TCS-OX2-29
编号: 61117
Cas号: 372523-75-6
纯度: 98%
TCS-OX2-29 is a potent and selective OX2 receptor antagonist with IC50 of 40 nM. Displays >250-fold selectivity for OX2 over OX1.
TCS-OX2-29 shows selectivity for ion channels, and transporters (<30% inhibition at 10 M), which includes G-protein coupled receptors associated with food intake including galanin and neuripeptide Y.
TCS-OX2-29 Inhibits orexin A induced IP3 accumulation and ERK1/2 phosphorylation in CHO cells transfected with the OX2 receptor.
仅供研究使用。 我们不向患者出售。
化学信息
| 名称 | TCS-OX2-29 |
|---|---|
| Iupac 化学名称 | TCS-OX2-29 |
| 同义词 | TCS OX2 29 |
| 英文同义词 | TCS OX2 29 |
| 分子式 | C23H31N3O3 |
| 分子量 | 397.51 |
| Smile | CC(C)(C)[C@@H](C(=O)N1CCc2cc(c(cc2C1)OC)OC)NCc3ccncc3.Cl |
| InChiKey | NHKNHFJTMINMBP-ZMBIFBSDSA-N |
| InChi | InChI=1S/C23H31N3O3.ClH/c1-23(2,3)21(25-14-16-6-9-24-10-7-16)22(27)26-11-8-17-12-19(28-4)20(29-5)13-18(17)15-26;/h6-7,9-10,12-13,21,25H,8,11,14-15H2,1-5H3;1H/t21-;/m1./s1 |
| Cas号 | 372523-75-6 |
| MDL | MFCD12828766 |
| 相关CAS号 |
订购信息
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