武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
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定制合成
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订购信息
联系我们
公司简介
联系我们
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产品名字索引 B
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产品名字索引 B
Blonanserin
(Catalog# : 102612, Cas# :
132810-10-7
)
Blonanserin is a D2/5-HT2 receptor antagonist, atypical antipsychotic.
BRD73954
(Catalog# : 102601, Cas# :
1440209-96-0
)
BRD73954 ia a potent and selective HDAC inhibitor with IC50 of 36 nM and 120 nM for H
BIO-32546
(Catalog# : 101916, Cas# :
1548743-66-3
)
Coming soon!
BIO-acetoxime
(Catalog# : 101401, Cas# :
667463-85-6
)
BIO-Acetoxime is a potent and selective GSK-3a/b inhibitor that reduces invasiveness
BIX01294
(Catalog# : 101203, Cas# :
935693-62-2
)
BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 M.
Bardoxolone methyl
(Catalog# : 92303, Cas# :
218600-53-4
)
Bardoxolone methyl (also known as “RTA 402” and “CDDO-methyl ester”) is an or
BMS-626529
(Catalog# : 92207, Cas# :
701213-36-7
)
BMS-626529 is a potent HIV-1 attachment inhibitor, which is also the phosphonooxymeth
2-Bromo-3-Fluoro-6-Picoline
(Catalog# : 92202, Cas# :
374633-36-0
)
Coming soon!
6-benzyloxy-benzofuran
(Catalog# : 91831, Cas# :
320350-81-0
)
Coming soon!
2-Bromopyridine-5-carbaldehyde
(Catalog# : 91822, Cas# :
149806-06-4
)
Coming soon!
5-bromo-4-chloro-3-nitro-1Hpyrrolo[2,3-b]pyridine
(Catalog# : 91821, Cas# :
1477532-48-1
)
Coming soon!
1-(4-(benzyloxy)-6-methoxybenzofuran-2-yl)-2-bromoethanone
(Catalog# : 91820, Cas# :
1476847-52-5
)
Coming soon!
2-(benzyloxy)-6-hydroxy-4-methoxybenzaldehyde
(Catalog# : 91819, Cas# :
1476847-50-3
)
Coming soon!
8-bromo-1-((S)-2-methoxypropyl)-1H-imidazo[4,5-c]quinolin-2(3H)-one
(Catalog# : 91812, Cas# :
1369532-69-3
)
Coming soon!
6-Bromo-4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole
(Catalog# : 91804, Cas# :
1231930-33-8
)
Coming soon!
1-(1-benzothiophen-4-yl)piperazine
(Catalog# : 91704, Cas# :
846038-18-4
)
Coming soon!
4-(1,2-Benzothiazol-3-yl)-1-[(3aR,7aR)-octahydro-2H-isoindol-2-yl ]piperazin-1-ium-1-sulfonate
(Catalog# : 91410, Cas# :
186204-37-5
)
The related APILurasidone hydrochlorideThe related intermediates3-Piperazinobenzisoth
Benzenemethanamine, 3,5-difluoro-α-methyl-, (alphaS)- (9CI)
(Catalog# : 91121, Cas# :
444643-16-7
)
Coming soon!
Benzenemethanamine, 3,4-difluoro-α-methyl-, (alphaS)- (9CI)
(Catalog# : 91130, Cas# :
321318-17-6
)
Coming soon!
3-(2-Bromo-4-fluorophenyl)propionic acid
(Catalog# : 90710, Cas# :
174603-55-5
)
Coming soon!
3-(3-Bromophenyl)propionic acid
(Catalog# : 90707, Cas# :
42287-90-1
)
Coming soon!
3-(2-Bromophenyl)propionic acid
(Catalog# : 90706, Cas# :
15115-58-9
)
Coming soon!
1-Boc-2-Butylpiperazine hydrochloride
(Catalog# : 90109, Cas# :
1179359-55-7
)
Coming soon!
Benzyl 2-(aminomethyl)pyrrolidine-1-carboxylate hydrochloride
(Catalog# : 90107, Cas# :
119020-00-7
)
Coming soon!
Benzyl 4-(3-((tert-butoxycarbonyl)amino)azetidin-1-yl)piperidine-1-carboxylate
(Catalog# : 83125, Cas# :
883546-87-0
)
Coming soon!
1-Boc-3-azetidinemethanol
(Catalog# : 83123, Cas# :
142253-56-3
)
Coming soon!
1-Boc-3-hydroxyazetidine
(Catalog# : 83114, Cas# :
141699-55-0
)
Coming soon!
1-Boc-3-Azetidine-3-carboxylic acid
(Catalog# : 83113, Cas# :
142253-55-2
)
Coming soon!
1-benzothien-2-yl(5-bromo-2-fluorophenyl)methanol
(Catalog# : 82728, Cas# :
1034305-11-7
)
Coming soon!
5-Bromo-2-chloro-N-cyclopentylpyrimidin-4-amine
(Catalog# : 82724, Cas# :
179688-53-0
)
Coming soon!
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Opakalim
(Catalog# : 25193, Cas# :
2376397-93-0
)
Opakalim(BHV-7000)是Kv7.2/7.3钾通道(KCNQ2/3)的口服小分子激活剂,
DS68591889
(Catalog# : 25158, Cas# :
2488609-21-6
)
DS68591889 (PTDSS1i) 特异性抑制 PTDSS1,而 PTDSS1 可催化丝氨酸掺入 PC。
CAY 10566
(Catalog# : 10403, Cas# :
944808-88-2
)
CAY 10566是一种强效的选择性SCD-1抑制剂。
Cadefrecitinib (GLPG-3667)
(Catalog# : 20509, Cas# :
2308520-97-8
)
Cadefrecitinib(GLPG-3667)是一种口服小分子TYK2激酶抑制剂,目前正处
QBS10072S
(Catalog# : 25190, Cas# :
1802735-28-9
)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
Dencatistat (STP938)
(Catalog# : 25177, Cas# :
2377000-84-3
)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
DS-1001b
(Catalog# : 25178, Cas# :
1898207-64-1
)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
Z57346765
(Catalog# : 25191, Cas# :
1016340-64-9
)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
CBR-470-1
(Catalog# : 25192, Cas# :
2416095-06-0
)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
Safusidenib
(Catalog# : 25149, Cas# :
1898206-17-1
)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(