AT7867 Hcl is a potent ATP-competitive inhibitor of Akt1/2/3 and p70S6K/PKA with
IC50 of 32 nM/17 nM/47 nM and 85 nM/20 nM, respectively; little activity outside
the AGC kinase family.
仅供研究使用。 我们不向患者出售。
化学信息
| 名称 | AT7867 dihydrochloride |
| Iupac 化学名称 | AT 7867 dihydrochloride |
| 同义词 | AT-7867 dihydrochloride; AT 7867 dihydrochloride |
| 英文同义词 | AT-7867 dihydrochloride; AT 7867 dihydrochloride |
| 分子式 | C20H22Cl3N3 |
| 分子量 | 410.77 |
| InChiKey | |
| InChi | |
| Cas号 | 1431697-86-7 |
| 相关CAS号 | |
| 外观性状 | crystalline solid |
| 纯度 | 98% |
| 存储 | 3 years -20℃powder |
| 可溶性 | Soluble in DMSO |
| 处理方式 | |
| 运输条件 | Shipped under ambient temperature as non-hazardous chemical. |
| 海关编码 | |
| Targets | |
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study | |