武汉永璨生物科技有限公司
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
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产品名字索引 B
BRD0705
(Catalog# : 202112701, Cas# :
2056261-41-5
)
BRD0705 is a potent, paralog selective and orally active GSK3α inhibitor. BRD0705 ca
BLU-782
(Catalog# : 20121701, Cas# :
2141955-96-4
)
(2S,5R)-5-氨基-2-甲基哌啶-1-甲酸苄酯盐酸盐
(Catalog# : 20103006, Cas# :
1207853-23-3
)
Benpyrine racemate
(Catalog# : 2091907, Cas# :
1333714-43-4
)
(Rac)-Benpyrine is a racemate of Benpyrine. (Rac)-Benpyrine is a potent and orally ac
BAY-2416964
(Catalog# : 2091906, Cas# :
2242464-44-2
)
BAY-2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist
BI-894999
(Catalog# : 2091902, Cas# :
1660117-38-3
)
BI-894999 is a potent and selective BET inhibitor potentially useful for the Treatmen
4-溴-(2-丁氧基乙氧基)苯
(Catalog# : 2091206, Cas# :
39255-24-8
)
4-(2-丁氧基乙氧基)苯基硼酸
(Catalog# : 2091203, Cas# :
279262-28-1
)
6-BROMO-2-ETHYL-N,8-DIMETHYLIMIDAZO[1,2-A]PYRIDIN-3-AMINE
(Catalog# : 2091201, Cas# :
1628264-07-2
)
BCH001
(Catalog# : 208192, Cas# :
384859-58-9
)
BCH001是一种特异性PAPD5抑制剂,可在DC患者诱导的多能干细胞中恢
BMS-1166
(Catalog# : 2073102, Cas# :
1818314-88-3
)
BMS-1166是一种有效的PD-1 / PD-L1相互作用抑制剂,IC50为1.4 nM,可拮抗
BAY-1816032
(Catalog# : 2071615, Cas# :
1891087-61-8
)
BAY-1816032 is a potent and oral available BUB1 (budding uninhibited by benzimidazole
BAY-2402234
(Catalog# : 2071553, Cas# :
2225819-06-5
)
BAY-2402234 is a potent and selective dihydroorotate dehydrogenase (DHODH) inhibitor
BMVC-8C3O
(Catalog# : 2071550, Cas# :
1301708-12-2
)
BMVC-8C3O is a DNA G-quadruplexe (G4) ligand which can induce topological conversion
BAY-545
(Catalog# : 2071532, Cas# :
1699717-32-2
)
BAY-545 is a potent and selective antagonist of the A2B adenosine receptor.
Belnacasan
(Catalog# : 52004, Cas# :
273404-37-8
)
Belnacasan (VX-765) 是 VRT-043198 的口服生物活性前药,VRT-043198 是有效
BMS-1001
(Catalog# : 2062901, Cas# :
2113650-03-4
)
6-bromo-2-ethyl-8-methylimidazo[1,2-a]pyridin-3-amine
(Catalog# : 2062328, Cas# :
1549360-60-2
)
6-bromo-2-ethyl-8-methylimidazo[1,2-a]pyridin-3-amine hydrochloride
(Catalog# : 202327, Cas# :
1628263-43-3
)
4-bromo-2-fluoro-1-propan-2-yloxybenzene
(Catalog# : 2062316, Cas# :
202865-80-3
)
1-bromo-4-propan-2-ylsulfonylbenzene
(Catalog# : 2062315, Cas# :
70399-02-9
)
5-(2,4-bis(benzyloxy)-5-isopropylphenyl)-N-ethyl-4-iodoisoxazole-3-carboxamide
(Catalog# : 2062305, Cas# :
741414-22-8
)
7-bromo-2-(1-methyl-1H-pyrazol-4-yl)-quinoxaline
(Catalog# : 2062028, Cas# :
1083325-87-4
)
(3-bromoprop-1-en-2-yl)benzene
(Catalog# : 2062001, Cas# :
3360-54-1
)
BW-A 78U
(Catalog# : 2051512, Cas# :
101155-02-6
)
BW-A 78U is a PDE4 inhibitor with an IC50 of 3 μM.
9-溴-2-羟基-7-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮
(Catalog# : S-204156, Cas# :
663619-90-7
)
BB-Cl-Amidine
(Catalog# : 204505, Cas# :
1802637-39-3
)
BB-Cl-A是一种通过激活内质网应激途径治疗犬和猫乳腺癌的新型疗
BAY-218
(Catalog# : 204301, Cas# :
2162982-11-6
)
BAY-218, also known as BAY-2335218, is a potent and selective small-molecule AhR inhi
Blarcamesine ( AVex-73 ; AE-37 )
(Catalog# : 6111902, Cas# :
195615-83-9
)
ANAVEX2-73 (blacamesine) 是一种 Sigma-1 受体激动剂和毒蕈碱受体调节剂
(6bR,10aS)-2-oxo-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxaline-8-carboxylic acid ethyl ester
(Catalog# : ITI007_2, Cas# :
313369-16-3
)
Sun-shine Chemical is a supplier Lumateperone and its intermediate from 100g scale to
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
KL1333
(Catalog# : 25201, Cas# :
1800405-30-4
)
KL1333是一种口服的小有机分子,与NAD(P)H:醌氧化还原酶1(NQO1)
Palupiprant ( E7046 )
(Catalog# : 24055, Cas# :
1369489-71-3
)
E7046 is a potent and selective antagonist of the type 4 prostaglandin E2 (PGE2) rece
Oveporexton ( TAK-861 )
(Catalog# : 25194, Cas# :
2460722-04-5
)
Oveporexton是一种口服小分子选择性食欲素2型受体(OX2R)激动剂。
VT-3989
(Catalog# : 25200, Cas# :
2506273-81-8
)
VT3989是一种首创的强效口服TEAD棕榈酰化抑制剂,可阻断YAP转录活
JX06
(Catalog# : 25199, Cas# :
729-46-4
)
JX06 是一种有效的,选择性的,共价的 PDK 抑制剂。
Bezuclastinib
(Catalog# : 25198, Cas# :
1616385-51-3
)
Bezuclastinib是KIT D816V突变体以及其他KIT外显子17突变体激酶活性的口
Bexobrutideg ( NX-5948 )
(Catalog# : 25197, Cas# :
2649400-34-8
)
Bexobrutideg(NX-5948)是一种BTK降解剂。
Rosolutamide ( AJ-201 ; ASC-JM17 )
(Catalog# : 25196, Cas# :
1039760-91-2 , 2074613-88-8 [ALTERNATIVE]
)
Rosolutamide (formerly known as AJ-201, ASC-JM-17 or ALZ-002) 是一种姜黄素类似
Soclenicant (BNC-210 ; IW-2143)
(Catalog# : 25195, Cas# :
1020634-41-6
)
Soclenicant (BNC-210;IW-2143)是一种新型的α7烟碱型乙酰胆碱受体负
Umbralisib
(Catalog# : 25085, Cas# :
1532533-67-7
)
Umbralisib, also known as TGR1202 and RP5264 , is a highly specific, orally available