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产品目录

编号化学名称Cas号纯度化学结构
011309EPZ0156661616391-65-198% 
EPZ-015666 是一种强效、选择性的口服生物药,PRMT5抑制剂与Ki为5 nm
178311EED2262083627-02-398.0%
EED226是一种强效、选择性抑制剂,口服生物EED抑制剂。在EZH2MUT临
651701厄达替尼(JNJ-42756493)1346242-81-698% Min.
Erdafitinib(JNJ-42756493) is a potent and selective panfibroblast growth factor recep
178157Ethyl 2-cyclohexyl-2-oxoacetate13275-31-596.0% 
Ethyl 2-cyclohexyl-2-oxoacetate
178903E74491140964-99-398.0% 
E7449是一种可口服的小分子抑制剂,核酶聚(ADP-核糖)聚合酶(PARP)1和
2017878Elenbecestat ( E2609 )1388651-30-6≧98.0%
Elenbecestat是一种β-Site淀粉样前体蛋白裂解酶BACE)抑制剂,主要用
20178213依托泊苷磷酸酯117091-64-298.0% 
依托泊苷磷酸盐是一种半合成足叶草毒素的磷酸盐。
20178210Elamipretide736992-21-598% 
Elamipretide, 也称为MTP-131或D-Arg-Dmt-Lys-Phe-NH2,是一种心肌过氧化酶抑
20177314[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯388071-27-098.0% 
[(1S)-2-(3,5-二氟苯基)-1-[(2S)-环氧乙烷基]乙基]氨基甲酸叔丁酯
17031018Etrasimod1206123-37-699.73% 
Etrasimod,也被称为APD334,是一种多功能S1P1受体的功能拮抗剂,用
17031010eFT-5081849590-01-798% 
eFT-508 (eFT508)是一种有效且选择性的MNK1 / 2抑制剂,可能导致肿瘤细
17022806盐酸Epetraborole1234563-16-698%
盐酸Epetraborole是一种新型的leucyl - trna合成酶(LeuRS)抑制剂。
17022718依利格鲁司特491833-29-598% 
依利格鲁司特, 也叫Genz-112638, 是一种有效的选择性的葡萄糖酰胺合
17011802EX-527 S-enantiomer848193-68-098% 
EX-527 S-enantiomer是一种有效的选择性SIRT1抑制剂,IC50为123 nM;没有对
17011801EX-527 R-enantiomer848193-69-198% 
EX-527 R-enantiomer是对活性形式EX-527 S-enantiomer(推测为参考)的负控制
170113014E1RCat328998-25-098% 
4E1RCat是eIF4F翻译起始复合物的一种抑制剂,它阻止eIF4E:eIF4G和eIF4E
17011103Etomoxir钠盐828934-41-498% 
Etomoxir是一种在线粒体内膜的外表面的一种不可逆转的CPT-1抑制剂
711401Eganelisib ( IPI-549 )1693758-51-8≧98.0%
Eganelisib (IPI-549) 是一种首创、口服、高选择性 PI3Kγ 抑制剂,单独
16122944Ezutromid945531-77-198% 
Ezutromid, also known as BMN-195 and SMTC-1100, is a first orally bioavailable utroph
16122943EXP-3174124750-92-198% 
EXP-3174, also known as Losartan Carboxylic Acid, is a physiologically active metabol
16122942Ertiprotafib251303-04-598% 
Ertiprotafib, also known as PTP-112, is a Protein Tyrosine Phosphatase 1B Inhibitor (
16122941Eptapirone179756-85-598% 
Eptapirone, also known as F11440, is a potent, selective, high efficacy 5-HT1A recept
16122940Eprodisate Sodium36589-58-998% 
Eprodisate, also known as 3-PDS; NC-503; 3PDS, is an orally available disodium salt f
16122939Emeramide ( BDTH2 )351994-94-0≧98.0%
Emeramide, also known as BDTH2, is a mercury and heavy metal chelator. BDTH2 molecule
16122938EMD534085858668-07-298% 
EMD534085 is a kinesin inhibitor currently in clinical development.
16122811Ellipticine519-23-398% 
Ellipticine is a DNA intercalating agent and a DNA topoisomerase II inhibitor. Ellipt
16122810Elacestrant dihydrochloride1349723-93-8≧98.0%
Elacestrant dihydrochloride, also known as RAD1901, is an orally available, selective
16122767Etravirine (TMC125)269055-15-498% 
Etravirine (TMC125) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used
16122763Efavirenz154598-52-498% 
Efavirenz is a synthetic non-nucleoside reverse transcriptase (RT) inhibitor with ant
16122762Epoxomicin134381-21-898% 
Epoxomicin is a selective proteasome inhibitor with anti-inflammatory activity, inhib