编号 | 化学名称 | Cas号 | 纯度 | 化学结构 |
---|---|---|---|---|
186253 | INX 08189 | 1234490-83-5 | >98% | |
INX 08189 是一种RNA引导的RNA聚合酶(NS5B)抑制剂,可用于丙型肝炎病 | ||||
186222 | IWP-O1 | 2074607-48-8 | >98% | |
IWP-O1是一种高效的Porcn抑制剂,对Wnt蛋白的分泌至关重要,它有助 | ||||
185232 | INCB057643 | 1820889-23-3 | >98% | |
INCB057643是一种BET抑制剂。在卵巢癌中,INCB054329降低了同源重组效 | ||||
185216 | Iberdomide | 1323403-33-3 | >98% | |
Iberdomide,也称为CC-220,可用于治疗系统性红斑狼疮。 | ||||
185215 | INCB3344 | 1262238-11-8 | >98% | |
INCB3344是CCR2受体的一种有效的选择性拮抗剂,它在结合拮抗的IC(5 | ||||
18492 | iCRT3 | 901751-47-1 | >98% | |
iCRT3是Wnt/β-catenin信号的拮抗剂,在Wnt responsive STF16-luc reporter assay | ||||
184317 | IDO-IN-2 | 1668565-74-9 | >98% | |
IDO抑制剂1是IDO的有效抑制剂(吲哚胺-(2,3)-二氧合酶),IC50为3nm。 | ||||
18433 | IPI-3063 | 1425043-73-7 | >98% | |
IPI-3063是一种选择性的Phosphoinoside-3-激酶p110δ 抑制剂。IPI-3063能有 | ||||
1712292 | 5-碘-1-甲基咪唑 | 71759-88-1 | >98% | |
5-碘-1-甲基咪唑是一种分子砌块。 | ||||
1710123 | 6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-amine | 1448427-99-3 | >98% | |
6-(4-isopropyl-4H-1,2,4-triazol-3-yl)pyridin-2-amine | ||||
179134 | IDRA-21 | 22503-72-6 | 98.0% | |
IDRA-21是一种阳性的AMPA受体调节剂。IDRA-21抑制突触和突触外NMDA受 | ||||
1791118 | ISCK03 | 945526-43-2 | 98.0% | |
ISCK03是一种有效的c-kit抑制剂。ISCK03抑制在501mel人黑素瘤细胞的SC | ||||
1783019 | IACS-9571 | 1800477-30-8 | 98.0% | |
IACS-9571是一种有效的选择性TRIM24和BRPF1抑制剂。布罗莫结构域包括 | ||||
17031013 | Importazole | 662163-81-7 | 98% | |
Importazole是一种运输受体importin-β的小分子抑制剂,专门阻止import | ||||
17030309 | IDE1 | 1160927-48-9 | 98% | |
IDE1是一种高效的细胞渗透性明确内胚层形成诱导剂(EC50 = 125 nM,ESC | ||||
17022713 | ISX-9 | 832115-62-5 | 98% | |
ISX-9 is a neurogenic agent. Isx-9 promotes neurogenesis in vivo, enhancing the proli | ||||
16123024 | Ixazomib (MLN-2238) | 1072833-77-2 | 98% | |
Ixazomib, also known as MLN-2238, is a potent proteasome inhibitor (PI) with potentia | ||||
16123023 | Isovaleramide | 541-46-8 | 98% | |
Isovaleramide, also known as NPS-1776, is a drug potentially for the treatment of mig | ||||
16123022 | Isosorbide Mononitrate | 16051-77-7 | 98% | |
Isosorbide Mononitrate is a drug used principally in the treatment of angina pectoris | ||||
16123021 | IQ-1S | 23146-22-7 | 98% | |
IQ-1S is a potent and selective c-Jun N-Terminal Kinase Inhibitor. IQ-1S inhibits mur | ||||
16123020 | Ingenol Mebutate | 75567-37-2 | 98% | |
Ingenol mebutate, also known as ingenol-3-angelate, is a substance found in the sap o | ||||
16123019 | Imperatorin | 482-44-0 | 98% | |
Imperatorin, aslo known as Pentosalen, Marmelosin, is a furocoumarin and a phytochemi | ||||
16123018 | Iloprost | 78919-13-8 | 98% | |
Iloprost is a drug used to treat pulmonary arterial hypertension (PAH), scleroderma, | ||||
16123017 | IKK-16 | 873225-46-8 | 98% | |
IKK-16 is a potent and slective inhibitor of IB kinase (IKK) (IC50 values are 40, 70 | ||||
16122822 | IDO-IN-1 | 914638-30-5 | 98% | |
IDO-IN-1 is a potent and selective indoleamine-2,3-dioxygenase (IDO) inhibitor with I | ||||
16122821 | Idalopirdine (Lu AE58054) | 467459-31-0 | 98% | |
Idalopirdine, also known as Lu AE58054 or Iladopirdine, is a potent and selective 5-H | ||||
16122820 | IC87201 | 866927-10-8 | 98% | |
IC87201 is a nNOS-PDZ/PSD-95-PDZ inhibitor. IC87201 showed great promise in cellular | ||||
16122741 | ITSA-1 (ITSA1) | 200626-61-5 | 98% | |
ITSA-1 (ITSA1) is an HDAC activator via TSA suppression, but shows no activity toward | ||||
16122729 | 5-Iodotubercidin | 24386-93-4 | 98% | |
5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibi | ||||
6111507 | IMR-1A | 331862-41-0 | 98% | |
IMR-1A is the metabolite of IMR-1. IMR-1 is a novel class of Notch inhibitors targeti |