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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
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MAPK
Membrane Transporter/Ion Channel
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NF-κB
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产品名字索引 D
1,2-dichloro-2-phenyl-3-phthalimidopropane
(Catalog# : 2062007, Cas# :
85278-20-2
)
1,1-Difluorocyclopropane-1-dibenzosuberyl Pyrazinium Bromide
(Catalog# : 2062005, Cas# :
312905-15-0
)
1,4-DPCA
(Catalog# : 204608, Cas# :
331830-20-7
)
1,4-DPCA is a potent and selective inhibitor of prolyl 4-hydroxylase.
Daprodustat (Synonyms: GSK1278863)
(Catalog# : 112596, Cas# :
960539-70-2
)
Daprodustat (Synonyms: GSK1278863) is an orally active hypoxia-inducible factor proly
Darapladib
(Catalog# : 193202, Cas# :
356057-34-6
)
Darapladib,也被称为SB-480848,是一种可逆的脂蛋白相关磷脂酶A2 (Lp
D-609
(Catalog# : 19371, Cas# :
83373-60-8
)
D-609,又称D-609 free,是一种潜在的用于胰腺癌治疗的磷脂酶C抑制
Degarelix acetate
(Catalog# : 192262, Cas# :
934246-14-7
)
Degarelix, 也称为FE-200486和ASP-3550,是一种具有促性腺激素释放激素
DCC-2618 ( Ripretinib )
(Catalog# : 1811121, Cas# :
1442472-39-0
)
Ripretinib,又名DCC-2618,是一种有效的、口服活性和选择性KIT/PDGFR抑
Derazantinib
(Catalog# : 189273, Cas# :
1234356-69-4
)
Derazantinib又名ARQ-087,是一种口服生物有效的成纤维细胞生长因子
D-Lin-MC3-DMA
(Catalog# : 18942, Cas# :
1224606-06-7
)
D-Lin-MC3-DMA是为脂质纳米颗粒(LNPs)传递siRNA而合成的最有效的阳离子
Dipraglurant
(Catalog# : 187131, Cas# :
872363-17-2
)
Dipraglurant,也被称为ADX-48621,是mGlu5受体的负变构调制器,该受体
Daun02
(Catalog# : 18793, Cas# :
290304-24-4
)
Daun02是一种细胞生存能力抑制剂和DNA分析抑制剂,IC50值分别为1.5
dBET1
(Catalog# : 186261, Cas# :
1799711-21-9
)
dBET1是BET bromodomains的竞争性拮抗剂,其目的是劫持Cereblon E3泛素连
2-D08
(Catalog# : 186231, Cas# :
144707-18-6
)
2-D08是一种合成黄酮类物质,可以抑制类间酰化。2-D08显示抗聚集
柔红霉素
(Catalog# : 186212, Cas# :
20830-81-3
)
柔红霉素通过拓扑异构酶介导与DNA的相互作用来表现细胞毒性,从
DEL-22379
(Catalog# : 186155, Cas# :
181223-80-3
)
DEL-22379是一种有效的选择性二聚反应抑制剂。
德拉沙星
(Catalog# : 18612, Cas# :
189279-58-1
)
德拉沙星,也被称为ABT-492, RX-3341和WQ-3034,是一种非锌离子氟喹诺
Delpazolid
(Catalog# : 18611, Cas# :
1219707-39-7
)
Delpazolid,又称LCB01-0371,是一种新型的环胺唑酮恶唑啉酮。
Desidustat
(Catalog# : 185231, Cas# :
1616690-16-4
)
Desidustat是一种抗贫血药。
多韦替尼乳酸盐
(Catalog# : 18575, Cas# :
915769-50-5
)
多韦替尼,也称为TKI-258或CHIR-258,是一种口服生物药效应的FGFR3抑制
Defensamide
(Catalog# : 184212, Cas# :
1104874-94-3
)
Defensamide, also known as MHP and methyl caprooyl tyrosinate, is an activator of sph
2-(4-(((2,4-dimethylbenzoyl)oxy)methyl)phenyl)acetic acid
(Catalog# : 183215, Cas# :
2097334-16-0
)
2-(4-(((2,4-dimethylbenzoyl)oxy)methyl)phenyl)acetic acid is a drug intermediate.
DCG04
(Catalog# : 179813, Cas# :
314263-42-8
)
DCG04是一种多价配体针对甘露糖-6-磷酸受体中基于活动的探针定位
3,5-Dichloro-N-[(1,1-dimethylethoxy)carbonyl]-L-tyrosine methyl ester
(Catalog# : 178222, Cas# :
261926-09-4
)
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2,6-二溴苄腈
(Catalog# : 1781502, Cas# :
67197-53-9
)
2-(2,6-dibroMophenyl)acetonitrile 是有机合成反应中的一个重要合成砌块
达鲁舍替
(Catalog# : 1781107, Cas# :
827318-97-8
)
达鲁舍替,也称为PHA-739358,是一种小分子3 -氨基吡唑衍生物,具
6-(4,5-dihydro-1H-imidazol-2-yl)-2-methoxy-3-[3-(morpholin-4-yl)propoxy]aniline
(Catalog# : 2017080116, Cas# :
1032571-01-9
)
6-(4,5-dihydro-1H-imidazol-2-yl)-2-methoxy-3-(3-morpholin-4-ylpropoxy)aniline
多巴酚丁胺盐酸盐
(Catalog# : 17030803, Cas# :
49745-95-1
)
多巴酚丁胺是一种交感神经药物,用于治疗心力衰竭和心源性休克
Defactinib
(Catalog# : 120111, Cas# :
1073154-85-4
)
Defactinib是一种有效的FAK磷酸化抑制剂;通过依赖AKT的途径克服抵抗
环酯红霉素
(Catalog# : 17030310, Cas# :
55224-05-0
)
环酯红霉素, 又称红霉素环碳酸盐,是一种由链霉素产生的抑菌抗
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制