武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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Aldehydes
Amines
Amino Acids
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Boronic Acids
Bromides
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Deuterated
Fluorides
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Indoles and Oxindoles
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Pyridines
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 V
Valecobulin
(Catalog# : 193114, Cas# :
1188371-47-2
)
Valecobulin是一种抗肿瘤的β-微管蛋白聚合抑制剂。微管蛋白聚合抑
Vecabrutinib
(Catalog# : 192154, Cas# :
1510829-06-7
)
Vecabrutinib,又名SNS-062;FP-182, BSK-4841, BIIB-062;是一种有效的,非共价
Valemetostat
(Catalog# : 192141, Cas# :
1809336-39-7
)
Valemetostat是一种抗肿瘤药物。
Verdiperstat
(Catalog# : 1812285, Cas# :
890655-80-8
)
Verdiperstat,又称AZD-3241,是一种选择性和不可逆的髓过氧化物酶抑
Vaborbactam
(Catalog# : 181253, Cas# :
1360457-46-0
)
Vaborbactam,也称为RPX7009, 是一种有效且具有选择性的β-内酰胺酶抑
VU0463271
(Catalog# : 1810151, Cas# :
1391737-01-1
)
VU0463271抑制协同转运蛋白KCC2。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
Verteporfin
(Catalog# : 187201, Cas# :
129497-78-5
)
Verteporfin,也被称为苯卟啉衍生物A或BPD-MA,是一种苯卟啉衍生物,
维立韦罗马来酸盐
(Catalog# : 185214, Cas# :
599179-03-0
)
维立韦罗,也称为SCH 417690和SCH-D, 是一种有效的、具有口服活性和选
Verinurad
(Catalog# : 18583, Cas# :
1352792-74-5
)
Verinurad,也称为RDEA3170,是一种有机阴离子转运体URAT1 (SLC22A12)抑制
VcMMAE
(Catalog# : 18582, Cas# :
646502-53-6
)
VcMMAE是一种MMAE衍生物,它与valine-citrulline (Vc)链接器。VcMMAE可用于
VH298
(Catalog# : 18581, Cas# :
2097381-85-4
)
VH298是一种有效的VHL抑制剂,通过不同的机制和抒发缺氧反应稳定
VU0467154
(Catalog# : 18576, Cas# :
1451993-15-9
)
VU0467154 is a positive allosteric modulator of theM4 muscarinic acetylcholine recept
Voxilaprevir
(Catalog# : 18572, Cas# :
1535212-07-7
)
Voxilaprevir是一种丙型肝炎病毒(HCV)非结构蛋白3/4A蛋白酶抑制剂。
Verubecestat TFA
(Catalog# : 18417, Cas# :
2095432-65-6
)
Verubecestat,也被称为MK-8931或SCH 900931,是一种有效的选择性的-分泌
Valbenazine
(Catalog# : 1783010, Cas# :
1025504-45-3
)
Valbenazine,也叫 NBI- 98854和MT - 5199,是一种有效的选择性的VMAT2抑制
沃拉帕沙
(Catalog# : 178307, Cas# :
705260-08-8
)
沃拉帕沙,也被称为SCH 530348,是一种基于天然产品himbacine的凝血
Voruciclib
(Catalog# : 178306, Cas# :
1000023-04-0
)
Voruciclib,又称P1446A-05,是一种蛋白质激酶抑制剂,专门针对细胞
Voxelotor(GBT440, GTX011)
(Catalog# : 178916, Cas# :
1446321-46-5
)
Voxelotor(GBT440,GTX011)是一种新的小分子化合物,它能增加血红蛋白与
维利西呱
(Catalog# : 2017886, Cas# :
1350653-20-1
)
维利西呱,也称为BAY1021189或BAY10-21189, 是一种有效和口服活性sGC刺
Varlitinib
(Catalog# : 2017885, Cas# :
845272-21-1
)
ARRY334543是一种有效且选择性的ErbB-1和ErbB-2抑制剂(IC50分别为7和2 n
VX-984 (M9831)
(Catalog# : 2017879, Cas# :
1562396-65-9
)
VX-984, 也称为M9831,是一种ATP-竞争性抑制剂,依赖蛋白激酶(DNA-PK)的
Volasertib
(Catalog# : 20178219, Cas# :
755038-65-4
)
Volasertib, 也称为BI-6727,是一种dihydropteridinone Polo样激酶1 (Plk1) 抑制
VPS34抑制剂1
(Catalog# : 17031001, Cas# :
1383716-46-8
)
VPS34抑制剂1(化合物19, PIK-III类似物)是VPS34的有效和选择性抑制剂,
维帕他韦
(Catalog# : 17022808, Cas# :
1377049-84-7
)
维帕他韦(VEL, GS-5816)是一种新的泛基因型丙型肝炎病毒(HCV)非结构
伏立诺他
(Catalog# : 17022704, Cas# :
149647-78-9
)
伏立诺他(SAHA)是IC50为10nm的HDAC1 / 3抑制剂。
氨己烯酸
(Catalog# : 17011903, Cas# :
60643-86-9
)
氨己烯酸, 是一种抗癫痫药物,抑制γ-aminobutyric酸的分解(GABA)充当
Vadadustat ( AKB-6548 )
(Catalog# : 6121401, Cas# :
1000025-07-9
)
Vadadustat (AKB-6548), a novel, titratable, oral hypoxia-inducible factor prolyl hydr
VLX1570
(Catalog# : 611932, Cas# :
1431280-51-1
)
VLX1570 is a competitive inhibitor of proteasome DUB activity with IC50 ranging from
Voxtalisib ( XL-765)
(Catalog# : 160926001, Cas# :
934493-76-2
)
PI3K/mTOR dual kinase inhibitor XL765 inhibits both PI3K kinase and mTOR kinase, whic
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶