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抑制剂/受体激动剂
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Epigenetics
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Cytoskeletal Signaling
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others
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Aldehydes
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Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Deuterated
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Indoles and Oxindoles
Iodos
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Peg Linkers
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Quinolines
Sulfonamides
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Pyridines
Pyrimidines
Quinolines
Sulfonamides
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Trifluoroborates
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Other Heterocycles
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联系我们
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产品名字索引 V
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产品名字索引 V
维立韦罗马来酸盐
(Catalog# : 185214, Cas# :
599179-03-0
)
维立韦罗,也称为SCH 417690和SCH-D, 是一种有效的、具有口服活性和选
Verinurad
(Catalog# : 18583, Cas# :
1352792-74-5
)
Verinurad,也称为RDEA3170,是一种有机阴离子转运体URAT1 (SLC22A12)抑制
VcMMAE
(Catalog# : 18582, Cas# :
646502-53-6
)
VcMMAE是一种MMAE衍生物,它与valine-citrulline (Vc)链接器。VcMMAE可用于
VH298
(Catalog# : 18581, Cas# :
2097381-85-4
)
VH298是一种有效的VHL抑制剂,通过不同的机制和抒发缺氧反应稳定
VU0467154
(Catalog# : 18576, Cas# :
1451993-15-9
)
VU0467154 is a positive allosteric modulator of theM4 muscarinic acetylcholine recept
Voxilaprevir
(Catalog# : 18572, Cas# :
1535212-07-7
)
Voxilaprevir是一种丙型肝炎病毒(HCV)非结构蛋白3/4A蛋白酶抑制剂。
Verubecestat TFA
(Catalog# : 18417, Cas# :
2095432-65-6
)
Verubecestat,也被称为MK-8931或SCH 900931,是一种有效的选择性的-分泌
Valbenazine
(Catalog# : 1783010, Cas# :
1025504-45-3
)
Valbenazine,也叫 NBI- 98854和MT - 5199,是一种有效的选择性的VMAT2抑制
沃拉帕沙
(Catalog# : 178307, Cas# :
705260-08-8
)
沃拉帕沙,也被称为SCH 530348,是一种基于天然产品himbacine的凝血
Voruciclib
(Catalog# : 178306, Cas# :
1000023-04-0
)
Voruciclib,又称P1446A-05,是一种蛋白质激酶抑制剂,专门针对细胞
Voxelotor(GBT440, GTX011)
(Catalog# : 178916, Cas# :
1446321-46-5
)
Voxelotor(GBT440,GTX011)是一种新的小分子化合物,它能增加血红蛋白与
维利西呱
(Catalog# : 2017886, Cas# :
1350653-20-1
)
维利西呱,也称为BAY1021189或BAY10-21189, 是一种有效和口服活性sGC刺
Varlitinib
(Catalog# : 2017885, Cas# :
845272-21-1
)
ARRY334543是一种有效且选择性的ErbB-1和ErbB-2抑制剂(IC50分别为7和2 n
VX-984 (M9831)
(Catalog# : 2017879, Cas# :
1562396-65-9
)
VX-984, 也称为M9831,是一种ATP-竞争性抑制剂,依赖蛋白激酶(DNA-PK)的
Volasertib
(Catalog# : 20178219, Cas# :
755038-65-4
)
Volasertib, 也称为BI-6727,是一种dihydropteridinone Polo样激酶1 (Plk1) 抑制
VPS34抑制剂1
(Catalog# : 17031001, Cas# :
1383716-46-8
)
VPS34抑制剂1(化合物19, PIK-III类似物)是VPS34的有效和选择性抑制剂,
维帕他韦
(Catalog# : 17022808, Cas# :
1377049-84-7
)
维帕他韦(VEL, GS-5816)是一种新的泛基因型丙型肝炎病毒(HCV)非结构
伏立诺他
(Catalog# : 17022704, Cas# :
149647-78-9
)
伏立诺他(SAHA)是IC50为10nm的HDAC1 / 3抑制剂。
氨己烯酸
(Catalog# : 17011903, Cas# :
60643-86-9
)
氨己烯酸, 是一种抗癫痫药物,抑制γ-aminobutyric酸的分解(GABA)充当
Vadadustat ( AKB-6548 )
(Catalog# : 6121401, Cas# :
1000025-07-9
)
Vadadustat (AKB-6548), a novel, titratable, oral hypoxia-inducible factor prolyl hydr
VLX1570
(Catalog# : 611932, Cas# :
1431280-51-1
)
VLX1570 is a competitive inhibitor of proteasome DUB activity with IC50 ranging from
Voxtalisib ( XL-765)
(Catalog# : 160926001, Cas# :
934493-76-2
)
PI3K/mTOR dual kinase inhibitor XL765 inhibits both PI3K kinase and mTOR kinase, whic
Vorapaxar(free base)
(Catalog# : 16070916, Cas# :
618385-01-6
)
Vorapaxar, also known as SCH 530348, is a thrombin receptor (protease-activated recep
VX-702
(Catalog# : 16070804, Cas# :
745833-23-2
)
VX-702, one of a series of second-generation, is an orally active p38 MAP kinase inhi
Vsp34-IN-1
(Catalog# : 011115, Cas# :
1523404-29-6
)
Coming soon!
VP 14637
(Catalog# : 011112, Cas# :
235106-62-4
)
Coming soon!
Vipadenant
(Catalog# : 010436, Cas# :
442908-10-3
)
Vipadenant is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69
Vatalanib
(Catalog# : 010434, Cas# :
212141-54-3
)
Vatalanib free base is an inhibitor of VEGFR2/KDR with IC50 of 37 nM, less potent aga
VE-821
(Catalog# : 122817, Cas# :
1232410-49-9
)
VE-821 is a potent and selective ATP competitive inhibitor of ATR with Ki/IC50 of 13
VU 0364439
(Catalog# : 122401, Cas# :
1246086-78-1
)
VU 0364439 is a mGlu4 positive allosteric modulator, with EC50 of 19.8 nM.
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).
NVL-655 ( ALK-IN-27 )
(Catalog# : 24003, Cas# :
2739866-40-9
)
NVL-655是一种新型脑渗透性ALK选择性抑制剂,旨在解决目前可用的