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重点产品

编号化学名称Cas号纯度化学结构
122941Pacritinib(SB1518)937272-79-2≧98.0%
Pacritinib (SB1518) 是一种高选择性激酶抑制剂,对 JAK2、FLT3、IRAK1 和
1662118MK-8931 ( Verubecestat )1286770-55-598% by HPLC/HNMR 
MK-8931(verubecestat)是一种BACE抑制剂,是由默沙东公司研制开发。主
611902PF-049790641220699-06-8≧98.0%
PF-04979064 is a potent and selective PI3K/mTOR dual kinase inhibitor with an IC(50)
6111110Nastorazepide209219-38-598% 
Nastorazepide (Z-360) is a selective, orally available, 1,5-benzodiazepine-derivative
6112701JPH203(KYT-0353)1037592-40-7≧98.0%
JPH203(also known as KYT-0353) is a potent and selective LAT1 selective ( L-type amin
6121401Vadadustat ( AKB-6548 )1000025-07-998% 
Vadadustat (AKB-6548), a novel, titratable, oral hypoxia-inducible factor prolyl hydr
16122810Elacestrant dihydrochloride1349723-93-8≧98.0%
Elacestrant dihydrochloride, also known as RAD1901, is an orally available, selective
16122847WWL70947669-91-2≧98.0%
WWL70是选择性ABHD6抑制剂,在创伤性脑损伤和多发性硬化症的动物
16123054MK-10641207253-08-4≧98.0%
MK-1064是一种有效的、选择性和口服的Orexin OX2受体拮抗剂,用于治
1710901Netarsudil (AR-13324) 2HCl1253952-02-1≧98.0%
Netarsudil (a.k.a. AR-13324)是一种ROCK抑制剂,Ki值为 0.2-10.3 nM。它目前
71161SBI02069651884220-36-398% 
SBI0206965是一种有效的选择性自噬激酶ULK1抑制剂。许多肿瘤变得沉
17012102lumateperone(Tosylate)1187020-80-998%
Lumateperone (ITI-722/ITI-007)是一种新型的双5HT2A受体拮抗剂/多巴胺磷蛋