武汉永璨生物科技有限公司
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolic Enzyme/Protease
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
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Amines
Amino Acids
Anilines
Boronic Acids
Bromides
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Chiral Compounds
Deuterated
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Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
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On Sale
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产品名字索引 R
R547
(Catalog# : 1811151, Cas# :
741713-40-6
)
R547是口服生物有效的二氨基嘧啶环磷酰胺依赖性激酶抑制剂(CDKI)
Regadenoson
(Catalog# : 1810224, Cas# :
313348-27-5
)
Regadenoson是一种A2A腺苷受体激动剂,是一种冠状血管舒张剂,通常
RMC-4550
(Catalog# : 186251, Cas# :
2172651-73-7
)
RMC-4550一种有效且具有选择性的SHP2抑制剂。
RGX-104盐酸盐
(Catalog# : 186234, Cas# :
610318-03-1
)
RGX-104是一种具有潜在免疫调节和抗肿瘤活性的肝X受体激动剂。
Resminostat HCl
(Catalog# : 185317, Cas# :
1187075-34-8
)
Resminostat HCl是一种有效的HDAC1/3/6抑制剂。
Rovazolac
(Catalog# : 185234, Cas# :
1454288-88-0
)
Rovazolac是一种抗炎药。
Rolapitant游离
(Catalog# : 185152, Cas# :
5552292-08-7
)
Rolapitant,也被称为SCH-619734,是一种口服生物可用的,具有中央作
RO10-5824
(Catalog# : 185141, Cas# :
189744-46-5
)
RO10-5824是一种D4-选择性局部激动剂。RO10-5824是管理可卡因使用障碍
利卡司琼
(Catalog# : 184281, Cas# :
117086-68-7
)
利卡司琼,也称为Brl 46470,是止吐剂。
R-IMPP
(Catalog# : 18413, Cas# :
2133832-83-2
)
R-IMPP是PCSK9的转化抑制剂。
Rimegepant
(Catalog# : 18441, Cas# :
1289023-67-1
)
Rimegepant,也称为BMS-927711,在治疗偏头痛的临床试验中,是一种有
Ritlecitinib ( PF-06651600 )
(Catalog# : 18435, Cas# :
1792180-81-4
)
Ritlecitinib ( PF-06651600 )是一种有效的选择性JAK3抑制剂,是一种具有
R-GNE-140
(Catalog# : 18432, Cas# :
2003234-63-5
)
R-GNE-140是一种新型高效的乳酸脱氢酶(LDHA)抑制剂,LDHA的IC50为3nM,
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopropan-2-yl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183217, Cas# :
2097334-19-3
)
(2R,14R)-4-((R)-1-((R)-4-benzyl-2-oxooxazolidin-3-yl)-3-(tert-butoxycarbonyl)-1-oxopr
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate
(Catalog# : 183216, Cas# :
2097334-18-2
)
(R)-4-(2-(4-benzyl-2-oxooxazolidin-3-yl)-2-oxoethyl)benzyl 2,4-dimethylbenzoate是一
Relebactam
(Catalog# : 1712156, Cas# :
1174018-99-5
)
Relebactam, also known as MK-7655, a potent and selective β-lactamase inhibitor.
盐酸利莫那班
(Catalog# : 179137, Cas# :
158681-13-1
)
利莫那班,又名SR141716,是一种抑制食欲的减肥药。它是为大麻素
Riviciclib HCl
(Catalog# : 179131, Cas# :
920113-03-7
)
Riviciclib,也称为P276-00,是具有潜在抗肿瘤活性的黄酮和细胞周期
RVT-501
(Catalog# : 17917, Cas# :
947620-48-6
)
RVT-501也称为E-6005,是4型磷酸二酯酶(PDE-4)抑制剂用于治疗特应
Roluperidone ( CYR-101 )
(Catalog# : 2017889, Cas# :
359625-79-9
)
Roluperidone, also known as MIN-101, CYR-101, and MT-210, is a 5-HT2A and sigma 2 rec
雷尼司他
(Catalog# : 178118, Cas# :
147254-64-6
)
雷尼司他,也被称为AS-3201、SX-3201,是一种醛糖还原酶抑制剂,由Dai
RG7800 ( RO6885247 )
(Catalog# : 174192, Cas# :
1449598-06-4
)
RG7800(RO6885247)是一种小分子改变生存运动神经元2的拼接。
罗拉吡坦盐酸盐
(Catalog# : 17030609, Cas# :
914462-92-3
)
罗拉吡坦, 也被称为SCH-619734是一种用于口服的,具有中央作用,选
RAF709
(Catalog# : 17030605, Cas# :
1628838-42-5
)
RAF709是一种Raf激酶抑制剂。
RPI-1
(Catalog# : 17030301, Cas# :
269730-03-2
)
RPI-1是一种ATP依赖的RET激酶抑制剂。通过口服RPI-1,导致生长阻滞
Recilisib钠盐
(Catalog# : 17022712, Cas# :
334969-03-8
)
Recilisib,也被称为 ON 01210钠,是一种放射性保护剂,它可以在接受
RO4987655
(Catalog# : 17011603, Cas# :
874101-00-5
)
RO4987655,也称为CH4987655, 是一种口服活性的小分子,靶向活性蛋白激
Ro 08-2750
(Catalog# : 17011602, Cas# :
37854-59-4
)
Ro 08-2750是一个强有力的和选择性的神经生长因子(神经生长因子)抑
Ribociclib HCl
(Catalog# : 17011305, Cas# :
1211443-80-9
)
Ribociclib HCl是一种有效且可口服的细胞周期蛋白依赖性激酶(CDK)抑
雷替曲塞
(Catalog# : 17011303, Cas# :
112887-68-0
)
雷替曲塞,也称为ZD 1694, 是1998年以来用于治疗结直肠癌的一种抗代
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive Oxygen Species(ROS)
----
SOD
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolic Enzyme/Protease
----
PPAR
----
Proteasome
----
P450
----
Caspase
----
HSP
----
HIV Protease
----
PDE
----
MMP
----
Factor Xa
----
γ-secretase
----
Phospholipase
----
DPP4
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
NADPH-oxidase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
Isocitrate Dehydrogenase (IDH)
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
FPTase
----
RAR/RXR
----
Acetyl-CoA Carboxylase
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Glutaminase
----
Ketohexokinase(KHK)
----
Lipase
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
----
Phosphoglycerate Dehydrogenase (PHGDH)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
----
CGRP-Receptor
----
TRP-Channel
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
-- Nuclear Receptor
----
Androgen Receptor(AR)
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
ECI830
(Catalog# : 26A031, Cas# :
3054692-62-2
)
ECI830是一种实验性的CDK2抑制剂。
GNE-317
(Catalog# : 52282, Cas# :
1394076-92-6
)
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
DPTX-3186
(Catalog# : 26A010, Cas# :
3118994-80-9
)
DPTX3186 是一种口服的小分子凝聚体调节剂 (c-mod),可抑制 β-catenin
Avasopasem manganese (GC-4419; M-40419)
(Catalog# : 25108, Cas# :
435327-40-5
)
Avasopasem manganese, 也称为GC-4419、M 40419和SC-72325A,是超氧化物歧化酶
Iclepertin (BI-425809)
(Catalog# : 24084, Cas# :
1421936-85-7
)
Iclepertin(BI-425809)是一种口服的GlyT-1小分子抑制剂,用于治疗与
Kartogenin ( KGN )
(Catalog# : 52215, Cas# :
4727-31-5
)
Kartogenin(KGN)是一种合成小分子,通过激活smad-4/5通路刺激软骨细
Imisopasem manganese ( M40403; GC4403 )
(Catalog# : 72602, Cas# :
218791-21-0
)
Imisopasem manganese ( M40403; GC4403 ) 是一种稳定的非肽类 MnSOD 类似物,
Apecotrep (BI 764198)
(Catalog# : 26A048, Cas# :
2311863-36-0
)
Apecotrep(BI 764198)是一种潜在的同类首创、口服、选择性的TRPC6抑
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,
BH-30643
(Catalog# : 26A047, Cas# :
3062177-59-4
)
BH-30643是一种新型、口服、非共价、大环、突变选择性OMNI-EGFR抑制