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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
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Protein Tyrosine Kinase
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Cas号索引 1
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Cas号索引 1
1629869-44-8 | Pimodivir ( VX-787 )
(Catalog# : 2071401)
Pimodivir (VX-787) 是一种可口服的甲型流感病毒聚合酶抑制剂,通过
1454619-14-7 | PU-WS13
(Catalog# : 206701)
PU-WS13 is a potent, Grp94-specific Hsp90 inhibitor of the purine scaffold class. PU-
1953130-87-4 | PTI-428(PTI428)
(Catalog# : 31619)
PTI-428是一种研究性CFTR放大器,开发用于治疗CFTR基因中发生F508del
1415637-72-7 | PF-05085727
(Catalog# : 1932011)
PF-05085727是一种强效、选择性和脑穿透性磷酸二酯酶2A抑制剂。
1252637-35-6 | Petesicatib
(Catalog# : 193206)
Petesicatib是一种组织蛋白酶抑制剂的候选药物。
187235-37-6 | Pretomanid
(Catalog# : 193110)
Pretomanid,也被称为PA-824,一种生物还原药物。PA-824具有较强的体
1341224-83-6 | PF-4136309
(Catalog# : 192282)
PF-4136309,又称INCB8761,是一种口服的人趋化因子受体2 (CCR2)拮抗剂
1078166-57-0 | PF04418948
(Catalog# : 191141)
PF-04418948是一种新型高效选择性前列腺素EP2受体拮抗剂。
1352879-65-2 | PF74
(Catalog# : 1812253)
PF-3450074,又称PF74,是一种针对HIV衣壳蛋白的HIV-1抑制剂。PF74与HI
1672665-49-4 | PT2385
(Catalog# : 1812135)
PT2385是一种口服活性小分子缺氧诱导因子(HIF)-2alpha抑制剂,具有潜
133413-70-4 | PF 1022A
(Catalog# : 1811232)
PF1022A是一种新型的驱虫药,与嗜乳激素样跨膜受体结合,对线虫
146464-95-1 | 普拉曲沙
(Catalog# : 1811221)
普拉曲沙是二氢叶酸还原酶(DHFR)的一种叶酸模拟抑制剂,对叶酸还
1037589-69-7 | PF-05231023
(Catalog# : 1811162)
PF-05231023是一种长效FGF21仿生产品。PF-05231023可以减轻非人类灵长类
1311174-68-1 | PH-002
(Catalog# : 1810234)
PH-002是一种新型的载脂蛋白(apo) E4分子内区域相互作用的神经细胞
1513857-77-6 | Pemigatinib (INCB054828)
(Catalog# : 1810164)
Pemigatinib是一种酪氨酸激酶抑制剂,也是一种抗肿瘤药物候选药物
1022899-36-0 | PCI-33380
(Catalog# : 18943)
PCI-33380是基于ibrutinib支架设计的,已被用于细胞和体内研究,证实
1613373-33-3 | PCO371
(Catalog# : 187125)
PCO371是一种有效的、选择性的PTHR1激动剂,用于治疗低甲状旁腺功
1927857-61-1 | PQR530
(Catalog# : 18756)
PQR530是一种高效的日常pan-PI3K/mTORC1/2抑制剂。
1269662-73-8 | Pyrotinib
(Catalog# : 18731)
Pyrotinib,又称SHR -1258,是一种口服生物利用的双激酶抑制剂,是表
1268244-85-4 | PX20606反式消旋体
(Catalog# : 186274)
PX20606, 也称为PX-102, 是一种FXR激动剂。
1394033-54-5 | PF-05180999
(Catalog# : 186153)
PF-05180999是一个强有力的和选择性PDE2a抑制剂(PDE2a的IC50 = 0.001μM,
1428333-96-3 | Pritelivir甲磺酸盐
(Catalog# : 186152)
Pritelivir,又名AIC-316和BAY 57-1293,是一种有效的螺旋酶抑制剂。
1446261-44-4 | Pamiparib
(Catalog# : 185233)
Pamiparib是高选择性PARP-1/2抑制剂。临床试验中表现出良好的抗肿瘤
1005168-10-4 | PAC 14028
(Catalog# : 185223)
PAC-14028是高效的选择性的瞬时受体电位香草酸亚型1 (TRPV1) 拮抗剂
1402727-29-0 | PE859
(Catalog# : 185157)
PE859是一个强有力的IC50值分别为0.66和1.2μM的tau和Aβ聚合抑制剂。
190383-31-4 | PD 168 077
(Catalog# : 185156)
PD168077是一种多巴胺D4受体激动剂,对记忆巩固有促进作用。
1622291-66-0 | PF-06462894
(Catalog# : 185155)
PF-06462894是一种形态学上的mGlu5 (mGlu5 Ki = 6nm)。
1393124-08-7 | PF-06291874
(Catalog# : 185154)
PF-06291874是一种胰高血糖素受体拮抗剂,对2型糖尿病患者有效。
1353552-97-2 | Poseltinib
(Catalog# : 185153)
Poseltinib, 也称为HM-71224和LY3337641,一种酪氨酸激酶抑制剂。
1353900-92-1 | Pibrentasvir
(Catalog# : 185148)
Pibrentasvir,也被称为ABT-530,是一种蛋白酶抑制剂,可用于治疗丙
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
845959-55-9 | Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
1246960-09-7 | SPG-601 ( VSN-16R )
(Catalog# : 24042)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
1421438-81-4 | LY3039478 ( Crenigacestat )
(Catalog# : 17021601)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
72882-78-1 | PF-9366
(Catalog# : 184107)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
2925330-18-1 | MAT2A-IN-22
(Catalog# : 26A021)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
| Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
2361124-03-8 | Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
2170608-85-0 | PZ-3022
(Catalog# : 26A039)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
2170608-82-7 | PZ-2891
(Catalog# : 193282)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
902614-04-4 | Pantothenate kinase-IN-2
(Catalog# : 26A038)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,