武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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产品名字索引 D
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产品名字索引 D
1,4-DPCA
(Catalog# : 204608, Cas# :
331830-20-7
)
1,4-DPCA is a potent and selective inhibitor of prolyl 4-hydroxylase.
Daprodustat (Synonyms: GSK1278863)
(Catalog# : 112596, Cas# :
960539-70-2
)
Daprodustat (Synonyms: GSK1278863) is an orally active hypoxia-inducible factor proly
Darapladib
(Catalog# : 193202, Cas# :
356057-34-6
)
Darapladib,也被称为SB-480848,是一种可逆的脂蛋白相关磷脂酶A2 (Lp
D-609
(Catalog# : 19371, Cas# :
83373-60-8
)
D-609,又称D-609 free,是一种潜在的用于胰腺癌治疗的磷脂酶C抑制
Degarelix acetate
(Catalog# : 192262, Cas# :
934246-14-7
)
Degarelix, 也称为FE-200486和ASP-3550,是一种具有促性腺激素释放激素
DCC-2618 ( Ripretinib )
(Catalog# : 1811121, Cas# :
1442472-39-0
)
Ripretinib,又名DCC-2618,是一种有效的、口服活性和选择性KIT/PDGFR抑
Derazantinib
(Catalog# : 189273, Cas# :
1234356-69-4
)
Derazantinib又名ARQ-087,是一种口服生物有效的成纤维细胞生长因子
D-Lin-MC3-DMA
(Catalog# : 18942, Cas# :
1224606-06-7
)
D-Lin-MC3-DMA是为脂质纳米颗粒(LNPs)传递siRNA而合成的最有效的阳离子
Dipraglurant
(Catalog# : 187131, Cas# :
872363-17-2
)
Dipraglurant,也被称为ADX-48621,是mGlu5受体的负变构调制器,该受体
Daun02
(Catalog# : 18793, Cas# :
290304-24-4
)
Daun02是一种细胞生存能力抑制剂和DNA分析抑制剂,IC50值分别为1.5
dBET1
(Catalog# : 186261, Cas# :
1799711-21-9
)
dBET1是BET bromodomains的竞争性拮抗剂,其目的是劫持Cereblon E3泛素连
2-D08
(Catalog# : 186231, Cas# :
144707-18-6
)
2-D08是一种合成黄酮类物质,可以抑制类间酰化。2-D08显示抗聚集
柔红霉素
(Catalog# : 186212, Cas# :
20830-81-3
)
柔红霉素通过拓扑异构酶介导与DNA的相互作用来表现细胞毒性,从
DEL-22379
(Catalog# : 186155, Cas# :
181223-80-3
)
DEL-22379是一种有效的选择性二聚反应抑制剂。
德拉沙星
(Catalog# : 18612, Cas# :
189279-58-1
)
德拉沙星,也被称为ABT-492, RX-3341和WQ-3034,是一种非锌离子氟喹诺
Delpazolid
(Catalog# : 18611, Cas# :
1219707-39-7
)
Delpazolid,又称LCB01-0371,是一种新型的环胺唑酮恶唑啉酮。
Desidustat
(Catalog# : 185231, Cas# :
1616690-16-4
)
Desidustat是一种抗贫血药。
多韦替尼乳酸盐
(Catalog# : 18575, Cas# :
915769-50-5
)
多韦替尼,也称为TKI-258或CHIR-258,是一种口服生物药效应的FGFR3抑制
Defensamide
(Catalog# : 184212, Cas# :
1104874-94-3
)
Defensamide, also known as MHP and methyl caprooyl tyrosinate, is an activator of sph
2-(4-(((2,4-dimethylbenzoyl)oxy)methyl)phenyl)acetic acid
(Catalog# : 183215, Cas# :
2097334-16-0
)
2-(4-(((2,4-dimethylbenzoyl)oxy)methyl)phenyl)acetic acid is a drug intermediate.
DCG04
(Catalog# : 179813, Cas# :
314263-42-8
)
DCG04是一种多价配体针对甘露糖-6-磷酸受体中基于活动的探针定位
3,5-Dichloro-N-[(1,1-dimethylethoxy)carbonyl]-L-tyrosine methyl ester
(Catalog# : 178222, Cas# :
261926-09-4
)
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2,6-二溴苄腈
(Catalog# : 1781502, Cas# :
67197-53-9
)
2-(2,6-dibroMophenyl)acetonitrile 是有机合成反应中的一个重要合成砌块
达鲁舍替
(Catalog# : 1781107, Cas# :
827318-97-8
)
达鲁舍替,也称为PHA-739358,是一种小分子3 -氨基吡唑衍生物,具
6-(4,5-dihydro-1H-imidazol-2-yl)-2-methoxy-3-[3-(morpholin-4-yl)propoxy]aniline
(Catalog# : 2017080116, Cas# :
1032571-01-9
)
6-(4,5-dihydro-1H-imidazol-2-yl)-2-methoxy-3-(3-morpholin-4-ylpropoxy)aniline
多巴酚丁胺盐酸盐
(Catalog# : 17030803, Cas# :
49745-95-1
)
多巴酚丁胺是一种交感神经药物,用于治疗心力衰竭和心源性休克
Defactinib
(Catalog# : 120111, Cas# :
1073154-85-4
)
Defactinib是一种有效的FAK磷酸化抑制剂;通过依赖AKT的途径克服抵抗
环酯红霉素
(Catalog# : 17030310, Cas# :
55224-05-0
)
环酯红霉素, 又称红霉素环碳酸盐,是一种由链霉素产生的抑菌抗
丹参素
(Catalog# : 17021315, Cas# :
76822-21-4
)
丹参素,一种中药制剂,具有潜在的抗肿瘤和抗血管生成作用。
2,3-dimethyl-2,5-cyclohexadiene-1,4 dione
(Catalog# : 17011908, Cas# :
526-86-3
)
2,5-Cyclohexadiene-1,4-dione,2,3-dimethyl-
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
HC-7366
(Catalog# : 25076, Cas# :
2803470-63-3
)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
Flavopiridol ( 夫拉平度 )
(Catalog# : 237071, Cas# :
146426-40-6
)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
AG-270
(Catalog# : 25176, Cas# :
2201056-66-6
)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分
AZD-5904
(Catalog# : 181121, Cas# :
618913-30-7
)
AZD5904是一个有效的口服生物利用率MPO抑制剂。在临床前研究中,AZ
ALT-007
(Catalog# : 25157, Cas# :
2035010-37-6
)
ALT-007 是一种口服生物可利用的 SPT 抑制剂,比多球菌素更有效,