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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
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Cas号索引 1
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Cas号索引 1
1609960-30-6 | TH287
(Catalog# : 193135)
TH287是人7,8-二氢-8-草酸鸟苷三磷酸酶MTH1 (NUDT1)的有效抑制剂,IC50
1793059-58-1 | Tinostamustine盐酸盐
(Catalog# : 193112)
Tinostamustine,也称为EDO-S101,是一种烷基化有机去乙酰化酶抑制剂(H
191114-48-4 | Telithromycin
(Catalog# : 19374)
Telithromycin,也被称为HMR-3647和RU-66647,是一种半合成红霉素衍生物
1604810-84-5 | THZ2
(Catalog# : 192252)
THZ2,是THZ1的类似物,具有治疗三阴性乳腺癌(TNBC)的潜力,是一种
1227637-23-1 | Tegatrabetan
(Catalog# : 192145)
Tegatrabetan, 也称为Tegavivint和BC2059,是一种口服生物利用率和有效的
1359993-59-1 | Telratolimod
(Catalog# : 192144)
Telratolimod,也被称为 3M-052或MEDI-9197,是toll样受体7 (TLR-7)和toll样受
1260533-36-5 | TAS-116
(Catalog# : 191286)
TAS- 116是一种对热休克蛋白90 (Hsp90)亚型alpha和beta的有效选择性抑制
106635-81-8 | Tafenoquine succinate ( 他非诺喹琥珀酸盐 )
(Catalog# : 191123)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
106635-80-7 | Tafenoquine ( 他非诺喹 )
(Catalog# : 191122)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
1558021-37-0 | TP0463518
(Catalog# : 1812282)
TP0463518是一种新型高效的HIF脯氨酰羟化酶(PHD)抑制剂。TP0463518竞争
1009816-48-1 | Thiamet G
(Catalog# : 1812133)
Thiamet G是一种有效且具有选择性的O-GlcNAcase抑制剂.
1164462-05-8 | TG4-155
(Catalog# : 181232)
TG4-155 是一种大脑渗透EP2拮抗剂(KB = 2.4nM),在EP4(KB = 11.4µM)小组其他
123948-87-8 | Topotecan
(Catalog# : 1811212)
Topocecan是喜树碱的半合成衍生物,具有抗肿瘤活性。
1448169-71-8 | TAS-120
(Catalog# : 1811191)
TAS-120是成纤维细胞生长因子受体(FGFR)的口服生物有效抑制剂,具
1038984-31-4 | Tulrampator ( CX-1632 )
(Catalog# : 1811161)
Tulrampator,也被称为S-47445和CX-1632,是AMPA受体(AMPAR)的积极变构调制
1226056-71-8 | Thiazovivin
(Catalog# : 1811122)
Thiazovivin是一种具有选择性的,抑制浓度为2µM的ROCK活动的细胞-渗透
1862212-48-3 | TH 1217
(Catalog# : 1811021)
TH 1217是一种有效的dCTP焦磷酸酶1抑制剂。
1137868-52-0 | TAK-960
(Catalog# : 18762)
TAK-960是一种可口服的PLK1抑制剂,具有潜在的抗肿瘤活性。
1353644-70-8 | Theliatinib
(Catalog# : 186235)
Theliatinib又称HMPL-309,是一种新型的小分子、表皮生长因子受体酪
1616493-44-7 | Tucidinostat
(Catalog# : 186233)
Tucidinostat是组蛋白去乙酰化酶(HDAC) 1、2、3和10的一种苯甲酰胺类抑
1111556-37-6 | Takinib
(Catalog# : 18672)
Takinib选择性TAK1抑制剂,TNF-α刺激后细胞凋亡模型,类风湿性关节炎
1314890-29-3 | TMP269
(Catalog# : 185254)
TMP269是一种具有高强度、选择性和可渗透性的IIa型HDAC抑制剂,其
1374743-00-6 | Trilaciclib (G1T28)
(Catalog# : 185235)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
171235-71-5 | TAPI-1
(Catalog# : 185181)
TAPI-1是TACE的抑制剂。它抑制TNF-a、TNFRI(p60)和TNFRII(p80)的裂解。
158899-10-6 | TLN-232
(Catalog# : 18594)
TLN-232, 也称为CAP-232,是一种具有潜在抗肿瘤活性的合成环七肽。
140194-24-7 | 醋酸曲普瑞林
(Catalog# : 18592)
醋酸曲普瑞林是一种促性腺激素释放激素激动剂(GnRH激动剂),用作
1383816-29-2 | Tropifexor
(Catalog# : 18591)
Tropifexor, 也称为LJN452, 是一种用于治疗胆静性肝病和非酒精性脂肪
1702809-17-3 | THZ531
(Catalog# : 184172)
THZ531是一种共价CDK12和CDK13共价抑制剂。环素依赖性激酶12和13 (CDK
1802220-02-5 | TPX-0005
(Catalog# : 18423)
TPX-0005是一种Src/FAK/Janus激酶2 (JAK2)抑制剂。TPX-0005 + EGFR TKI抑制RTKs
1402601-82-4 | TUG-770
(Catalog# : 1791519)
TUG-770是高度有效的游离脂肪酸受体1(FFA1/GPR40)治疗2型糖尿病的激动
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2308520-97-8 | Cadefrecitinib (GLPG-3667)
(Catalog# : 20509)
Cadefrecitinib(GLPG-3667)是一种口服小分子TYK2激酶抑制剂,目前正处
1802735-28-9 | QBS10072S
(Catalog# : 25190)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
2377000-84-3 | Dencatistat (STP938)
(Catalog# : 25177)
Dencatistat 是一种口服生物可利用的小分子胞苷三磷酸合酶 1 (CTPS1)
1898207-64-1 | DS-1001b
(Catalog# : 25178)
DS-1001 是一种口服的脑渗透性突变 IDH1 选择性抑制剂。
1016340-64-9 | Z57346765
(Catalog# : 25191)
Z57346765 是一种 PGK1 特异性抑制剂,可降低 PGK1 糖酵解中代谢酶的
2416095-06-0 | CBR-470-1
(Catalog# : 25192)
CBR-470-1 是诱导 Nrf2 活性的糖酵解酶 PGK1 的抑制剂。
1898206-17-1 | Safusidenib
(Catalog# : 25149)
Safusidenib,也称为DS-1001,是一种口服异柠檬酸脱氢酶[NADP]细胞质(
2803470-63-3 | HC-7366
(Catalog# : 25076)
HC-7366 is a potent and selective activator of the general control nonderepressible 2
146426-40-6 | Flavopiridol ( 夫拉平度 )
(Catalog# : 237071)
Alvocidib is a synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is subst
2201056-66-6 | AG-270
(Catalog# : 25176)
MAT2A 抑制剂 AG-270 是一种口服的蛋氨酸腺苷转移酶 II α (MAT2A) 小分