武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
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Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
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Thiazoles
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产品名字索引 T
Tafenoquine-d3 succinate
(Catalog# : 2061704, Cas# :
1133378-83-2
)
Tafenoquine-d3 is a trideuerium-labeled Tafenoquine derivative. Tafenoquine, also kno
TLR4-C34
(Catalog# : 2061501, Cas# :
40592-88-9
)
TLR4-C34 is a TLR4 inhibitor that inhibits TLR4 signaling in enterocytes and macropha
TH257
(Catalog# : 2061311, Cas# :
2244678-29-1
)
TH257 is a Potent and selective allosteric LIMK 1/2 inhibitor.
TH-263
(Catalog# : 2061303, Cas# :
313520-94-4
)
TH-263 is an inactive analog control for the type III allosteric LIM-kinase (LIMK) in
2,4,6-三[(1,1-联苯)-4-基]-1,3-5-三嗪
(Catalog# : S-204158, Cas# :
31274-51-8
)
4-(2,2,2-三氟乙氧基)苯基硼酸
(Catalog# : S-203041, Cas# :
886536-37-4
)
g scale to Kg scale may be provided.
TVB-3664
(Catalog# : 2041503)
TVB-3664 is a FASN inhibitor which significantly reduces tubulin palmitoylation and m
TD-106
(Catalog# : 193184, Cas# :
2250288-69-6
)
TD-106是一种可用于靶向蛋白降解的小脑(CRBN)调制器。TD-106诱导BRD4
Tafamidis meglumine
(Catalog# : 193183, Cas# :
951395-08-7
)
Tafamidis meglumine,也被称为Fx-1006或PF-06291826,是一种改善经胸腺素
Tafamidis
(Catalog# : 193182, Cas# :
594839-88-0
)
Tafamidis也被称为Fx-1006或PF-06291826,是一种改善经胸腺素相关的遗传
TH287
(Catalog# : 193135, Cas# :
1609960-30-6
)
TH287是人7,8-二氢-8-草酸鸟苷三磷酸酶MTH1 (NUDT1)的有效抑制剂,IC50
Tinostamustine盐酸盐
(Catalog# : 193112, Cas# :
1793059-58-1
)
Tinostamustine,也称为EDO-S101,是一种烷基化有机去乙酰化酶抑制剂(H
Telithromycin
(Catalog# : 19374, Cas# :
191114-48-4
)
Telithromycin,也被称为HMR-3647和RU-66647,是一种半合成红霉素衍生物
TH34
(Catalog# : 192273, Cas# :
2196203-96-8
)
TH34是一种有效的HDAC6/8/10抑制剂。TH34在人类高级别神经母细胞瘤细
THZ2
(Catalog# : 192252, Cas# :
1604810-84-5
)
THZ2,是THZ1的类似物,具有治疗三阴性乳腺癌(TNBC)的潜力,是一种
Tegatrabetan
(Catalog# : 192145, Cas# :
1227637-23-1
)
Tegatrabetan, 也称为Tegavivint和BC2059,是一种口服生物利用率和有效的
Telratolimod
(Catalog# : 192144, Cas# :
1359993-59-1
)
Telratolimod,也被称为 3M-052或MEDI-9197,是toll样受体7 (TLR-7)和toll样受
TAS-116
(Catalog# : 191286, Cas# :
1260533-36-5
)
TAS- 116是一种对热休克蛋白90 (Hsp90)亚型alpha和beta的有效选择性抑制
他米巴罗汀
(Catalog# : 191254, Cas# :
94497-51-5
)
他米巴罗汀,也称为SY-1425,是一种具有口服活性的合成类维生素
Tafenoquine succinate ( 他非诺喹琥珀酸盐 )
(Catalog# : 191123, Cas# :
106635-81-8
)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
Tafenoquine ( 他非诺喹 )
(Catalog# : 191122, Cas# :
106635-80-7
)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
TP0463518
(Catalog# : 1812282, Cas# :
1558021-37-0
)
TP0463518是一种新型高效的HIF脯氨酰羟化酶(PHD)抑制剂。TP0463518竞争
Thiamet G
(Catalog# : 1812133, Cas# :
1009816-48-1
)
Thiamet G是一种有效且具有选择性的O-GlcNAcase抑制剂.
他匹莫德盐酸盐
(Catalog# : 181252, Cas# :
309915-12-6
)
他匹莫德,又称SCIO-469,是一种口服生物可利用的小分子p38丝裂原
TG4-155
(Catalog# : 181232, Cas# :
1164462-05-8
)
TG4-155 是一种大脑渗透EP2拮抗剂(KB = 2.4nM),在EP4(KB = 11.4µM)小组其他
Tebanicline盐酸盐
(Catalog# : 181231, Cas# :
203564-54-9
)
Tebanicline盐酸盐,也被称为ABT-594和Ebanicline,是雅培公司开发的一
Topotecan
(Catalog# : 1811212, Cas# :
123948-87-8
)
Topocecan是喜树碱的半合成衍生物,具有抗肿瘤活性。
TAS-120
(Catalog# : 1811191, Cas# :
1448169-71-8
)
TAS-120是成纤维细胞生长因子受体(FGFR)的口服生物有效抑制剂,具
Tulrampator ( CX-1632 )
(Catalog# : 1811161, Cas# :
1038984-31-4
)
Tulrampator,也被称为S-47445和CX-1632,是AMPA受体(AMPAR)的积极变构调制
Thiazovivin
(Catalog# : 1811122, Cas# :
1226056-71-8
)
Thiazovivin是一种具有选择性的,抑制浓度为2µM的ROCK活动的细胞-渗透
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AD-8007
(Catalog# : 26A018, Cas# :
1497439-74-3
)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
ZY-444
(Catalog# : 26A020, Cas# :
1802650-31-2
)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
AD-5584
(Catalog# : 26A019, Cas# :
2306525-79-9
)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
IDB-003
(Catalog# : 26A017, Cas# :
3079716-11-0
)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
Vafidemstat
(Catalog# : 18891, Cas# :
1357362-02-7
)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
LLL12
(Catalog# : 25075, Cas# :
1260247-42-4
)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
ECC-5004
(Catalog# : 26A015, Cas# :
2758659-09-3
)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
SILA-123
(Catalog# : 26A014, Cas# :
2911585-37-8
)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
Encaleret sulfate
(Catalog# : 26A013, Cas# :
1214922-52-7
)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011, Cas# :
1431303-72-8
)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶