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抑制剂/受体激动剂
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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Cas号索引 1
1256359-13-3 | 4,4,5,5-tetramethyl-2-(4-propan-2-ylsulfonylphenyl)-1,3,2-dioxaborolane
(Catalog# : 2062024)
1133378-83-2 | Tafenoquine-d3 succinate
(Catalog# : 2061704)
Tafenoquine-d3 is a trideuerium-labeled Tafenoquine derivative. Tafenoquine, also kno
1609960-30-6 | TH287
(Catalog# : 193135)
TH287是人7,8-二氢-8-草酸鸟苷三磷酸酶MTH1 (NUDT1)的有效抑制剂,IC50
1793059-58-1 | Tinostamustine盐酸盐
(Catalog# : 193112)
Tinostamustine,也称为EDO-S101,是一种烷基化有机去乙酰化酶抑制剂(H
191114-48-4 | Telithromycin
(Catalog# : 19374)
Telithromycin,也被称为HMR-3647和RU-66647,是一种半合成红霉素衍生物
1604810-84-5 | THZ2
(Catalog# : 192252)
THZ2,是THZ1的类似物,具有治疗三阴性乳腺癌(TNBC)的潜力,是一种
1227637-23-1 | Tegatrabetan
(Catalog# : 192145)
Tegatrabetan, 也称为Tegavivint和BC2059,是一种口服生物利用率和有效的
1359993-59-1 | Telratolimod
(Catalog# : 192144)
Telratolimod,也被称为 3M-052或MEDI-9197,是toll样受体7 (TLR-7)和toll样受
1260533-36-5 | TAS-116
(Catalog# : 191286)
TAS- 116是一种对热休克蛋白90 (Hsp90)亚型alpha和beta的有效选择性抑制
106635-81-8 | Tafenoquine succinate ( 他非诺喹琥珀酸盐 )
(Catalog# : 191123)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
106635-80-7 | Tafenoquine ( 他非诺喹 )
(Catalog# : 191122)
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo
1558021-37-0 | TP0463518
(Catalog# : 1812282)
TP0463518是一种新型高效的HIF脯氨酰羟化酶(PHD)抑制剂。TP0463518竞争
1009816-48-1 | Thiamet G
(Catalog# : 1812133)
Thiamet G是一种有效且具有选择性的O-GlcNAcase抑制剂.
1164462-05-8 | TG4-155
(Catalog# : 181232)
TG4-155 是一种大脑渗透EP2拮抗剂(KB = 2.4nM),在EP4(KB = 11.4µM)小组其他
123948-87-8 | Topotecan
(Catalog# : 1811212)
Topocecan是喜树碱的半合成衍生物,具有抗肿瘤活性。
1448169-71-8 | TAS-120
(Catalog# : 1811191)
TAS-120是成纤维细胞生长因子受体(FGFR)的口服生物有效抑制剂,具
1038984-31-4 | Tulrampator ( CX-1632 )
(Catalog# : 1811161)
Tulrampator,也被称为S-47445和CX-1632,是AMPA受体(AMPAR)的积极变构调制
1226056-71-8 | Thiazovivin
(Catalog# : 1811122)
Thiazovivin是一种具有选择性的,抑制浓度为2µM的ROCK活动的细胞-渗透
1862212-48-3 | TH 1217
(Catalog# : 1811021)
TH 1217是一种有效的dCTP焦磷酸酶1抑制剂。
1137868-52-0 | TAK-960
(Catalog# : 18762)
TAK-960是一种可口服的PLK1抑制剂,具有潜在的抗肿瘤活性。
1353644-70-8 | Theliatinib
(Catalog# : 186235)
Theliatinib又称HMPL-309,是一种新型的小分子、表皮生长因子受体酪
1616493-44-7 | Tucidinostat
(Catalog# : 186233)
Tucidinostat是组蛋白去乙酰化酶(HDAC) 1、2、3和10的一种苯甲酰胺类抑
1111556-37-6 | Takinib
(Catalog# : 18672)
Takinib选择性TAK1抑制剂,TNF-α刺激后细胞凋亡模型,类风湿性关节炎
1314890-29-3 | TMP269
(Catalog# : 185254)
TMP269是一种具有高强度、选择性和可渗透性的IIa型HDAC抑制剂,其
1374743-00-6 | Trilaciclib (G1T28)
(Catalog# : 185235)
Trilaciclib是一种小分子竞争性细胞周期蛋白依赖性激酶4和6(CDK4 /
171235-71-5 | TAPI-1
(Catalog# : 185181)
TAPI-1是TACE的抑制剂。它抑制TNF-a、TNFRI(p60)和TNFRII(p80)的裂解。
158899-10-6 | TLN-232
(Catalog# : 18594)
TLN-232, 也称为CAP-232,是一种具有潜在抗肿瘤活性的合成环七肽。
140194-24-7 | 醋酸曲普瑞林
(Catalog# : 18592)
醋酸曲普瑞林是一种促性腺激素释放激素激动剂(GnRH激动剂),用作
1383816-29-2 | Tropifexor
(Catalog# : 18591)
Tropifexor, 也称为LJN452, 是一种用于治疗胆静性肝病和非酒精性脂肪
1702809-17-3 | THZ531
(Catalog# : 184172)
THZ531是一种共价CDK12和CDK13共价抑制剂。环素依赖性激酶12和13 (CDK
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
1497439-74-3 | AD-8007
(Catalog# : 26A018)
AD-8007是一种选择性且可穿透血脑屏障的乙酰辅酶A合成酶2(ACSS2)
1802650-31-2 | ZY-444
(Catalog# : 26A020)
ZY-444是一种通过抑制PC活性发挥抗癌作用的药物。
2306525-79-9 | AD-5584
(Catalog# : 26A019)
AD-5584是一种新型脑渗透性ACSS2抑制剂。
3079716-11-0 | IDB-003
(Catalog# : 26A017)
IDB-003在体内抑制MDA-MB-231肿瘤生长。
1357362-02-7 | Vafidemstat
(Catalog# : 18891)
Vafidemstat又称ORY 2001,是一种赖氨酸特异性组蛋白去甲基化酶(LSD1)
1260247-42-4 | LLL12
(Catalog# : 25075)
LLL12是一种强效的STAT3抑制剂。LLL12在小鼠异种移植物模型中显示出
2758659-09-3 | ECC-5004
(Catalog# : 26A015)
ECC5004是一款每日一次、低剂量、小分子GLP-1受体激动剂。
2911585-37-8 | SILA-123
(Catalog# : 26A014)
SILA-123是一种II型FLT3抑制剂,对FLT3-WT(IC50=2.1 nM)和FLT3-ITD(IC50=1
1214922-52-7 | Encaleret sulfate
(Catalog# : 26A013)
Encaleret是一种正在研究的钙敏感受体的小分子拮抗剂,用于钙稳态
1431303-72-8 | Iadademstat ( ORY-1001 ) hydrochloride
(Catalog# : 26A011)
Iadademstat(ORY-1001)是一种口服活性、高效和选择性的表观遗传酶