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抑制剂/受体激动剂
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Anti-infection
Apoptosis
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Cas号索引 1
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Cas号索引 1
1494684-33-1 | Risovalisib mesylate
(Catalog# : 24078)
CYH33 (CYH-33) is a novel potent, PI3Kα-selective inhibitor with IC50 of 5.9 nM/598
1423719-27-0 | (R,S)-BI 1015550
(Catalog# : 230403)
BI 1015550 is a novel PDE4 inhibitor showing a preferential enzymatic inhibition of P
139339-45-0 | Ro 24-7429
(Catalog# : 2320201)
Ro24-7429是一种有效的口服活性HIV-1 反式激活蛋白Tat 拮抗剂和一种
1239729-06-6 | 布瑞拉沙秦(Brilaroxazine)
(Catalog# : 822224)
RP-5063(Brilaroxazine) 是一种多模式的血清素和多巴胺受体调节剂,
1859053-21-6 | Rucaparib Camsylate
(Catalog# : 20316)
Rucaparib camsylate is a potent, orally available inhibitor of poly ADP-ribose polyme
1281870-42-5 | Rhosin hydrochloride
(Catalog# : 21235)
1831116-75-6 | (R,Z)-1-(4-((3-chloro-4-((3-fluorobenzyl)oxy)phenyl)amino) quinazolin-6-yl)but-2-yn-1-one O-morpholin-3-ylmethyl oxime
(Catalog# : 20123102)
1809275-69-1 | Razuprotafib sodium
(Catalog# : 201221)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
1008510-37-9 | Razuprotafib
(Catalog# : 20102901)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
1787294-07-8 | Remibrutinib ( LOU064 )
(Catalog# : 2073103)
Remibrutinib ( LOU064 ) is a Potent and Highly Selective Covalent Inhibitor of Bruton
1809249-37-3 | Remdesivir
(Catalog# : 2071545)
Remdesivir, also known as GS-5734, is a prodrug form of the antiviral nucleoside anal
171230-81-2 | (R)-methyl 2-(tert-butyldimethylsilyloxy)propanoate
(Catalog# : 202329)
1221443-23-7 | 3-[(2RS)-tetrahydro-2H-pyran-2-yloxy]propanoic acid
(Catalog# : 2062017)
1369768-29-5 | [(1R,2S)-2-(3-fluorophenyl)-2-(hydroxymethyl)cyclopropyl]-methyl acetate
(Catalog# : 2062004)
1443530-05-9 | Rogaratinib
(Catalog# : 192277)
Rogaratinib, 也称为BAY-1163877, 是一种异常的成纤维细胞生长因子受体
1342276-76-9 | RKI-1313
(Catalog# : 19183)
RKI-1313是RKI-1447 (GLXC-05200)的阴性对照,是Rho-相关ROCK激酶的有效抑
1187075-34-8 | Resminostat HCl
(Catalog# : 185317)
Resminostat HCl是一种有效的HDAC1/3/6抑制剂。
1454288-88-0 | Rovazolac
(Catalog# : 185234)
Rovazolac是一种抗炎药。
189744-46-5 | RO10-5824
(Catalog# : 185141)
RO10-5824是一种D4-选择性局部激动剂。RO10-5824是管理可卡因使用障碍
117086-68-7 | 利卡司琼
(Catalog# : 184281)
利卡司琼,也称为Brl 46470,是止吐剂。
1289023-67-1 | Rimegepant
(Catalog# : 18441)
Rimegepant,也称为BMS-927711,在治疗偏头痛的临床试验中,是一种有
1792180-81-4 | Ritlecitinib ( PF-06651600 )
(Catalog# : 18435)
Ritlecitinib ( PF-06651600 )是一种有效的选择性JAK3抑制剂,是一种具有
1174018-99-5 | Relebactam
(Catalog# : 1712156)
Relebactam, also known as MK-7655, a potent and selective β-lactamase inhibitor.
158681-13-1 | 盐酸利莫那班
(Catalog# : 179137)
利莫那班,又名SR141716,是一种抑制食欲的减肥药。它是为大麻素
147254-64-6 | 雷尼司他
(Catalog# : 178118)
雷尼司他,也被称为AS-3201、SX-3201,是一种醛糖还原酶抑制剂,由Dai
1449598-06-4 | RG7800 ( RO6885247 )
(Catalog# : 174192)
RG7800(RO6885247)是一种小分子改变生存运动神经元2的拼接。
1628838-42-5 | RAF709
(Catalog# : 17030605)
RAF709是一种Raf激酶抑制剂。
1211443-80-9 | Ribociclib HCl
(Catalog# : 17011305)
Ribociclib HCl是一种有效且可口服的细胞周期蛋白依赖性激酶(CDK)抑
112887-68-0 | 雷替曲塞
(Catalog# : 17011303)
雷替曲塞,也称为ZD 1694, 是1998年以来用于治疗结直肠癌的一种抗代
150812-13-8 | 瑞替加滨
(Catalog# : 17011108)
瑞替加滨是一种新型的抗惊厥剂,具有活动范围广泛的癫痫模型。
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-- Angiogenesis
----
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----
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----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
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----
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----
DYRK
----
c-Myc
----
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----
ROCK inhibitor
----
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----
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-- Cytoskeleton
----
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----
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----
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----
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----
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----
β-catenin
----
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-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
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----
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----
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----
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----
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----
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----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
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----
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----
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----
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----
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----
Histone Demethylase
----
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----
HDAC
----
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----
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----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
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----
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----
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----
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----
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----
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----
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MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
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EAAT2
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GABA Receptor
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----
Na+/K+ ATPase
----
nAChR
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----
GlyT1
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P2X Receptor
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P-glycoprotein
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----
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-- Metabolic Enzyme/Protease
----
PPAR
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----
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----
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----
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----
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----
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----
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----
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----
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----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
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----
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----
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----
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----
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----
UGT
----
MMP
----
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----
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----
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----
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----
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----
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----
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----
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----
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-- Neuronal Signaling
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
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----
Vps34
-- Stem Cells & Wnt
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ROCK
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----
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----
smo
----
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-- TGF-beta/Smad
----
PKC
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ROCK
----
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-- Ubiquitin
----
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----
p97
----
Deubiquitinase
----
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Antibody-drug Conjugate/ADC Related
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Newest added products
-- Nuclear Receptor
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抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
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--
Boronic Acids
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On Sale
新产品
天然化合物
最新产品
3054692-62-2 | ECI830
(Catalog# : 26A031)
ECI830是一种实验性的CDK2抑制剂。
1394076-92-6 | GNE-317
(Catalog# : 52282)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
3118994-80-9 | DPTX-3186
(Catalog# : 26A010)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
435327-40-5 | Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
1421936-85-7 | Iclepertin (BI-425809)
(Catalog# : 24084)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
4727-31-5 | Kartogenin ( KGN )
(Catalog# : 52215)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
218791-21-0 | Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
2311863-36-0 | Apecotrep (BI 764198)
(Catalog# : 26A048)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
902614-04-4 | Pantothenate kinase-IN-2
(Catalog# : 26A038)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
3062177-59-4 | BH-30643
(Catalog# : 26A047)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制