武汉永璨生物科技有限公司
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
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Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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产品名字索引 S
Saridegib
(Catalog# : 1812251, Cas# :
1037210-93-7
)
Saridegib,又称IPI-926,是一种口服生物利用的环帕胺衍生物,是Hed
SAR260301
(Catalog# : 1812134, Cas# :
1260612-13-2
)
SAR260301是强有力的和选择性组 I 磷脂酰肌醇-3-激酶(PI3K)β特定抑制
Sparsentan
(Catalog# : 1812132, Cas# :
254740-64-2
)
Sparsentan, 也称为RE-021, PS433540和DARA-a,是一种日常血管紧张素II和内
SR-0987
(Catalog# : 1810263, Cas# :
303126-97-8
)
SR-0987是一个T细胞-特异性RORγ(RORγt)受体激动剂。SR-0987诱导IL-17的
SGC-CBP30
(Catalog# : 1810244, Cas# :
1613695-14-9
)
SGC-CBP30是CREBBP (CBP)和EP300的有效选择性抑制剂;它们是一般的转录共
ST2825
(Catalog# : 1810243, Cas# :
894787-30-5
)
ST-2825是MyD88抑制剂。ST2825在小鼠实验性外伤性脑损伤后提供神经保
Seletalisib
(Catalog# : 1810221, Cas# :
1362850-20-1
)
Seletalisib,也被称为UCB-5857,是一种有效的选择性PI3激酶抑制剂,
Simenepag
(Catalog# : 1810172, Cas# :
910562-15-1
)
Simenepag,又名AGN-210676,是一种用于治疗青光眼和高眼压的小分子
SB-273005
(Catalog# : 186221, Cas# :
205678-31-5
)
SB-273005是一种整合素αvβ3的抑制剂。
STF-083010
(Catalog# : 185151, Cas# :
307543-71-1
)
STF-083010,也称为IRE1抑制剂I, 是IRE1/XBP1通路的抑制剂。
SAR407899游离
(Catalog# : 185115, Cas# :
923359-38-0
)
SAR407899是一种有效且具有选择性的、前景的抗高血压活性Rho激酶抑
SB-334867游离
(Catalog# : 185114, Cas# :
792173-99-0
)
SB-334867是一种阿立新拮抗剂。
SC-560
(Catalog# : 185113, Cas# :
188817-13-2
)
SC-560是一种有效的具有口服活性和选择性的COX-1抑制剂。
Seladelpar
(Catalog# : 185112, Cas# :
851528-79-5
)
Seladelpar,也被称为MBX-8025和RWJ-800025,是一种选择性的过氧化物酶
SEL120-34A盐酸盐
(Catalog# : 18574, Cas# :
1609452-30-3
)
SEL120-34A是一种高效、选择性的CDK8抑制剂,活跃于AML细胞中,具有
SR-4370
(Catalog# : 1842814, Cas# :
1816294-67-3
)
SR-4370是一种HDAC抑制剂。
SGC2085盐酸盐
(Catalog# : 184287, Cas# :
1821908-49-9
)
SGC2085是一种强效的选择性共激活剂,它可以使精氨酸甲基转移酶
S38093盐酸盐
(Catalog# : 184176, Cas# :
1222097-72-4
)
S38093是组胺H3受体的反向激动剂。
STO-609醋酸盐
(Catalog# : 184123, Cas# :
1173022-21-3
)
STO-609是一种细胞渗透性抑制剂,钙/钙调蛋白依赖性激酶激酶(CaMK
Super-TDU
(Catalog# : 18495, Cas# :
1599441-71-0
)
Super-TDU是靶向YAP-TEADs interaction的抑制性多肽。
SSD114 HCl
(Catalog# : 18427, Cas# :
N/A
)
SSD114是一种GABAB阳性变构调制器。SSD114增强gaba刺激[35S]GTP S与本地
(S)-(4-(3-(tert-butoxycarbonyl)-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)phenyl)methyl 2,4-dimethylbenzoate
(Catalog# : 183219, Cas# :
1253955-19-9
)
(S)-(4-(3-(tert-butoxycarbonyl)-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)phenyl)met
(S)-3-(tert-butoxycarbonyl)-2-(4-((2,4-dimethylbenzoyloxy)methyl)phenyl)propanoic acid
(Catalog# : 183218, Cas# :
2097334-20-6
)
(S)-3-(tert-butoxycarbonyl)-2-(4-((2,4-dimethylbenzoyloxy)methyl)phenyl)propanoic aci
(S)-2-羟基丁酸正丁酯
(Catalog# : 1712291, Cas# :
132513-51-0
)
(S)-2-羟基丁酸正丁酯是一种分子砌块。
SCR7 pyrazine
(Catalog# : 1712261, Cas# :
14892-97-8
)
SCR7吡嗪是DNA连接酶IV的小分子抑制剂,防止非同源端连接通过干扰
S38093
(Catalog# : 17101615, Cas# :
862896-30-8
)
S 38093 是一种大脑渗透的 H3 receptor 拮抗剂,对大鼠,小鼠和人的
SAR-7334盐酸
(Catalog# : 17101610, Cas# :
1333207-63-8
)
SAR-7334是一种新颖的、高效的、生物可利用的TRPC6通道,打开了新
SEN-826
(Catalog# : 1710168, Cas# :
1160833-51-1
)
SEN-826是一种潜在抗癌剂。
SRT3025 HCl
(Catalog# : 17101310, Cas# :
2070015-26-6
)
SRT3025是一种可口服的小分子激活SIRT1酶。
Senexin A
(Catalog# : 1710136, Cas# :
1366002-50-7
)
Senexin A是一种强效的选择性与抑制剂(IC50 = 280 nm)。Senexin A结合
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
AZD0095
(Catalog# : 237072, Cas# :
2750001-23-9
)
AZD0095 is a Selective Inhibitor of Monocarboxylate Transporter 4 (MCT4) for Oncology.
2-MNG
(Catalog# : 24129, Cas# :
2101538-28-5
)
2-巯基烟酰甘氨酸是一种新型强效黑素生成抑制剂,具有独特的作
MAT2A-IN-9
(Catalog# : 25147, Cas# :
2439277-80-0
)
MAT2A-IN-9(化合物167)是一种2-氧代喹唑啉衍生物,是一种强效的M
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
Atebimetinib
(Catalog# : 25148, Cas# :
2669009-92-9
)
阿替美替尼(IMM-1-104)是一种口服的小分子MEK1和MEK2激酶变构抑制
Acoramidis hydrochloride
(Catalog# : 24068, Cas# :
2242751-53-5
)
Acoramidis是一种口服、强效、高选择性小分子转甲状腺素蛋白(TTR
Crelosidenib
(Catalog# : 24101, Cas# :
2230263-60-0
)
Crelosidenib ( [LY3410738)是一种有效的选择性的具有口服活性的突变
LOXO-435
(Catalog# : 25080, Cas# :
2833703-74-3
)
LOXO-435是FGFR3的选择性小分子抑制剂。它对野生型和致癌激活的FGF
Gridegalutamide
(Catalog# : 25138, Cas# :
2446928-30-7
)
Gridegalutamide, also known as BMS-986365 and CC-94676, is a heterobifunctional, firs
Chiauranib
(Catalog# : 25146, Cas# :
1256349-48-0
)
Chiauranib also known as orally available, small molecule inhibitor of select serine-