武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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Aldehydes
Amines
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Boronic Acids
Bromides
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Indoles and Oxindoles
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
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定制合成
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订购信息
联系我们
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产品名字索引 S
S63845
(Catalog# : 171071, Cas# :
1799633-27-4
)
s63845是专门结合MCL1的BH3结合槽高亲和力的小分子。s63845有效杀死
Salermide
(Catalog# : 1791511, Cas# :
1105698-15-4
)
salermide是一个强大的肿瘤特异性凋亡的影响长寿基因蛋白质抑制剂
SD-06
(Catalog# : 1791320, Cas# :
271576-80-8
)
SD-06是治疗关节炎的MAPK p38α抑制剂。
Sulfatinib
(Catalog# : 179135, Cas# :
1308672-74-3
)
Sulfatinib是一种口服的血管内皮生长因子受体(VEGFR)1, 2,3,和成
S107 HCl
(Catalog# : 1791111, Cas# :
927871-76-9
)
S107是类型1 利阿诺定受体(RYR1)稳定剂;结合 RyR1提高calstabin-1亲
司美利特盐酸盐
(Catalog# : 179830, Cas# :
101526-62-9
)
司美利特,也称为CK-1752,是III类抗心律失常药。它是一种选择性
SNX-2112
(Catalog# : 179815, Cas# :
908112-43-6
)
SNX-2112,又称为PF 04928473,是一种HSP90抑制剂,目前正在进行1期临
SU-1498
(Catalog# : 17984, Cas# :
168835-82-3
)
SU-1498是一种选择性的受体酪氨酸激酶抑制剂,血管内皮生长因子
SF2523
(Catalog# : 17918, Cas# :
1174428-47-7
)
SF2523是一种高效、选择行的日常pan-PI3K/BRD4抑制剂。具有明显的选
SAR-20347
(Catalog# : 1781101, Cas# :
1450881-55-6
)
SAR-20347是一种强力JAK1和酪氨酸激酶2的双抑制剂 (TYK2).
SB756050
(Catalog# : 20178811, Cas# :
447410-57-3
)
SB-756050是一种G蛋白结合胆汁酸受体1(GPBAR1)激动剂,可能用于治疗
SAR-405
(Catalog# : 2017882, Cas# :
1523406-39-4
)
SAR-405是一种有效且选择性的PIK3C3/Vps34抑制剂,防止自噬和协同MTO
雷帕霉素(钠盐)
(Catalog# : 20177313, Cas# :
148554-65-8
)
雷帕霉素是第一个体内open-ring代谢物,不影响mTOR的雷帕霉素抑制Ch
SU5402
(Catalog# : 174191, Cas# :
215543-92-3
)
SU5402是一种成纤维细胞生长因子受体(FGFR)特异性酪氨酸激酶抑
SAR-020106
(Catalog# : 17031004, Cas# :
1184843-57-9
)
SAR-020106是一种 ATP -竞争性、强效和选择性的CHK1抑制剂,其IC50为1
SH5-07
(Catalog# : 17031002, Cas# :
1456632-41-9
)
SH5-07是一种健壮的氧肟抗酸的STAT3抑制剂,它能在体外诱导抗肿瘤
SUN11602
(Catalog# : 17030603, Cas# :
704869-38-5
)
SUN11602是一种新型的苯胺类化合物,它模仿了碱性成纤维细胞生长
Sardomozide HCl
(Catalog# : 17030306, Cas# :
138794-73-7
)
Sardomozide,又名SAM486A或CGP48664,是第二代多胺合成抑制剂,它抑制
钠盐沙库必曲
(Catalog# : 17030108, Cas# :
149690-05-1
)
沙库必曲,也被称为AHU377,是血管紧张素受体神经内肽酶抑制剂被
SHP099游离
(Catalog# : 17030107, Cas# :
1801747-42-1
)
<SHP099是强有力的,选择性,具有口服生物利用率,是一种IC50 = 0.07μM的
司马西特
(Catalog# : 17022802, Cas# :
425386-60-3
)
司马西特(LY450139) 是一种针对Aβ42的γ-分泌酶阻断剂, Aβ40和Aβ38的
泰地唑胺杂质 A
(Catalog# : 17021402, Cas# :
1431699-67-0
)
泰地唑胺杂质 A是磷酸四唑磷酸酯活跃的一部分,对革兰氏阳性菌
STO-609
(Catalog# : 17021319, Cas# :
52029-86-4
)
STO-609是一个特定抑制剂。
S49076
(Catalog# : 17021309, Cas# :
1265965-22-7
)
S49076是一种新型的、能有效抑制IC50值低于20 nmol/ L的MET、AXL / MER和
SRT2183
(Catalog# : 17021306, Cas# :
1001908-89-9
)
SRT2183是sirtuin子型SIRT1的小分子激活剂,目前由Sirtris制药公司开发
SW044248
(Catalog# : 17011714, Cas# :
522650-83-5
)
SW044248是一个强有力的和选择性拓扑异构酶抑制剂。SW044248杀死大
舒更葡糖钠
(Catalog# : 17011713, Cas# :
343306-79-6
)
舒更葡糖钠是治疗神经肌肉阻滞的药物。
链脲菌素
(Catalog# : 17011712, Cas# :
18883-66-4
)
链脲菌素是一种从链球菌中分离出来的甲基亚硝基脲类抗肿瘤抗生
Sotagliflozin
(Catalog# : 17011711, Cas# :
1018899-04-1
)
Sotagliflozin,也称为LX4211,是一种口服活性和双SGLT1 / SGLT2抑制剂,在
索利霉素
(Catalog# : 17011710, Cas# :
760981-83-7
)
索利霉素,也称为CEM-101和OP-1068, 是一种用于治疗社区获得性肺炎(C
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-