GDC-0810 ( Brilanestrant , ARN-810 )
Catalog No: 90731
CAS Number: 1365888-06-7
Purity: ≧98.0%
GDC-0810 (Brilanestrant, ARN-810, RG6046) is a selective estrogen receptor degrader (SERD) that is designed to bind to the estrogen receptor to limit its function. In addition, when SERDs bind to the estrogen receptor, they may be able to change the shape of the receptor in such a way that the cell eliminates it by degradation.
仅供研究使用。 我们不向患者出售。
Chemical Information
| Name | GDC-0810 ( Brilanestrant , ARN-810 ) |
|---|---|
| Iupac Chemical Name | (E)-3-(4-((E)-2-(2-chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl)phenyl)acrylic acid |
| Synonyms | Brilanestrant ; GDC-0810 ; GDC 0810 ; GDC0810 ; ARN-810 ; ARN 810 ; ARN810 |
| 英文同义词 | Brilanestrant ; GDC-0810 ; GDC 0810 ; GDC0810 ; ARN-810 ; ARN 810 ; ARN810 |
| Molecular Formula | C26H20ClFN2O2 |
| Molecular Weight | 446.90 |
| Smile | O=C(O)/C=C/C1=CC=C(/C(C2=CC3=C(NN=C3)C=C2)=C(C4=CC=C(F)C=C4Cl)/CC)C=C1 |
| InChiKey | BURHGPHDEVGCEZ-KJGLQBJMSA-N |
| InChi | InChI=1S/C26H20ClFN2O2/c1-2-21(22-10-9-20(28)14-23(22)27)26(18-8-11-24-19(13-18)15-29-30-24)17-6-3-16(4-7-17)5-12-25(31)32/h3-15H,2H2,1H3,(H,29,30)(H,31,32)/b12-5+,26-21+ |
| CAS Number | 1365888-06-7 |
| 相关CAS号 | 1365888-06-7 |
Ordering Information
| 包装 | Price | 库存 | Purity | 备货期 |
|---|---|---|---|---|
| 大货 | Enquiry | Enquiry | Enquiry |
| 外观性状 | Off-white solid to white solid |
|---|---|
| Purity | ≧98.0% |
| Storage | 3 years -20ºCpowder 6 months-80ºCin solvent |
| Solubility | Soluble in DMSO |
| 处理方式 | |
| Shipping Condition | Shipped under ambient temperature |
| 海关编码 |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
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