino) quinazolin-6-yl)but-2-yn-1-one O-morpholin-3-ylmethyl oxime
(Catalog# : 20123102)
1809275-69-1 | Razuprotafib sodium
(Catalog# : 201221)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
1008510-37-9 | Razuprotafib
(Catalog# : 20102901)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
1787294-07-8 | Remibrutinib ( LOU064 )
(Catalog# : 2073103)
Remibrutinib ( LOU064 ) is a Potent and Highly Selective Covalent Inhibitor of Bruton
1809249-37-3 | Remdesivir
(Catalog# : 2071545)
Remdesivir, also known as GS-5734, is a prodrug form of the antiviral nucleoside anal
171230-81-2 | (R)-methyl 2-(tert-butyldimethylsilyloxy)propanoate
(Catalog# : 202329)
1221443-23-7 | 3-[(2RS)-tetrahydro-2H-pyran-2-yloxy]propanoic acid
(Catalog# : 2062017)
1369768-29-5 | [(1R,2S)-2-(3-fluorophenyl)-2-(hydroxymethyl)cyclopropyl]-methyl acetate
(Catalog# : 2062004)
1443530-05-9 | Rogaratinib
(Catalog# : 192277)
Rogaratinib, 也称为BAY-1163877, 是一种异常的成纤维细胞生长因子受体
1342276-76-9 | RKI-1313
(Catalog# : 19183)
RKI-1313是RKI-1447 (GLXC-05200)的阴性对照,是Rho-相关ROCK激酶的有效抑
1187075-34-8 | Resminostat HCl
(Catalog# : 185317)
Resminostat HCl是一种有效的HDAC1/3/6抑制剂。
1454288-88-0 | Rovazolac
(Catalog# : 185234)
Rovazolac是一种抗炎药。
189744-46-5 | RO10-5824
(Catalog# : 185141)
RO10-5824是一种D4-选择性局部激动剂。RO10-5824是管理可卡因使用障碍
117086-68-7 | 利卡司琼
(Catalog# : 184281)
利卡司琼,也称为Brl 46470,是止吐剂。
1289023-67-1 | Rimegepant
(Catalog# : 18441)
Rimegepant,也称为BMS-927711,在治疗偏头痛的临床试验中,是一种有
1792180-81-4 | Ritlecitinib ( PF-06651600 )
(Catalog# : 18435)
Ritlecitinib ( PF-06651600 )是一种有效的选择性JAK3抑制剂,是一种具有
1174018-99-5 | Relebactam
(Catalog# : 1712156)
Relebactam, also known as MK-7655, a potent and selective β-lactamase inhibitor.
158681-13-1 | 盐酸利莫那班
(Catalog# : 179137)
利莫那班,又名SR141716,是一种抑制食欲的减肥药。它是为大麻素
147254-64-6 | 雷尼司他
(Catalog# : 178118)
雷尼司他,也被称为AS-3201、SX-3201,是一种醛糖还原酶抑制剂,由Dai
1449598-06-4 | RG7800 ( RO6885247 )
(Catalog# : 174192)
RG7800(RO6885247)是一种小分子改变生存运动神经元2的拼接。
1628838-42-5 | RAF709
(Catalog# : 17030605)
RAF709是一种Raf激酶抑制剂。
1211443-80-9 | Ribociclib HCl
(Catalog# : 17011305)
Ribociclib HCl是一种有效且可口服的细胞周期蛋白依赖性激酶(CDK)抑
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
-- PROTAC
----
Molecular Glues
--
Antibody-drug Conjugate/ADC Related
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2102501-84-6 | PF-06835919 ( MDK-1846 )
(Catalog# : 193264)
MDK1846是一种强效的酮己糖激酶(KHK)抑制剂。
2671128-05-3 | FHD-286
(Catalog# : 20471)
FHD-286 is an oral, small-molecule, selective, allosteric inhibitor of BRG1 and BRM i
3002056-30-3 | NST-628
(Catalog# : 24058)
NST-628 是具有血脑屏障渗透性的 MAPK 通路分子胶,能够抑制 RAF 磷
2893778-31-7 | PHGDH-IN-3
(Catalog# : 25077)
PHGDH-IN-3 is an orally active phosphoglycerate dehydrogenase (PHGDH) inhibitor.
2882165-79-7 | CFT1946
(Catalog# : 25078)
CFT1946 是一种口服生物可利用的小分子降解剂,可降解实体瘤中的
68238-36-8 | 异硫蓝
(Catalog# : 178017)
Isosulfan blue 是一种用于淋巴管造影中淋巴管识别的蓝色染料。Isos
2803470-63-3 | HC-7366
(Catalog# : 25076)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
2226636-04-8 | Soquelitinib ( CPI-818 )
(Catalog# : 20671)
Soquelitinib(CPI-818)是一种高度选择性的共价白细胞介素-2诱导的T
2230263-60-0 | Crelosidenib
(Catalog# : 24101)
Crelosidenib is an isocitrate dehydrogenase 1 (IDH1) inhibitor. It is an antineoplast
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12 is a potent STAT3 inhibitor. LLL12 inhibits colony formation and cell migration