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抑制剂/受体激动剂
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Cytoskeletal Signaling
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others
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Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
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Indoles and Oxindoles
Iodos
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Peg Linkers
Phenols
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Pyridines
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Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
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Other Azoles
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产品名字索引 T
TP0463518
(Catalog# : 1812282, Cas# :
1558021-37-0
)
TP0463518是一种新型高效的HIF脯氨酰羟化酶(PHD)抑制剂。TP0463518竞争
Thiamet G
(Catalog# : 1812133, Cas# :
1009816-48-1
)
Thiamet G是一种有效且具有选择性的O-GlcNAcase抑制剂.
他匹莫德盐酸盐
(Catalog# : 181252, Cas# :
309915-12-6
)
他匹莫德,又称SCIO-469,是一种口服生物可利用的小分子p38丝裂原
TG4-155
(Catalog# : 181232, Cas# :
1164462-05-8
)
TG4-155 是一种大脑渗透EP2拮抗剂(KB = 2.4nM),在EP4(KB = 11.4µM)小组其他
Tebanicline盐酸盐
(Catalog# : 181231, Cas# :
203564-54-9
)
Tebanicline盐酸盐,也被称为ABT-594和Ebanicline,是雅培公司开发的一
Topotecan
(Catalog# : 1811212, Cas# :
123948-87-8
)
Topocecan是喜树碱的半合成衍生物,具有抗肿瘤活性。
TAS-120
(Catalog# : 1811191, Cas# :
1448169-71-8
)
TAS-120是成纤维细胞生长因子受体(FGFR)的口服生物有效抑制剂,具
Tulrampator ( CX-1632 )
(Catalog# : 1811161, Cas# :
1038984-31-4
)
Tulrampator,也被称为S-47445和CX-1632,是AMPA受体(AMPAR)的积极变构调制
Thiazovivin
(Catalog# : 1811122, Cas# :
1226056-71-8
)
Thiazovivin是一种具有选择性的,抑制浓度为2µM的ROCK活动的细胞-渗透
TH 1217
(Catalog# : 1811021, Cas# :
1862212-48-3
)
TH 1217是一种有效的dCTP焦磷酸酶1抑制剂。
TW-37
(Catalog# : 18831, Cas# :
877877-35-5
)
TW-37是Bcl-2家族蛋白的一种小分子抑制剂,抑制了胰腺癌细胞生长
TAK-715
(Catalog# : 187202, Cas# :
303162-79-0
)
TAK-715是一种有效的p38 MAPK抑制剂。它表现出有效的抑制活性,对主
TAK-960
(Catalog# : 18762, Cas# :
1137868-52-0
)
TAK-960是一种可口服的PLK1抑制剂,具有潜在的抗肿瘤活性。
Theliatinib
(Catalog# : 186235, Cas# :
1353644-70-8
)
Theliatinib又称HMPL-309,是一种新型的小分子、表皮生长因子受体酪
Tucidinostat
(Catalog# : 186233, Cas# :
1616493-44-7
)
Tucidinostat是组蛋白去乙酰化酶(HDAC) 1、2、3和10的一种苯甲酰胺类抑
Takinib
(Catalog# : 18672, Cas# :
1111556-37-6
)
Takinib选择性TAK1抑制剂,TNF-α刺激后细胞凋亡模型,类风湿性关节炎
TMP269
(Catalog# : 185254, Cas# :
1314890-29-3
)
TMP269是一种具有高强度、选择性和可渗透性的IIa型HDAC抑制剂,其
Trilaciclib (G1T28)
(Catalog# : 185235, Cas# :
1374743-00-6
)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
TAPI-1
(Catalog# : 185181, Cas# :
171235-71-5
)
TAPI-1是TACE的抑制剂。它抑制TNF-a、TNFRI(p60)和TNFRII(p80)的裂解。
TG100572盐酸盐
(Catalog# : 185175, Cas# :
867331-64-4
)
TG-100572是一种有效且具有选择性的VEGFR2/Src激酶抑制剂。
TLN-232
(Catalog# : 18594, Cas# :
158899-10-6
)
TLN-232, 也称为CAP-232,是一种具有潜在抗肿瘤活性的合成环七肽。
TRC051384
(Catalog# : 18593, Cas# :
867164-40-7
)
TRC051384是热休克蛋白Hsp70的诱导物。
醋酸曲普瑞林
(Catalog# : 18592, Cas# :
140194-24-7
)
醋酸曲普瑞林是一种促性腺激素释放激素激动剂(GnRH激动剂),用作
Tropifexor
(Catalog# : 18591, Cas# :
1383816-29-2
)
Tropifexor, 也称为LJN452, 是一种用于治疗胆静性肝病和非酒精性脂肪
THZ531
(Catalog# : 184172, Cas# :
1702809-17-3
)
THZ531是一种共价CDK12和CDK13共价抑制剂。环素依赖性激酶12和13 (CDK
托格列净
(Catalog# : 184311, Cas# :
903565-83-3
)
托格列净,也称为CSG452,是一种高效、高选择性的SGLT2抑制剂,在
TPX-0005
(Catalog# : 18423, Cas# :
1802220-02-5
)
TPX-0005是一种Src/FAK/Janus激酶2 (JAK2)抑制剂。TPX-0005 + EGFR TKI抑制RTKs
tert-butyl ((1H-benzo[d][1,2,3]triazol-1-yl)methyl)carbamate
(Catalog# : 183214, Cas# :
305860-41-7
)
tert-butyl (1H-benzo[d][1,2,3]triazol-1-yl)methylcarbamate is a drug intermediate.
Timapiprant
(Catalog# : 1712152, Cas# :
851723-84-7
)
Timapiprant, also known as OC000459, is a potent, selective and orally active CRTH2 a
TUG-770
(Catalog# : 1791519, Cas# :
1402601-82-4
)
TUG-770是高度有效的游离脂肪酸受体1(FFA1/GPR40)治疗2型糖尿病的激动
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).