武汉永璨生物科技有限公司
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
Other Building Blocks
On Sale
中间体
技术服务
定制合成
工艺研发
订购信息
联系我们
公司简介
联系我们
搜索
首页
网站地图
Cas号索引 1
按首字母搜索
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
1
2
3
4
5
6
7
8
9
«
55
56
57
58
59
60
61
62
63
64
»
Cas号索引 1
1361951-15-6 | TP-3654
(Catalog# : 178303)
TP-3654是一种Pim-1和Pim-3激酶抑制剂,可用于治疗前列腺癌、急性髓
1326712-16-6 | TAK1抑制剂
(Catalog# : 1791412)
TAK1 inhibitor isis discontinued.TAK1抑制剂是一种有效的、相对选择性的
1351636-18-4 | Tirabrutinib游离 ( ONO-4059 )
(Catalog# : 17031303)
Tirabrutinib,也被称为ONO- 4059,是在抑制剂中,一种强大的、具有口
1610882-30-8 | TCS-OX2-29盐酸盐
(Catalog# : 17031302)
TCS-OX2- 29或TCS OX2 29,也被称为TCSOX229和TCS - OX229,是一种选择性的
1603845-32-4 | TX1-85-1
(Catalog# : 17030713)
TX1-85-1是一种ErbB3抑制剂. TX2-121-1可能通过异位机制发挥Her3依赖性
183204-72-0 | Tipiracil HCl
(Catalog# : 17030710)
Tipiralacil,又称TPI,是胸腺嘧啶磷酸化酶抑制剂(TPI)。Tipiracil是TAS
1234365-97-9 | Tenapanor HCl
(Catalog# : 17030113)
Tenapanor, 也称为AZD-1722和RDX 5791, 是钠-质子(Na(+)/ H(+))交换器NHE3的抑
150915-40-5 | 盐酸替罗非班
(Catalog# : 17030103)
替罗非班是一种抗血小板药物。它属于一种名为糖蛋白IIb / IIIa抑
135598-68-4 | TAS-109
(Catalog# : 17022810)
TAS-109, 也称为DFP-10917和CNDAC,是一种具有潜在抗肿瘤活性的核苷酸脱
1256037-58-7 | TRX818
(Catalog# : 17022401)
TRX-818是一种可口服的生物制剂,具有潜在的抗肿瘤活性和抗血管
15421-84-8 | 乐可安
(Catalog# : 17021310)
乐可安是一种PDGF拮抗剂,可抑制PDGF生成胶质瘤细胞的增殖。
1439901-97-9 | ONO-4059盐酸盐
(Catalog# : 17012103)
ONO-4059是BTK的选择性和新型抑制剂,IC50为2.2 nm,ONO-4059与B细胞内的
113942-30-6 | 替莫唑胺酸
(Catalog# : 17011905)
替莫唑胺酸, 也称为TMZA, 是一种具有明显抗癌活性的替奥米特(TMZ)
1609960-31-7 | TH588
(Catalog# : 17011728)
TH588是NUDT1的一种有效抑制剂,其IC50值为5nm,具有良好的代谢稳定
1415716-58-3 | TG6-10-1
(Catalog# : 17011727)
TG6-10-1是前列腺素E2受体亚型EP2的有效和选择性拮抗剂。
1033805-22-9 | 特罗司他乙酯
(Catalog# : 17011722)
特罗司他乙酯, 也称为LX 1032或LX 1606, 是一种口服血清素合成抑制剂
161715-24-8 | 泰比培南酯
(Catalog# : 17011721)
泰比培南酯,也被称为ME1211和TBM-PI, 是一种新型口腔卡宾枪抗生素。
193620-69-8 | TAS-301
(Catalog# : 17011719)
TAS-301是一种有效的、选择性的球囊冠状动脉过度拉伸损伤后的收
174634-08-3 | TAS-103
(Catalog# : 17011718)
TAS-103,也称为BMS-247615, 是一种喹啉衍生物,在小鼠和人体肿瘤模型
150080-09-4 | Talabostat甲磺酸盐
(Catalog# : 17011717)
Talabostat, 也称为PT-100,具有抗肿瘤和造血作用的二肽肽酶抑制剂。
1312691-41-0 | TAK-659盐酸盐
(Catalog# : 17011716)
TAK-659是脾脏酪氨酸激酶(syk)的抑制剂,具有潜在的抗炎、免疫和抗
106463-17-6 | 盐酸坦索罗辛
(Catalog# : 17109008)
盐酸坦索罗辛是一个强有力的和选择性α1a肾上腺素能受体拮抗剂
1033040-23-1 | TPO agonist 1
(Catalog# : 6111515)
TPO agonist 1 can increase production of platelets by stimulating the TPO receptor in
1604810-83-4 | THZ1
(Catalog# : 6111013)
THZ1 is a novel selective and potent covalent CDK7 inhibitor with IC50(binding affini
1002789-86-7 | TZ9
(Catalog# : 611934)
TZ9 is a novel inhibitor of Rad6 ubiquitin conjugating enzyme(E2 enzyme); inhibits MD
1621523-07-6 | THZ1-R
(Catalog# : 611926)
THZ1-R is a non-cysteine reactive analog, which displays diminished activity for CDK7
1532533-78-0 | TGR-1202 hydrochloride
(Catalog# : 611905)
TGR-1202 hydrochloride is an orally available, next generation PI3Kdelta inhibitor, i
104987-11-3 | Tacrolimus
(Catalog# : 161009006)
It is also used in a topical preparation in the treatment of atopic dermatitis (eczem
103300-74-9 | Taltirelin
(Catalog# : 16071029)
Taltirelin
1314891-22-9 | TMP-195
(Catalog# : 16071020)
TMP-195
«
55
56
57
58
59
60
61
62
63
64
»
产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
2460722-04-5 | Oveporexton ( TAK-861 )
(Catalog# : 25194)
Oveporexton是一种口服小分子选择性食欲素2型受体(OX2R)激动剂。
2506273-81-8 | VT-3989
(Catalog# : 25200)
VT3989是一种首创的强效口服TEAD棕榈酰化抑制剂,可阻断YAP转录活
729-46-4 | JX06
(Catalog# : 25199)
JX06 是一种有效的,选择性的,共价的 PDK 抑制剂。
1616385-51-3 | Bezuclastinib
(Catalog# : 25198)
Bezuclastinib是KIT D816V突变体以及其他KIT外显子17突变体激酶活性的口
2649400-34-8 | Bexobrutideg ( NX-5948 )
(Catalog# : 25197)
Bexobrutideg(NX-5948)是一种BTK降解剂。
1039760-91-2 , 2074613-88-8 [ALTERNATIVE] | Rosolutamide ( AJ-201 ; ASC-JM17 )
(Catalog# : 25196)
Rosolutamide (formerly known as AJ-201, ASC-JM-17 or ALZ-002) 是一种姜黄素类似
1020634-41-6 | Soclenicant (BNC-210 ; IW-2143)
(Catalog# : 25195)
Soclenicant (BNC-210;IW-2143)是一种新型的α7烟碱型乙酰胆碱受体负
1532533-67-7 | Umbralisib
(Catalog# : 25085)
Umbralisib, also known as TGR1202 and RP5264 , is a highly specific, orally available
1802735-28-9 | QBS10072S
(Catalog# : 25190)
QBS10072S 是一种血脑屏障 (BBB) 渗透剂,由细胞毒性化疗结构域 N-双
1820812-16-5 | TAK-071
(Catalog# : 186269)
TAK-071 是一种毒蕈碱 M1 受体正变构调节剂。