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抑制剂/受体激动剂
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+86-17702719238
sales@sun-shinechem.com
首页
抑制剂/受体激动剂
Angiogenesis
Anti-infection
Apoptosis
Autophagy
Cell Cycle
Cytoskeleton
DNA Damage
Epigenetics
GPCR & G Protein
Immunology & Inflammation
JAK/STAT
MAPK
Membrane Transporter/Ion Channel
Metabolism
Neuronal Signaling
NF-κB
Protein Tyrosine Kinase
Proteases
PI3K/Akt/mTOR
Stem Cells & Wnt
TGF-beta/Smad
Ubiquitin
Vitamin D Related
PROTAC
Antibody-drug Conjugate/ADC Related
Microbiology
Others
分子砌块
Aldehydes
Amines
Amino Acids
Anilines
Boronic Acids
Bromides
Carboxes
Catalysts
Chiral Compounds
Deuterated
Fluorides
Imidazoles
Indoles and Oxindoles
Iodos
Nitro Compounds
Oxazoles
Peg Linkers
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Piperidines
Pyridines
Pyrimidines
Quinolines
Sulfonamides
Thiazoles
Trifluoroborates
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联系我们
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产品名字索引 I
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产品名字索引 I
IITZ-01
(Catalog# : 2071519, Cas# :
1807988-47-1
)
IITZ-01 (Autophagy inhibitor IITZ-01) is a novel potent lysosomotropic autophagy inhi
4-iodo-2-isopropyl-1-Methyl-1H-iMidazole
(Catalog# : 2062023, Cas# :
851870-24-1
)
1-iodo-2-methoxy-4-methylbenzene
(Catalog# : 2062008, Cas# :
186583-59-5
)
IUN76750
(Catalog# : 2051507, Cas# :
1690176-75-0
)
IUN76750 is a PAR-2 signaling pathway inhibitor. IUN76750 has CAS#1690176-75-0, has n
ICEC0942 mesylate
(Catalog# : 204306)
ICEC0942, also known as PPDA-001 and CT7001, is a potent, orally active and selective
ICEC0942 HCl
(Catalog# : 204305, Cas# :
1805789-54-1 (HCl)
)
ICEC0942, also known as PPDA-001 and CT7001, is a potent, orally active and selective
ICEC0942 free base
(Catalog# : 204304, Cas# :
1805833-75-3 (free base)
)
ICEC0942, also known as PPDA-001 and CT7001, is a potent, orally active and selective
ITI-214
(Catalog# : 54192, Cas# :
1160521-50-5
)
ITI214 是一种选择性的PDE1抑制剂。
ITI-214磷酸盐
(Catalog# : 512193, Cas# :
1642303-38-5
)
ITI-214 is a potent and selective phosphodiesterase 1 (PDE1) inhibitor. As the clinic
IDH889
(Catalog# : 19319, Cas# :
1429179-07-6
)
IDH889是一种有效的选择性IDH1抑制剂。IDH899为IDH (R132H) IC50 = 20 nM;细
INCB3284甲磺酸盐
(Catalog# : 191143, Cas# :
887401-93-6
)
INCB3284是一种有效的、选择性的、可口服的hCCR2拮抗剂。
Indeglitazar
(Catalog# : 1812131, Cas# :
835619-41-5
)
Indeglitazar,也称为PPM-204和PLX-204,是一个可口服的过氧化物酶体增
IU1-47
(Catalog# : 181025, Cas# :
670270-31-2
)
IU1-47是一种有效且具有选择性的USP14抑制剂。
Inarigivir soproxil
(Catalog# : 186277, Cas# :
942123-43-5
)
Inarigivir soproxil,也被称为SB 9200,是一种抗病毒药物。
IT-901
(Catalog# : 186276, Cas# :
1584121-99-2
)
IT-901是一个血液恶性肿瘤抑制剂,通过阻断NF-κB-Controlled氧化应激反
INX 08189
(Catalog# : 186253, Cas# :
1234490-83-5
)
INX 08189 是一种RNA引导的RNA聚合酶(NS5B)抑制剂,可用于丙型肝炎病
IWP-O1
(Catalog# : 186222, Cas# :
2074607-48-8
)
IWP-O1是一种高效的Porcn抑制剂,对Wnt蛋白的分泌至关重要,它有助
INCB057643
(Catalog# : 185232, Cas# :
1820889-23-3
)
INCB057643是一种BET抑制剂。在卵巢癌中,INCB054329降低了同源重组效
Iberdomide
(Catalog# : 185216, Cas# :
1323403-33-3
)
Iberdomide,也称为CC-220,可用于治疗系统性红斑狼疮。
INCB3344
(Catalog# : 185215, Cas# :
1262238-11-8
)
INCB3344是CCR2受体的一种有效的选择性拮抗剂,它在结合拮抗的IC(5
iCRT3
(Catalog# : 18492, Cas# :
901751-47-1
)
iCRT3是Wnt/β-catenin信号的拮抗剂,在Wnt responsive STF16-luc reporter assay
IDO-IN-2
(Catalog# : 184317, Cas# :
1668565-74-9
)
IDO抑制剂1是IDO的有效抑制剂(吲哚胺-(2,3)-二氧合酶),IC50为3nm。
IPI-3063
(Catalog# : 18433, Cas# :
1425043-73-7
)
IPI-3063是一种选择性的Phosphoinoside-3-激酶p110δ 抑制剂。IPI-3063能有
5-碘-1-甲基咪唑
(Catalog# : 1712292, Cas# :
71759-88-1
)
5-碘-1-甲基咪唑是一种分子砌块。
6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-amine
(Catalog# : 1710123, Cas# :
1448427-99-3
)
6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-amine
IDRA-21
(Catalog# : 179134, Cas# :
22503-72-6
)
IDRA-21是一种阳性的AMPA受体调节剂。IDRA-21抑制突触和突触外NMDA受
ISCK03
(Catalog# : 1791118, Cas# :
945526-43-2
)
ISCK03是一种有效的c-kit抑制剂。ISCK03抑制在501mel人黑素瘤细胞的SC
IACS-9571
(Catalog# : 1783019, Cas# :
1800477-30-8
)
IACS-9571是一种有效的选择性TRIM24和BRPF1抑制剂。布罗莫结构域包括
异硫蓝
(Catalog# : 178017, Cas# :
68238-36-8
)
Isosulfan blue 是一种用于淋巴管造影中淋巴管识别的蓝色染料。Isos
Importazole
(Catalog# : 17031013, Cas# :
662163-81-7
)
Importazole是一种运输受体importin-β的小分子抑制剂,专门阻止import
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产品分类
信号通路
-- Angiogenesis
----
VEGFR
----
JAK
----
EGFR
----
PDGFR
----
FLT3
----
FGFR
----
Src
----
ALK
----
Syk
----
HIF
-- Anti-infection
----
CMV
----
Filovirus
----
HBV
----
HCV
----
HIV
----
HSV
----
Influenza Virus
----
RSV
----
SARS-CoV
----
Antibacterial
----
Antifungal
----
Parasite
-- Apoptosis
----
PD-1
----
PD-L1
----
Bcl-2
----
Caspase
----
TNF-alpha
----
Survivin
----
IAP
----
PERK
----
p53
----
Mdm2
----
E1/E2/E3 Enzyme
-- Autophagy
----
LRRK2
----
CXCR
----
Autophagy
-- Cell Cycle
----
CDK
----
PD-1
----
PD-L1
----
Chk
----
ROCK
----
PLK
----
APC
----
Wee1
----
DYRK
----
c-Myc
----
Aurora Kinase
----
ROCK inhibitor
----
Eukaryotic Initiation Factor (eIF)
----
NEKs
-- Cytoskeleton
----
HSP
----
Kinesin
----
Integrin
----
Dynamin
----
Wnt
----
β-catenin
----
Gap Junction Protein
-- DNA Damage
----
PARP
----
DNA/RNA Synthesis
----
Sirtuin
----
Topoisomerase
----
DNA-PK
----
Telomerase
----
RAD51
----
HDAC
----
ATM
----
DNA alkylator
----
Mps1
-- Epigenetics
----
PARP
----
JAK
----
Pim
----
PKC
----
PKD
----
Sirtuin
----
Histone Demethylase
----
Histone Acetyltransferase
----
HDAC
----
HIF-PH
----
Aurora Kinase
----
Histone Methyltransferase
----
METTL3
----
Epigenetic Reader Domain
----
Methionine Adenosyltransferase (MAT)
-- GPCR & G Protein
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
Endothelin Receptor
----
SGLT
----
OX Receptor
----
CaSR
----
CXCR
----
Vasopressin Receptor
----
Glucagon Receptor
----
Prostaglandin Receptor
----
5-HT Receptor
----
Adrenergic Receptor
----
Cannabinoid Receptor
----
Sphingosine 1 Phosphate Receptor
----
PKA
----
Adenosine Receptor
----
GnRH
----
LPL Receptor
----
Ras
----
Cholecystokinin Receptor
----
Melanocortin Receptor
----
RXFP Receptor
----
Bradykinin Receptor
----
GLP Receptor
-- Immunology & Inflammation
----
PD-1
----
PD-L1
----
COX
----
CCR
----
Histamine Receptor
----
TLR
----
CXCR
----
MALT
----
TDO
----
NOS
----
NADPH-oxidase
----
IDO
----
Thrombopoietin Receptor(TPO)
----
NLR inhibitor
----
Interleukin Related
----
CD73
----
Complement System
----
Aryl Hydrocarbon Receptor
----
Kallikrein
----
IRAK
----
Reactive-Oxygen-Species-ROS
-- JAK/STAT
----
JAK
----
STAT
----
Pim
----
EGFR
-- MAPK
----
MEK
----
Raf
----
p38 MAPK
----
ERK
----
MNK
----
Mixed Lineage Kinase
----
JNK
----
MAP4K
-- Membrane Transporter/Ion Channel
----
BCRP
----
CFTR
----
EAAT2
----
GABA Receptor
----
HCN Channel
----
Monoamine Transporter
----
Na+/Ca2+ Exchanger
----
Na+/K+ ATPase
----
nAChR
----
Calcium Channel
----
Chloride Channel
----
CRAC Channel
----
GlyT1
----
iGluR
----
P2X Receptor
----
P-glycoprotein
----
Amino acid transporter
----
Monocarboxylate Transporter
----
Potassium Channel
----
Proton Pump
-- Metabolism
----
PPAR
----
P450
----
HSP
----
PDE
----
Factor Xa
----
Phospholipase
----
FAAH
----
CETP
----
Lipoxygenase
----
HMG-CoA Reductase
----
Fatty Acid Synthase
----
FXR
----
NAMPT
----
TDO
----
Carbonic Anhydrase
----
Monoamine Oxidase
----
IDO
----
Mitochondrial Metabolism
----
MAGL
----
Epoxide Hydrolase
----
LXR
----
Myeloperoxidase (MPO)
----
RAR/RXR
----
Acyltransferase
----
UGT
----
MMP
----
ATP Citrate Lyase
----
Ketohexokinase(KHK)
----
Lactate dehydrogenase
----
Glyoxalase (GLO)
----
E1/E2/E3 Enzyme
----
PANK(pantothenate kinase)
-- Neuronal Signaling
----
COX
----
Histamine Receptor
----
Dopamine Receptor
----
Opioid Receptor
----
GABA Receptor
----
OX Receptor
----
Amyloid-β
----
5-HT Receptor
----
γ-secretase
----
Adrenergic Receptor
----
NMDA Receptor
----
GlyT1
----
Beta-secretase
----
Sigma Receptor
----
mAChR
----
α-Synuclein
----
Tau Protein
----
Cannabinoid Receptor
----
Transthyretin (TTR)
----
Melanocortin Receptor
----
Glucosylceramide Synthase (GCS)
-- NF-κB
----
NF-κB
----
HDAC
----
IKK
----
Keap1-Nrf2
-- Protein Tyrosine Kinase
----
VEGFR
----
EGFR
----
PDGFR
----
IGF-1R
----
FLT3
----
FGFR
----
c-Kit
----
Src
----
ALK
----
Ephrin receptor
----
BTK
----
Trk receptor
----
c-Met/HGFR
----
Syk (Spleen tyrosine kinase)
----
TAM Receptor
----
ULK1
----
CSF-1R
----
TYK2
----
ROS Kinase
----
Bcr-Abl
----
FAK
----
RET
----
Phosphoglycerate Kinase (PGK)
-- Proteases
----
Proteasome
----
Caspase
----
HIV Protease
----
MMP
----
γ-secretase
----
DPP4
----
Isocitrate Dehydrogenase (IDH)
----
FPTase
----
Acetyl-CoA Carboxylase
----
Glutaminase
----
Lipase
-- PI3K/Akt/mTOR
----
PI3K
----
Akt
----
GSK-3
----
S6 Kinase
----
AMPK
----
DNA-PK
----
MELK
----
PIKfyve
----
PI4K
----
PTEN
----
mTOR
----
ATM
----
PDK-1
----
ATR
----
Vps34
-- Stem Cells & Wnt
----
GSK-3
----
JAK
----
STAT
----
ROCK
----
TGF-beta/Smad
----
Wnt
----
γ-secretase
----
β-catenin
----
smo
----
Notch
-- TGF-beta/Smad
----
PKC
----
ROCK
----
TGF-beta/Smad
-- Ubiquitin
----
Proteasome
----
p97
----
Deubiquitinase
----
DUB
-- Vitamin D Related
----
VD/VDR
-- PROTAC
----
Molecular Glues
----
PROTACs
--
Antibody-drug Conjugate/ADC Related
--
Microbiology
-- Others
----
PKK
----
Others modulator
----
Estrogen Receptor/ERR
----
ChoKα
----
Newest added products
抑制剂/受体激动剂
中间体
分子砌块
--
Aldehydes
--
Amines
--
Amino Acids
--
Anilines
--
Boronic Acids
--
Bromides
--
Carboxes
--
Catalysts
--
Chiral Compounds
--
Deuterated
--
Fluorides
--
Imidazoles
--
Indoles and Oxindoles
--
Iodos
--
Nitro Compounds
--
Oxazoles
--
Peg Linkers
--
Phenols
--
Piperidines
--
Pyridines
--
Pyrimidines
--
Quinolines
--
Sulfonamides
--
Thiazoles
--
Trifluoroborates
--
Other Azoles
--
Other Heterocycles
--
Other Building Blocks
--
On Sale
新产品
天然化合物
最新产品
Mitoquinol mesylate (MitoQ)
(Catalog# : 26A042, Cas# :
845959-55-9
)
Mitoquinol mesylate (MitoQ) 是一种线粒体靶向抗氧化剂,具体而言,它
SPG-601 ( VSN-16R )
(Catalog# : 24042, Cas# :
1246960-09-7
)
SPG-601(原名VSN-16R)是一种口服给药、同类首创的小分子药物,是
LY3039478 ( Crenigacestat )
(Catalog# : 17021601, Cas# :
1421438-81-4
)
LY3039478 ( Crenigacestat ) 是一种选择性 NOTCH1 抑制剂,通过阻断 VEGFA/
PF-9366
(Catalog# : 184107, Cas# :
72882-78-1
)
PF-9366是一种新型的人蛋氨酸腺苷转移酶2A (Mat2A),肝外同种型。
MAT2A-IN-22
(Catalog# : 26A021, Cas# :
2925330-18-1
)
MAT2A-IN-22 (Compound 29-1) 是一种可透过血脑屏障的和口服有效的 MAT2A
Pantothenate kinase-IN-3
(Catalog# : 26A041)
泛酸激酶-IN-3(亦称化合物21,https://doi.org/10.1021/acs.jmedchem.5c03452)
Claziprotamidum ( Claziprotamide ; BBP-671 )
(Catalog# : 26A040, Cas# :
2361124-03-8
)
Claziprotamidum(Claziprotamide;BBP-671)是一种强效、口服有效且能透过
PZ-3022
(Catalog# : 26A039, Cas# :
2170608-85-0
)
PZ-3022是一种别构型的PanK激活剂,能够抵消C3-CoA的抑制作用。
PZ-2891
(Catalog# : 193282, Cas# :
2170608-82-7
)
PZ-2891是一种强效的、选择性的、口服活性泛酸激酶(PANK)调制剂,
Pantothenate kinase-IN-2
(Catalog# : 26A038, Cas# :
902614-04-4
)
Pantothenate kinase-IN-2是一种泛酸激酶抑制剂,对PanK2的IC50值为92 nM,