编号 | 化学名称 | Cas号 | 纯度 | 化学结构 |
---|---|---|---|---|
1811121 | DCC-2618 ( Ripretinib ) | 1442472-39-0 | >98% | |
Ripretinib,又名DCC-2618,是一种有效的、口服活性和选择性KIT/PDGFR抑 | ||||
1811162 | PF-05231023 | 1037589-69-7 | >98% | |
PF-05231023是一种长效FGF21仿生产品。PF-05231023可以减轻非人类灵长类 | ||||
5141902 | Avatrombopag maleate | 677007-74-8 | 96% | |
Avatrombopag maleate 是一种口服生物可用的小分子血栓生成素受体激动 | ||||
1811211 | Anlotinib HCl ( AL-3818 ) | 1360460-82-7 | ≧98.0% | |
Anlotinib也被称为AL3818,是一种受体酪氨酸激酶(RTK)抑制剂,具有潜 | ||||
19132 | Cilofexor ( GS-9674 ) | 1418274-28-8 | ≧98.0% | |
Cilofexor(也称为 GS-9674)是一种非甾体法尼醇 X 受体(FXR)激动剂 | ||||
191122 | Tafenoquine ( 他非诺喹 ) | 106635-80-7 | ≧98.0% | |
Tafenoquine is being investigated as a potential treatment for malaria, as well as fo | ||||
191146 | AR-9281 | 913548-29-5 | >98% | |
AR-9281是一种可溶性环氧化物水解酶(s-EH)抑制剂,有望用于高血压 | ||||
19356 | AZ876 | 898800-26-5 | >98% | |
AZ876,又称AZ-876,是一种肝脏X受体激动剂。AZ876可预防病理性心肌 | ||||
S510901 | Cenicriviroc Mesylate | 497223-28-6 | 98% Min. | |
Cenicriviroc(代号TAK-652,TBR-652)是用于治疗HIV感染的实验候选药物 | ||||
512193 | ITI-214磷酸盐 | 1642303-38-5 | 98% Min. | |
ITI-214 is a potent and selective phosphodiesterase 1 (PDE1) inhibitor. As the clinic | ||||
52001 | Selisistat ( EX-527 ) | 49843-98-3 | ≧98.0% | |
Selisistat 是第一个确定的有效且可渗透细胞的 SIRT1 特异性抑制剂, | ||||
6111901 | UNC2541 | 1612782-86-1 | 98% Min. | |
UNC2541 is a potent and MerTK-specific inhibitor and exhibits sub-micro molar inhibit |