编号 | 化学名称 | Cas号 | 纯度 | 化学结构 |
---|---|---|---|---|
20103003 | ML380 | 1627138-52-6 | ≧98.0% | |
ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator | ||||
2071535 | Danicopan | 1903768-17-1 | ≧98.0% | |
Danicopan, aslo known as ACH-4471 and ACH-0144471, is a highly potent, orally active | ||||
20259 | Elinzanetant ( NT-814 ) | 929046-33-3 | ≧98.0% | |
Elinzanetant,以前称为 NT-814 (45),是一种双重 NK1,3R 拮抗剂,因此有 | ||||
19381 | Abrocitinib | 1622902-68-4 | >98% | |
Abrocitinib(PF-04965842)是Pifzer研发的是一种Janus激酶抑制剂药物,目 | ||||
20294 | Paltusotine ( CRN-00808 ) | 2172870-89-0 | ≧98.0% | |
Paltusotine 是一类新型的、口服、选择性、非肽类2型生长抑素受体 | ||||
51703 | Luminespib ( NVP-AUY922 ; VER-52296 ) | 747412-49-3 | 98% | |
NVP-AUY922 is an experimental drug candidate for the treatment of cancer. It was disc | ||||
51902 | AT13148 | 1056901-62-2 | ≧98% | |
AT13148, a first-in-class multi-AGC kinase inhibitor, against gastric cancer cells. A | ||||
51603 | AZD6482 | 1173900-33-8 | ≧98.0% | |
AZD6482 is aPI3Kinhibitor withIC50of 10 nM, 8-, 87- and 109-fold more selective to PI | ||||
51905 | CPI-613(Devimistat ) | 95809-78-2 | ≧98.0% | |
CPI-613( Devimistat ) is an E1 pyruvate dehydrogenase (PDH) modulator that prevents c | ||||
52023 | DCC-2036(Rebastinib) | 1020172-07-9 | 98% | |
Rebastinib(DCC-2036;DCC2036) is an inhibitor of tyrosine kinases TIE2 and ABL1.Rebast | ||||
52019 | GSK 2656157 | 1337532-29-2 | 98% | |
GSK2656157 is an ATP-competitive and highly selective inhibitor ofPERKwithIC50of 0.9 | ||||
51608 | SSR128129E | 848318-25-2 | 98% | |
SSR128129E is an orally-active and allostericFGFR1inhibitor withIC50of 1.9 M, while n |