武汉永璨生物科技有限公司
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
Nuclear Receptor
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
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Chiral Compounds
Deuterated
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Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 V
Vesatolimod(GS-9620)
(Catalog# : 19529, Cas# :
1228585-88-3
)
DescriptionGS-9620 is a potent and selective orally active small molecule agonist ofT
Valecobulin
(Catalog# : 193114, Cas# :
1188371-47-2
)
Valecobulin是一种抗肿瘤的β-微管蛋白聚合抑制剂。微管蛋白聚合抑
Vecabrutinib
(Catalog# : 192154, Cas# :
1510829-06-7
)
Vecabrutinib,又名SNS-062;FP-182, BSK-4841, BIIB-062;是一种有效的,非共价
Valemetostat
(Catalog# : 192141, Cas# :
1809336-39-7
)
Valemetostat是一种抗肿瘤药物。
Verdiperstat
(Catalog# : 1812285, Cas# :
890655-80-8
)
Verdiperstat,又称AZD-3241,是一种选择性和不可逆的髓过氧化物酶抑
Vaborbactam
(Catalog# : 181253, Cas# :
1360457-46-0
)
Vaborbactam,也称为RPX7009, 是一种有效且具有选择性的β-内酰胺酶抑
VU0463271
(Catalog# : 1810151, Cas# :
1391737-01-1
)
VU0463271抑制协同转运蛋白KCC2。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
Verteporfin
(Catalog# : 187201, Cas# :
129497-78-5
)
Verteporfin,也被称为苯卟啉衍生物A或BPD-MA,是一种苯卟啉衍生物,
维立韦罗马来酸盐
(Catalog# : 185214, Cas# :
599179-03-0
)
维立韦罗,也称为SCH 417690和SCH-D, 是一种有效的、具有口服活性和选
Verinurad
(Catalog# : 18583, Cas# :
1352792-74-5
)
Verinurad,也称为RDEA3170,是一种有机阴离子转运体URAT1 (SLC22A12)抑制
VcMMAE
(Catalog# : 18582, Cas# :
646502-53-6
)
VcMMAE是一种MMAE衍生物,它与valine-citrulline (Vc)链接器。VcMMAE可用于
VH298
(Catalog# : 18581, Cas# :
2097381-85-4
)
VH298是一种有效的VHL抑制剂,通过不同的机制和抒发缺氧反应稳定
VU0467154
(Catalog# : 18576, Cas# :
1451993-15-9
)
VU0467154 is a positive allosteric modulator of theM4 muscarinic acetylcholine recept
Voxilaprevir
(Catalog# : 18572, Cas# :
1535212-07-7
)
Voxilaprevir是一种丙型肝炎病毒(HCV)非结构蛋白3/4A蛋白酶抑制剂。
Verubecestat TFA
(Catalog# : 18417, Cas# :
2095432-65-6
)
Verubecestat,也被称为MK-8931或SCH 900931,是一种有效的选择性的-分泌
Valbenazine
(Catalog# : 1783010, Cas# :
1025504-45-3
)
Valbenazine,也叫 NBI- 98854和MT - 5199,是一种有效的选择性的VMAT2抑制
沃拉帕沙
(Catalog# : 178307, Cas# :
705260-08-8
)
沃拉帕沙,也被称为SCH 530348,是一种基于天然产品himbacine的凝血
Voruciclib
(Catalog# : 178306, Cas# :
1000023-04-0
)
Voruciclib,又称P1446A-05,是一种蛋白质激酶抑制剂,专门针对细胞
Voxelotor(GBT440, GTX011)
(Catalog# : 178916, Cas# :
1446321-46-5
)
Voxelotor(GBT440,GTX011)是一种新的小分子化合物,它能增加血红蛋白与
维利西呱
(Catalog# : 2017886, Cas# :
1350653-20-1
)
维利西呱,也称为BAY1021189或BAY10-21189, 是一种有效和口服活性sGC刺
Varlitinib
(Catalog# : 2017885, Cas# :
845272-21-1
)
ARRY334543是一种有效且选择性的ErbB-1和ErbB-2抑制剂(IC50分别为7和2 n
VX-984 (M9831)
(Catalog# : 2017879, Cas# :
1562396-65-9
)
VX-984, 也称为M9831,是一种ATP-竞争性抑制剂,依赖蛋白激酶(DNA-PK)的
Volasertib
(Catalog# : 20178219, Cas# :
755038-65-4
)
Volasertib, 也称为BI-6727,是一种dihydropteridinone Polo样激酶1 (Plk1) 抑制
VPS34抑制剂1
(Catalog# : 17031001, Cas# :
1383716-46-8
)
VPS34抑制剂1(化合物19, PIK-III类似物)是VPS34的有效和选择性抑制剂,
维帕他韦
(Catalog# : 17022808, Cas# :
1377049-84-7
)
维帕他韦(VEL, GS-5816)是一种新的泛基因型丙型肝炎病毒(HCV)非结构
伏立诺他
(Catalog# : 17022704, Cas# :
149647-78-9
)
伏立诺他(SAHA)是IC50为10nm的HDAC1 / 3抑制剂。
氨己烯酸
(Catalog# : 17011903, Cas# :
60643-86-9
)
氨己烯酸, 是一种抗癫痫药物,抑制γ-aminobutyric酸的分解(GABA)充当
Vadadustat ( AKB-6548 )
(Catalog# : 6121401, Cas# :
1000025-07-9
)
Vadadustat (AKB-6548), a novel, titratable, oral hypoxia-inducible factor prolyl hydr
VLX1570
(Catalog# : 611932, Cas# :
1431280-51-1
)
VLX1570 is a competitive inhibitor of proteasome DUB activity with IC50 ranging from
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制