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产品目录

编号化学名称Cas号纯度化学结构
20496BRD4 degrader AT12098836-45-298% Min.
BRD4 degrader AT1 is an analogue of MZ1. It shows improved selectivity for BRD4 degra
20492BJJF0782531244-56-998% Min.
BJJF078 is a potent inhibitor of recombinant human and mouse Transglutaminase enzyme
20485BRD06392760881-74-998% Min.
BRD0639 is a potent PRMT5 inhibitor. BRD0639 engages the target in cells, disrupts PR
230402BI 1015550 ( Nerandomilast )1423719-30-5≧98.0%
BI 1015550 ( Nerandomilast ) 是一种口服磷酸二酯酶 4B (PDE4B) 优先抑制剂
20469BT44924759-42-298% Min.
BT44 is a novel RET agonist for the treatment of experimental neuropathies.
232251Brepocitinib ( PF-06700841 )1883299-62-4≧98.0%
Brepocitinib 是一种潜在的 TYK2 和 JAK1双重选择性抑制剂,IC50 分别为
20453BIIB0681798787-27-598% Min.
20451Baxdrostat1428652-17-898% Min.
Baxdrostat is an aldosterone synthase inhibitor.
20445BMS-9862512114324-48-898% Min.
20444BMS-9861951912445 -55-698% Min.
20428Branebrutinib1912445-55-698% Min.
Branebrutinib, also known as BMS-986195, is a potent, covalent, irreversible inhibito
171680Bexotegrast ( PLN-74809 )2376257-44-0≧98.0%
Bexotegrast(同义词:PLN-74809)是一种小分子、双重选择性 αVβ1 / α
1716534-溴-2-氰基-6-甲氧基吡啶886372-53-8≧95.0%
4-溴-2-氰基-6-甲氧基吡啶, CAS 886372-53-8
1714541-(4-溴-6-甲基吡啶-2-基)乙-1-酮1060810-24-3≧98.0%
1-(4-溴-6-甲基吡啶-2-基)乙-1-酮, CAS 1060810-24-3.
171452BGB 15025 ; BGB-15025 ; BGB150252766481-17-6≧98.0%
BGB-15025 是一种有效的选择性 HPK1 抑制剂,在多种肿瘤模型中作为
20419N-乙基-2-(4-甲酰基苯基)乙酰胺2477812-42-198% Min.
20403 497223-19-5497223-19-598% Min.
20391Benzeneacetic acid, 4-[[(2,4-dimethylbenzoyl)oxy]methyl]-, methyl ester2097334-15-998% Min.
20386497223-19-5497223-19-598% Min.
G203811,10-BIS[4-AZA-1-AZONIABICYCLO[2.2.2]OCTAN-1-YL]DECANE DIBROMIDE94630-53-298% Min.
203726-(苄氧基)-3,4-二氢萘-2(1H)-酮885280-42-298% Min.
L20357BIBF0775334951-90-598% Min.
BIBF0775 is an inhibitor of the transforming growth factor β receptor I (TGFβRI). X
6111905Blarcamesine HCl195615-84-098% Min.
Anavex2-73 is a muscarinic/σ1 ligand. ANAVEX2-73 (0.01-3.0 mg/kg i.p.) alleviated th
20271Bunamidine hydrochloride1055-55-698% Min.
Bunamidine is a anti-parasitic drug, which was approved by FDA for the treatment of t
20270BIT225917909-71-898% Min.
BIT-225 is a NCp7 zinc finger inhibitor potentially for the treatment of HCV infectio
21234BI-34062230836-55-098% Min.
BI-3406 is Potent & Selective SOS1::KRAS Inhibitor (IC50=5 nM), which Opens a New
21224 BI-1870041303515-32-3≧98.0%
BI-187004, also known as VTP-34072, is an 11β-hydroxysteroid dehydrogenase 1 inhibit
2021221Bafetinib887650-05-798% Min.
Bafetinib, also known as INNO-406 and NS187, is an orally bioavailable 2-phenylaminop
202112701BRD07052056261-41-598% Min.
BRD0705 is a potent, paralog selective and orally active GSK3α inhibitor. BRD0705 ca
20121701 BLU-7822141955-96-498% Min.