武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
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定制合成
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订购信息
联系我们
公司简介
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产品名字索引 T
TLR4-C34
(Catalog# : 2061501, Cas# :
40592-88-9
)
TLR4-C34 is a TLR4 inhibitor that inhibits TLR4 signaling in enterocytes and macropha
TH257
(Catalog# : 2061311, Cas# :
2244678-29-1
)
TH257 is a Potent and selective allosteric LIMK 1/2 inhibitor.
TH-263
(Catalog# : 2061303, Cas# :
313520-94-4
)
TH-263 is an inactive analog control for the type III allosteric LIM-kinase (LIMK) in
2,4,6-三[(1,1-联苯)-4-基]-1,3-5-三嗪
(Catalog# : S-204158, Cas# :
31274-51-8
)
4-(2,2,2-三氟乙氧基)苯基硼酸
(Catalog# : S-203041, Cas# :
886536-37-4
)
g scale to Kg scale may be provided.
TVB-3664
(Catalog# : 2041503)
TVB-3664 is a FASN inhibitor which significantly reduces tubulin palmitoylation and m
TD-106
(Catalog# : 193184, Cas# :
2250288-69-6
)
TD-106是一种可用于靶向蛋白降解的小脑(CRBN)调制器。TD-106诱导BRD4
Tafamidis meglumine
(Catalog# : 193183, Cas# :
951395-08-7
)
Tafamidis meglumine,也被称为Fx-1006或PF-06291826,是一种改善经胸腺素
Tafamidis
(Catalog# : 193182, Cas# :
594839-88-0
)
Tafamidis也被称为Fx-1006或PF-06291826,是一种改善经胸腺素相关的遗传
TH287
(Catalog# : 193135, Cas# :
1609960-30-6
)
TH287是人7,8-二氢-8-草酸鸟苷三磷酸酶MTH1 (NUDT1)的有效抑制剂,IC50
Tinostamustine盐酸盐
(Catalog# : 193112, Cas# :
1793059-58-1
)
Tinostamustine,也称为EDO-S101,是一种烷基化有机去乙酰化酶抑制剂(H
Telithromycin
(Catalog# : 19374, Cas# :
191114-48-4
)
Telithromycin,也被称为HMR-3647和RU-66647,是一种半合成红霉素衍生物
TH34
(Catalog# : 192273, Cas# :
2196203-96-8
)
TH34是一种有效的HDAC6/8/10抑制剂。TH34在人类高级别神经母细胞瘤细
THZ2
(Catalog# : 192252, Cas# :
1604810-84-5
)
THZ2,是THZ1的类似物,具有治疗三阴性乳腺癌(TNBC)的潜力,是一种
Tegatrabetan
(Catalog# : 192145, Cas# :
1227637-23-1
)
Tegatrabetan, 也称为Tegavivint和BC2059,是一种口服生物利用率和有效的
Telratolimod
(Catalog# : 192144, Cas# :
1359993-59-1
)
Telratolimod,也被称为 3M-052或MEDI-9197,是toll样受体7 (TLR-7)和toll样受
TAS-116
(Catalog# : 191286, Cas# :
1260533-36-5
)
TAS- 116是一种对热休克蛋白90 (Hsp90)亚型alpha和beta的有效选择性抑制
他米巴罗汀
(Catalog# : 191254, Cas# :
94497-51-5
)
他米巴罗汀,也称为SY-1425,是一种具有口服活性的合成类维生素
Tafenoquine succinate ( 他非诺喹琥珀酸盐 )
(Catalog# : 191123, Cas# :
106635-81-8
)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
Tafenoquine ( 他非诺喹 )
(Catalog# : 191122, Cas# :
106635-80-7
)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
TP0463518
(Catalog# : 1812282, Cas# :
1558021-37-0
)
TP0463518是一种新型高效的HIF脯氨酰羟化酶(PHD)抑制剂。TP0463518竞争
Thiamet G
(Catalog# : 1812133, Cas# :
1009816-48-1
)
Thiamet G是一种有效且具有选择性的O-GlcNAcase抑制剂.
他匹莫德盐酸盐
(Catalog# : 181252, Cas# :
309915-12-6
)
他匹莫德,又称SCIO-469,是一种口服生物可利用的小分子p38丝裂原
TG4-155
(Catalog# : 181232, Cas# :
1164462-05-8
)
TG4-155 是一种大脑渗透EP2拮抗剂(KB = 2.4nM),在EP4(KB = 11.4µM)小组其他
Tebanicline盐酸盐
(Catalog# : 181231, Cas# :
203564-54-9
)
Tebanicline盐酸盐,也被称为ABT-594和Ebanicline,是雅培公司开发的一
Topotecan
(Catalog# : 1811212, Cas# :
123948-87-8
)
Topocecan是喜树碱的半合成衍生物,具有抗肿瘤活性。
TAS-120
(Catalog# : 1811191, Cas# :
1448169-71-8
)
TAS-120是成纤维细胞生长因子受体(FGFR)的口服生物有效抑制剂,具
Tulrampator ( CX-1632 )
(Catalog# : 1811161, Cas# :
1038984-31-4
)
Tulrampator,也被称为S-47445和CX-1632,是AMPA受体(AMPAR)的积极变构调制
Thiazovivin
(Catalog# : 1811122, Cas# :
1226056-71-8
)
Thiazovivin是一种具有选择性的,抑制浓度为2µM的ROCK活动的细胞-渗透
TH 1217
(Catalog# : 1811021, Cas# :
1862212-48-3
)
TH 1217是一种有效的dCTP焦磷酸酶1抑制剂。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
MTX115325
(Catalog# : 186264, Cas# :
2750895-97-5
)
MTX115325是一种强效、选择性、脑渗透性USP30抑制剂,具有良好的类
LY-3381916
(Catalog# : 193123, Cas# :
2166616-75-5
)
LY-3381916是一种强效的、选择性的、脑透性的IDO1活性抑制剂,与缺
Opakalim
(Catalog# : 25193, Cas# :
2376397-93-0
)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
DS68591889
(Catalog# : 25158, Cas# :
2488609-21-6
)
DS68591889 (PTDSS1i) 特异性抑制 PTDSS1,而 PTDSS1 可催化丝氨酸掺入 PC。
CAY 10566
(Catalog# : 10403, Cas# :
944808-88-2
)
CAY 10566是一种强效的选择性SCD-1抑制剂。
Cadefrecitinib (GLPG-3667)
(Catalog# : 20509, Cas# :
2308520-97-8
)
Cadefrecitinib(GLPG-3667)是一种口服小分子TYK2激酶抑制剂,目前正处
QBS10072S
(Catalog# : 25190, Cas# :
1802735-28-9
)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的