Elinzanetant ( NT-814 )
编号: 20259
Cas号: 929046-33-3
纯度: ≧98.0%
Elinzanetant, previously known as NT-814 (45), is a dual NK1,3R antagonist and therefore has the potential to reduce GnRH pulsatility by blocking the endogenous effects of NKB and SP on the reproductive axis.
仅供研究使用。 我们不向患者出售。
化学信息
| 名称 | Elinzanetant ( NT-814 ) |
|---|---|
| Iupac 化学名称 | 2-[3,5-bis(trifluoromethyl)phenyl]-N-{4-(4-fluoro-2-methylphenyl)-6-[(7S,9aS)-7-(hydroxymethyl)hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]pyridin-3-yl}-N,2-dimethylpropanamide |
| 同义词 | Elinzanetant ; GSK1144814A ; NT-814 ; NT 814 ; NT814 ; GSK-1144814A ; GSK 1144814A |
| 英文同义词 | Elinzanetant ; GSK1144814A ; NT-814 ; NT 814 ; NT814 ; GSK-1144814A ; GSK 1144814A |
| 分子式 | C33H35F7N4O3 |
| 分子量 | 668.64 |
| Smile | CC(C)(C1=CC(C(F)(F)F)=CC(C(F)(F)F)=C1)C(N(C2=C(C3=CC=C(F)C=C3C)C=C(N4C[C@@]5([H])COCCN5C[C@H]4CO)N=C2)C)=O |
| InChiKey | DWRIJNIPBUFCQS-DQEYMECFSA-N |
| InChi | InChI=1S/C33H35F7N4O3/c1-19-9-23(34)5-6-26(19)27-13-29(44-16-25-18-47-8-7-43(25)15-24(44)17-45)41-14-28(27)42(4)30(46)31(2,3)20-10-21(32(35,36)37)12-22(11-20)33(38,39)40/h5-6,9-14,24-25,45H,7-8,15-18H2,1-4H3/t24-,25-/m0/s1 |
| Cas号 | 929046-33-3 |
| 相关CAS号 | 929046-33-3 |
订购信息
| 包装 | 价格 | 库存 | 纯度 | 备货期 |
|---|---|---|---|---|
| 大货 | 询价 | 询价 | 询价 |
| 外观性状 | Off-white Solid |
|---|---|
| 纯度 | ≧98.0% |
| 存储 | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| 可溶性 | Soluble in DMSO |
| 处理方式 | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| 运输条件 | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| 海关编码 |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
