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产品目录

编号化学名称Cas号纯度化学结构
122524GW2580870483-87-798% 
GW2580 is an orally bioavailable inhibitor of c-FMS kinase; completely inhibited huma
122805Balipodect ( TAK-063 ) 1238697-26-198% 
Balipodect (TAK 063 )is a novel PDE10A inhibitor. It has shown high inhibitory activi
122919Tenapanor1234423-95-098% 
Tenapanoris an inhibitor of the sodium-proton exchanger NHE3. Thisantiporter protein
122941Pacritinib(SB1518)937272-79-2≧98.0%
Pacritinib (SB1518) 是一种高选择性激酶抑制剂,对 JAK2、FLT3、IRAK1 和
51627MK76221227923-29-698% by HPLC 
MK-7622isused as adjunctive therapy to acetylcholinesterase inhibitors (AChEIs) for t
20267Almonertinib1899921-05-198% Min.
Almonertinib is an orally available inhibitor of the epidermal growth factor receptor
10403CAY10566944808-88-298% 
Coming soon!
25152Avutometinib ( 别名: Ro 5126766; CH5126766 )946128-88-7≧98.0%
Avutometinib(别名:RO-5126766、CH-5126766)是一种正在开发的 Ras-Raf-ME
011813Avoralstat918407-35-995.0% 
Avoralstat(前身为BCX4161)是一种有效的小分子口服血浆激肽释放酶
1662118MK-8931 ( Verubecestat )1286770-55-598% by HPLC/HNMR 
MK-8931(verubecestat)是一种BACE抑制剂,是由默沙东公司研制开发。主
611902PF-049790641220699-06-8≧98.0%
PF-04979064 is a potent and selective PI3K/mTOR dual kinase inhibitor with an IC(50)
6111110Nastorazepide209219-38-598% 
Nastorazepide (Z-360) is a selective, orally available, 1,5-benzodiazepine-derivative