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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
PI3K/Akt/mTOR
Epigenetics
Protein Tyrosine Kinase
Angiogenesis
Apoptosis
Autophagy
JAK/STAT
MAPK
Cytoskeletal Signaling
Cell Cycle
TGF-beta/Smad
DNA Damage
Stem Cells & Wnt
Ubiquitin
Neuronal Signaling
NF-κB
GPCR & G Protein
Metabolism
Anti-infection
Proteases
Immunology & Inflammation
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others
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产品名字索引 B
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产品名字索引 B
BI-3812
(Catalog# : 19124, Cas# :
2166387-64-8
)
BI-3812是BCL6 BTB/POZ区域与多个共抑制因子相互作用的有效抑制剂。
BAY 678
(Catalog# : 1812286, Cas# :
675103-36-3
)
BAY 678是一种有效且具有选择性的人类中性粒细胞弹性蛋白酶(HNE)抑
BN-82002
(Catalog# : 1812261, Cas# :
396073-89-5
)
BN-82002又称CDC25磷酸酶抑制剂I,是一种具有抗肿瘤特性的细胞渗透
BMS-509744
(Catalog# : 1811291, Cas# :
439575-02-7
)
BMS-509744是一种有效的白介素-2诱导T细胞激酶(ITK)抑制剂(IC50 = 19 nM
BMS-688521
(Catalog# : 1811281, Cas# :
893397-44-9
)
BMS-688521是白细胞功能相关抗原-1 (LFA-1)的小分子拮抗剂。它为LFA-1
BMS-986195
(Catalog# : 1811264, Cas# :
1912445-55-6
)
BMS-986195是一种有效,共价,Bruton’s酪氨酸激酶的不可逆抑制剂(B
BAY-299
(Catalog# : 1811262, Cas# :
2080306-23-4
)
BAY-299是一种有效且具有选择性的BRD1和TAF1抑制剂(IC50的值分别为
BMS-986165
(Catalog# : 1810163, Cas# :
1609392-27-9
)
BMS-986165是具有选择性、强效、变构抑制剂的酪氨酸激酶2 (Tyk2)。
Bictegravir
(Catalog# : 187181, Cas# :
1611493-60-7
)
Bictegravir,也称为GS - 9883,是一个强有力的,无助推的每日一次HIV- 1整
Basimglurant
(Catalog# : 187121, Cas# :
1034442-21-1
)
Basimglurant,又称RO 4917523和RG-7090,是一种新型的mGlu5阴性变构调制
3BDO
(Catalog# : 186232, Cas# :
890405-51-3
)
3BDO,一种丁基内酯衍生物,可以靶向FKBP1A,激活mTOR信号通路。它
BMS-986205
(Catalog# : 185314, Cas# :
1923833-60-6
)
BMS-986205是一种抗癌药物。
Birinapant
(Catalog# : 185182, Cas# :
1260251-31-7
)
Birinapant,也被称为TL32711,是一种合成的小分子,具有潜在的抗肿
Bryostatin 1
(Catalog# : 18573, Cas# :
83314-01-6
)
苔藓虫素1是一种有效的蛋白激酶C调制器,从苔藓虫体内分离出来
BMS-813160
(Catalog# : 1842812, Cas# :
1286279-29-5
)
BMS-813160是一种有效的选择性CCR2/CCR5拮抗剂,具有潜在的免疫调节
BRD7116
(Catalog# : 184282, Cas# :
329059-55-4
)
BRD7116是白血病干细胞(LSC)活性的有效选择性抑制剂(EC50 = 200 nM)。
盐酸巴多昔芬
(Catalog# : 18496, Cas# :
198480-56-7
)
Bazedoxifene,又名WAY-140424,是第三代选择性雌激素受体调节剂(SERM)
BQR695
(Catalog# : 184218, Cas# :
1513879-21-4
)
BQR695, also known as NVP-BQR695, is a potent and selective PI4K inhibitor.
BAY1143572
(Catalog# : 181242, Cas# :
1414943-88-6
)
Atuveciclib, also known as BAY1143572, is a highly selective, potent and orally avail
BAY-1436032
(Catalog# : 181181, Cas# :
1803274-65-8
)
BAY-1436032是一个强有力的,有选择性的,有效的突变异柠檬酸脱氢酶
BGB-283
(Catalog# : 17101620, Cas# :
1446090-77-2;1446090-79-4
)
BGB-283,也称为Beigene-283或Lifirafenib,是一种新的有效的和选择性的
Belizatinib
(Catalog# : 17101619, Cas# :
1357920-84-3
)
Belizatinib,也称为TSR-011,具有受体酪氨酸激酶间变性淋巴瘤激酶(
Bioymifi
(Catalog# : 1710165, Cas# :
1420071-30-2
)
Bioymifi是DR5的活性剂(Kd = 1.2 µM; IC50 = 2 µM). Bioymifi诱导凋亡的肿瘤
BLU-554
(Catalog# : 1710162, Cas# :
1707289-21-1
)
BLU-554是针对肝癌治疗的成纤维细胞生长因子受体4(FGFR4)抑制剂
BX-517
(Catalog# : 1791314, Cas# :
850717-64-5
)
BX-517,又名PDK1 inhibitor2,是强有力的和有选择性的PDK1抑制剂。
BBT-594
(Catalog# : 179133, Cas# :
882405-89-2
)
BBT594,也称为NVP-BBT594,是强有力的和有选择性的RET和JAK2抑制剂。
BAY41-4109消旋体
(Catalog# : 1791117, Cas# :
298708-79-9
)
Bay41-4109消旋体是对Bay41-4109和S-异构体Bay41-4109 R-异构体的混合物。
BAR-501
(Catalog# : 179821, Cas# :
1632118-69-4
)
BAR-501是一种选择性GPBAR1激动剂,没有任何的FXR激动剂活性。BAR-50
Batefenterol(free base)
(Catalog# : 179820, Cas# :
743461-65-6
)
Batefenterol,也称为 GSK961081和TD-5959,是一种毒蕈碱拮抗剂和β2-受体
BI-847325
(Catalog# : 83101, Cas# :
1207293-36-4
)
BI-847325是一种口服、具有选择性的日常生物MEK/Aurora激酶抑制剂,
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产品分类
信号通路
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Bcr-Abl
----
Src
----
ALK
----
Syk
----
FAK
----
BTK
----
HIF
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Cytoskeletal Signaling
----
Akt
----
Bcr-Abl
----
PKC
----
FAK
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
-- TGF-beta/Smad
----
Bcr-Abl
----
PKC
----
ROCK
----
TGF-beta/Smad
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
α-Synuclein
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Sigma Receptor
----
Ras
----
mAChR
----
Cholecystokinin Receptor
----
Melanocortin Receptor
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
-- Vitamin D Related
----
VD/VDR
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
-- others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
PLX8394
(Catalog# : 20613, Cas# :
1393466-87-9
)
PLX8394 is an orally bioavailable inhibitor of serine/threonine-protein kinase B-raf
Zelasudil
(Catalog# : 24014, Cas# :
2365193-22-0
)
Zelasudil 是一种有效的、高选择性的口服活性抑制剂,针对 Rho 相关
Ziftomenib ( KO-539 )
(Catalog# : 24013, Cas# :
2134675-36-6
)
Ziftomenib 是一种口服、有效、选择性的小分子抑制剂,针对 menin 和
Zunsemetinib
(Catalog# : 24012, Cas# :
1640282-42-3
)
Zunsemetinib是一种在研口服丝裂原活化蛋白激酶活化蛋白激酶2(MK2
Zongertinib ( BI 1810631 )
(Catalog# : 24011, Cas# :
2728667-27-2
)
Zongertinib [BI 1810631] 是一种人表皮生长因子受体 2 (HER2) 抑制剂。
Zasocitinib
(Catalog# : 24010, Cas# :
2272904-53-5
)
Zasocitinib是一种作用于非受体酪氨酸蛋白激酶 (TYK2)靶点的抑制
RNK-05047
(Catalog# : 24008, Cas# :
2503036-46-0
)
RNK-05047 为BRD4降解剂,其在小鼠荷瘤异种移植模型中展现出显著抑
Asengeprast (FT011)
(Catalog# : 24009, Cas# :
1001288-58-9
)
Asengeprast (FT011) 是一种抗纤维化剂,降低胶原蛋白 I 和 III 的 mRNA
ERAS-801 ( JGK-068S )
(Catalog# : 20635, Cas# :
2490431-16-6
)
ERAS-801 ( JGK-068S ) 是一种有效的 EGFR 抑制剂。
T-1095
(Catalog# : 24004, Cas# :
209746-59-8
)
T-1095 is a potent and selective inhibitor of Na+-glucose cotransporters (SGLTs).