武汉永璨生物科技有限公司
+86-17702719238
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抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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中间体
技术服务
定制合成
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订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
Vitamin D Related
Membrane Transporter/Ion Channel
others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
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定制合成
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订购信息
联系我们
公司简介
联系我们
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产品名字索引 B
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产品名字索引 B
BMS-1001
(Catalog# : 2062901, Cas# :
2113650-03-4
)
6-bromo-2-ethyl-8-methylimidazo[1,2-a]pyridin-3-amine
(Catalog# : 2062328, Cas# :
1549360-60-2
)
6-bromo-2-ethyl-8-methylimidazo[1,2-a]pyridin-3-amine hydrochloride
(Catalog# : 202327, Cas# :
1628263-43-3
)
4-bromo-2-fluoro-1-propan-2-yloxybenzene
(Catalog# : 2062316, Cas# :
202865-80-3
)
1-bromo-4-propan-2-ylsulfonylbenzene
(Catalog# : 2062315, Cas# :
70399-02-9
)
5-(2,4-bis(benzyloxy)-5-isopropylphenyl)-N-ethyl-4-iodoisoxazole-3-carboxamide
(Catalog# : 2062305, Cas# :
741414-22-8
)
7-bromo-2-(1-methyl-1H-pyrazol-4-yl)-quinoxaline
(Catalog# : 2062028, Cas# :
1083325-87-4
)
(3-bromoprop-1-en-2-yl)benzene
(Catalog# : 2062001, Cas# :
3360-54-1
)
BW-A 78U
(Catalog# : 2051512, Cas# :
101155-02-6
)
BW-A 78U is a PDE4 inhibitor with an IC50 of 3 μM.
9-溴-2-羟基-7-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮
(Catalog# : S-204156, Cas# :
663619-90-7
)
BB-Cl-Amidine
(Catalog# : 204505, Cas# :
1802637-39-3
)
BB-Cl-A是一种通过激活内质网应激途径治疗犬和猫乳腺癌的新型疗
BAY-218
(Catalog# : 204301, Cas# :
2162982-11-6
)
BAY-218, also known as BAY-2335218, is a potent and selective small-molecule AhR inhi
Blarcamesine ( AVex-73 ; AE-37 )
(Catalog# : 6111902, Cas# :
195615-83-9
)
ANAVEX2-73 (blacamesine) 是一种 Sigma-1 受体激动剂和毒蕈碱受体调节剂
(6bR,10aS)-3-methyl-2,3,6b,7,8,9,10,10a-octahydro-1H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxaline
(Catalog# : ITI007_3, Cas# :
313368-85-3
)
(6bR,10aS)-2-oxo-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxaline-8-carboxylic acid ethyl ester
(Catalog# : ITI007_2, Cas# :
313369-16-3
)
Sun-shine Chemical is a supplier Lumateperone and its intermediate from 100g scale to
6-bromo-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride
(Catalog# : ITI007_1, Cas# :
1059630-11-3
)
Sun-shine Chemical is a supplier ofLumateperone, we may provideLumateperone and its i
3-bromo-7-nitro-1-tosyl-1H-indole
(Catalog# : 511191, Cas# :
2091135-02-1
)
BMS-986104
(Catalog# : 193285, Cas# :
1622180-31-7
)
BMS-986104是一种强效的选择性S1P1受体调节剂,具有配体偏倚信号转
BAY-1316957
(Catalog# : 193263, Cas# :
1613264-40-6
)
BAY-1316957是一种高效、选择性、口服的人前列腺素E2受体亚型4 (hEP
BMS-986158
(Catalog# : 193255, Cas# :
1800340-40-2
)
BMS-986158是一种有效的选择性BET抑制剂。BMS-986158与BET蛋白BRD中的乙
BMS-986163
(Catalog# : 193207, Cas# :
1801151-09-6
)
BMS-986163是GluN2B的负变构调节剂,在重度抑郁症中具有潜在的应用
BAY-293
(Catalog# : 193121, Cas# :
2244904-70-7
)
BAY-293是一种有效的SOS1抑制剂,通过破坏IC50为21 nM的RAS-SOS1的相互
BMS-816336
(Catalog# : 19351, Cas# :
1009583-20-3
)
BMS-816336是一种口服活性、有效和选择性的11β-HSD1抑制剂。BMS- 8163
Belvarafenib
(Catalog# : 19341, Cas# :
1446113-23-0
)
Belvarafenib,又名GDC-5573、HM95573、RG6185,是RAF家族激酶的选择性抑制
Burixafor HBr
(Catalog# : 192221, Cas# :
1191450-19-7
)
Burixafor,又名TG-0054,是CXC趋化因子受体4 (CXCR4)的口服生物利用抑
BMS-986142
(Catalog# : 191284, Cas# :
1643368-58-4
)
BMS-986142是一种高效、选择性、可逆的BTK抑制剂。
Blu667
(Catalog# : 191282, Cas# :
2097132-94-8
)
BLU-667是一种有效的选择性 RET 抑制剂, IC50 为0.4 nM,对突变体 RET
BAY1238097
(Catalog# : 191257, Cas# :
1564268-08-1
)
BAY1238097是一种有效的选择性BET抑制剂。BAY1238097与BET蛋白BRD上乙酰
BMS-189453
(Catalog# : 191253, Cas# :
166977-43-1
)
BMS-189453也被称为BMS453,是一个强有力的和选择性RARβ受体激动剂和
BI-671800
(Catalog# : 191213, Cas# :
1093108-50-9
)
BI-671800是一种治疗哮喘患者的CRTH2拮抗剂。BI 671800与症状控制单纯
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).