武汉永璨生物科技有限公司
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抑制剂/受体激动剂
Angiogenesis
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Aldehydes
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Bromides
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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产品名字索引 R
Regadenoson
(Catalog# : 1810224, Cas# :
313348-27-5
)
Regadenoson是一种A2A腺苷受体激动剂,是一种冠状血管舒张剂,通常
RMC-4550
(Catalog# : 186251, Cas# :
2172651-73-7
)
RMC-4550一种有效且具有选择性的SHP2抑制剂。
RGX-104盐酸盐
(Catalog# : 186234, Cas# :
610318-03-1
)
RGX-104是一种具有潜在免疫调节和抗肿瘤活性的肝X受体激动剂。
Resminostat HCl
(Catalog# : 185317, Cas# :
1187075-34-8
)
Resminostat HCl是一种有效的HDAC1/3/6抑制剂。
Rovazolac
(Catalog# : 185234, Cas# :
1454288-88-0
)
Rovazolac是一种抗炎药。
Rolapitant游离
(Catalog# : 185152, Cas# :
5552292-08-7
)
Rolapitant,也被称为SCH-619734,是一种口服生物可用的,具有中央作
RO10-5824
(Catalog# : 185141, Cas# :
189744-46-5
)
RO10-5824是一种D4-选择性局部激动剂。RO10-5824是管理可卡因使用障碍
利卡司琼
(Catalog# : 184281, Cas# :
117086-68-7
)
利卡司琼,也称为Brl 46470,是止吐剂。
R-IMPP
(Catalog# : 18413, Cas# :
2133832-83-2
)
R-IMPP是PCSK9的转化抑制剂。
Rimegepant
(Catalog# : 18441, Cas# :
1289023-67-1
)
Rimegepant,也称为BMS-927711,在治疗偏头痛的临床试验中,是一种有
Ritlecitinib ( PF-06651600 )
(Catalog# : 18435, Cas# :
1792180-81-4
)
Ritlecitinib ( PF-06651600 )是一种有效的选择性JAK3抑制剂,是一种具有
R-GNE-140
(Catalog# : 18432, Cas# :
2003234-63-5
)
R-GNE-140是一种新型高效的乳酸脱氢酶(LDHA)抑制剂,LDHA的IC50为3nM,
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopropan-2-yl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183217, Cas# :
2097334-19-3
)
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopr
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183216, Cas# :
2097334-18-2
)
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate是一
Relebactam
(Catalog# : 1712156, Cas# :
1174018-99-5
)
Relebactam, also known as MK-7655, a potent and selective β-lactamase inhibitor.
盐酸利莫那班
(Catalog# : 179137, Cas# :
158681-13-1
)
利莫那班,又名SR141716,是一种抑制食欲的减肥药。它是为大麻素
Riviciclib HCl
(Catalog# : 179131, Cas# :
920113-03-7
)
Riviciclib,也称为P276-00,是具有潜在抗肿瘤活性的黄酮和细胞周期
RVT-501
(Catalog# : 17917, Cas# :
947620-48-6
)
RVT-501也称为E-6005,是4型磷酸二酯酶(PDE-4)抑制剂用于治疗特应
Roluperidone ( CYR-101 )
(Catalog# : 2017889, Cas# :
359625-79-9
)
Roluperidone, also known as MIN-101, CYR-101, and MT-210, is a 5-HT2A and sigma 2 rec
雷尼司他
(Catalog# : 178118, Cas# :
147254-64-6
)
雷尼司他,也被称为AS-3201、SX-3201,是一种醛糖还原酶抑制剂,由Dai
RG7800 ( RO6885247 )
(Catalog# : 174192, Cas# :
1449598-06-4
)
RG7800(RO6885247)是一种小分子改变生存运动神经元2的拼接。
罗拉吡坦盐酸盐
(Catalog# : 17030609, Cas# :
914462-92-3
)
罗拉吡坦, 也被称为SCH-619734是一种用于口服的,具有中央作用,选
RAF709
(Catalog# : 17030605, Cas# :
1628838-42-5
)
RAF709是一种Raf激酶抑制剂。
RPI-1
(Catalog# : 17030301, Cas# :
269730-03-2
)
RPI-1是一种ATP依赖的RET激酶抑制剂。通过口服RPI-1,导致生长阻滞
Recilisib钠盐
(Catalog# : 17022712, Cas# :
334969-03-8
)
Recilisib,也被称为 ON 01210钠,是一种放射性保护剂,它可以在接受
RO4987655
(Catalog# : 17011603, Cas# :
874101-00-5
)
RO4987655,也称为CH4987655, 是一种口服活性的小分子,靶向活性蛋白激
Ro 08-2750
(Catalog# : 17011602, Cas# :
37854-59-4
)
Ro 08-2750是一个强有力的和选择性的神经生长因子(神经生长因子)抑
Ribociclib HCl
(Catalog# : 17011305, Cas# :
1211443-80-9
)
Ribociclib HCl是一种有效且可口服的细胞周期蛋白依赖性激酶(CDK)抑
雷替曲塞
(Catalog# : 17011303, Cas# :
112887-68-0
)
雷替曲塞,也称为ZD 1694, 是1998年以来用于治疗结直肠癌的一种抗代
瑞替加滨
(Catalog# : 17011108, Cas# :
150812-13-8
)
瑞替加滨是一种新型的抗惊厥剂,具有活动范围广泛的癫痫模型。
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
----
Potassium Channel
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Methionine Adenosyltransferase (MAT)
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
NSD1 抑制剂 BT5
(Catalog# : 25207, Cas# :
2351225-46-0
)
BT5可有效抑制NSD1,与细胞中的SET结构域结合,并降低H3K36me2水平。
MA242 TFA
(Catalog# : 25206, Cas# :
1049704-18-8
)
MA242是一种MDM2和NFAT1双重抑制剂,可诱导MDM2自泛素化及降解,并抑
Dabogratinib ( TYRA-300 )
(Catalog# : 24073, Cas# :
2800223-30-5
)
Dabogratinib ( TYRA-300 )是一种口服选择性成纤维细胞生长因子受体3(
AF710B
(Catalog# : 25205, Cas# :
N/A
)
AF710B 是一种高效、选择性变构 M1 毒蕈碱和 σ1 受体激动剂。 AF710
MAT2A inhibitor 5
(Catalog# : 25204, Cas# :
2957874-18-7
)
MAT2A抑制剂5具有抑制MAT2A的高效力和对MTAP缺失的癌症细胞系的显著
(Rac)-AF710B
(Catalog# : 24083, Cas# :
1235733-73-9
)
AF-710B 是 σ 和 M1 毒蕈碱受体的激动剂;AF710B 是 AF710 的对映体。
Flurpiridaz-nonradiolabeled
(Catalog# : 25203, Cas# :
863888-33-9
)
Flurpiridaz是一种有前景的新型心脏PET成像示踪剂,是通过用氟-18放
Flurpiridaz-Precursor
(Catalog# : 25202, Cas# :
863888-32-8
)
现货
KL1333
(Catalog# : 25201, Cas# :
1800405-30-4
)
KL1333是一种口服的小有机分子,与NAD(P)H:醌氧化还原酶1(NQO1)
Palupiprant ( E7046 )
(Catalog# : 24055, Cas# :
1369489-71-3
)
E7046 is a potent and selective antagonist of the type 4 prostaglandin E2 (PGE2) rece