武汉永璨生物科技有限公司
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抑制剂/受体激动剂
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联系我们
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联系我们
+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
Phenols
Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
Other Azoles
Other Heterocycles
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On Sale
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定制合成
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联系我们
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产品名字索引 R
Ro5-3335
(Catalog# : 20460, Cas# :
30195-30-3
)
Ro5-3335 是一种亲脂性小分子 RUNX1 抑制剂。
Ritlecitinib tosylate
(Catalog# : 20452, Cas# :
2192215-81-7
)
Ritlecitinib, also known as PF-06651600, is a potent and selective JAK3 inhibitor. PF
Ro 24-7429
(Catalog# : 2320201, Cas# :
139339-45-0
)
Ro24-7429是一种有效的口服活性HIV-1 反式激活蛋白Tat 拮抗剂和一种
布瑞拉沙秦(Brilaroxazine)
(Catalog# : 822224, Cas# :
1239729-06-6
)
RP-5063(Brilaroxazine) 是一种多模式的血清素和多巴胺受体调节剂,
Rucaparib Camsylate
(Catalog# : 20316, Cas# :
1859053-21-6
)
Rucaparib camsylate is a potent, orally available inhibitor of poly ADP-ribose polyme
Rhosin hydrochloride
(Catalog# : 21235, Cas# :
1281870-42-5
)
(R,Z)-1-(4-((3-chloro-4-((3-fluorobenzyl)oxy)phenyl)amino) quinazolin-6-yl)but-2-yn-1-one O-morpholin-3-ylmethyl oxime
(Catalog# : 20123102, Cas# :
1831116-75-6
)
Razuprotafib sodium
(Catalog# : 201221, Cas# :
1809275-69-1
)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
Razuprotafib
(Catalog# : 20102901, Cas# :
1008510-37-9
)
Razuprotafib,也称为AKB-9778,是血管内皮蛋白酪氨酸磷酸酶(VE-PTP)
Remibrutinib ( LOU064 )
(Catalog# : 2073103, Cas# :
1787294-07-8
)
Remibrutinib ( LOU064 ) is a Potent and Highly Selective Covalent Inhibitor of Bruton
Remdesivir
(Catalog# : 2071545, Cas# :
1809249-37-3
)
Remdesivir, also known as GS-5734, is a prodrug form of the antiviral nucleoside anal
RK-287107
(Catalog# : 2071520, Cas# :
2171386-10-8
)
RK-287107 is a potent TNKS/TNKS2 inhibitor (IC50 = 14.4 nM) with >7000-fold select
RBN-2397
(Catalog# : 207101, Cas# :
2381037-82-5
)
(2R,6S)-tert-butyl 4-(4-aminobenzoyl)-2,6-dimethylpiperazine-1-carboxylate
(Catalog# : 2062334, Cas# :
2161337-98-8
)
(R)-methyl 2-(tert-butyldimethylsilyloxy)propanoate
(Catalog# : 202329, Cas# :
171230-81-2
)
3-[(2RS)-tetrahydro-2H-pyran-2-yloxy]propanoic acid
(Catalog# : 2062017, Cas# :
1221443-23-7
)
[(1R,2S)-2-(3-fluorophenyl)-2-(hydroxymethyl)cyclopropyl]-methyl acetate
(Catalog# : 2062004, Cas# :
1369768-29-5
)
Rigosertib
(Catalog# : 690120, Cas# :
592542-59-1
)
Rigosertib(ON-01910) is a multi-kinase inhibitor and a selective anti-cancer agent, w
Resatorvid
(Catalog# : 206102, Cas# :
243984-11-4
)
Resatorvid, also known as TAK-242, is a cell-permeable inhibitor of TLR4 signaling, b
RU320521
(Catalog# : 204503, Cas# :
2262452-06-0
)
RU320521, also known as RU521; RU.521 is a potent and selective inhibitor of cGAS, in
(2R)-2-乙炔-2-甲基-1-吡咯烷乙酸 1,1-二甲基乙酯
(Catalog# : 580586, Cas# :
2086689-88-3
)
(2R)-2-乙炔-2-甲基-1-吡咯烷乙酸 1,1-二甲基乙酯 是 Pamiparib合成中一
Remetinostat
(Catalog# : 193111, Cas# :
946150-57-8
)
Remetinostat,也被称为SHP-141,是一种外用制剂,含有组蛋白脱乙酰
RG7834
(Catalog# : 19355, Cas# :
2072057-17-9
)
RG7834,也称为RO7020322,是一种新型口服HBV病毒基因表达抑制剂阻断病
RWJ-56110
(Catalog# : 19353, Cas# :
252889-88-6
)
RWJ-56110是一种选择性蛋白酶活化受体-1 (PAR1)拮抗剂。它阻断凝血酶
RBC8
(Catalog# : 19313, Cas# :
361185-42-4
)
RBC8是一种RalA和RalB GTPase抑制剂(EC50 ~ 3.5μM)。RBC8抑制小鼠异种移植
Rogaratinib
(Catalog# : 192277, Cas# :
1443530-05-9
)
Rogaratinib, 也称为BAY-1163877, 是一种异常的成纤维细胞生长因子受体
Rebimastat
(Catalog# : 192254, Cas# :
259188-38-0
)
Rebimastat,又名BMS275291,是一种具有潜在抗肿瘤活性的巯基第二代
Retosiban
(Catalog# : 192193, Cas# :
820957-38-8
)
Retosiban,又称GSK-221149-A;是一种口服活性强、选择性强的亚纳米(Ki
RKI-1313
(Catalog# : 19183, Cas# :
1342276-76-9
)
RKI-1313是RKI-1447 (GLXC-05200)的阴性对照,是Rho-相关ROCK激酶的有效抑
RGX-104 free form
(Catalog# : 19181, Cas# :
610318-54-2
)
RGX-104,又称SB 742881,是肝脏X受体激动剂,具有潜在的免疫调节和
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,