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Proteases

Catalog NoChemical NameCAS NumberPurityChemical Structure
25149Safusidenib1898206-17-1≧98.0%
Safusidenib, also known as DS-1001, is an oral isocitrate dehydrogenase [NADP] cytopl
25176AG-2702201056-66-6≧98.0%
MAT2A Inhibitor AG-270 is an orally available small molecule inhibitor of methionine
24101Crelosidenib2230263-60-0≧98.0%
Crelosidenib is an isocitrate dehydrogenase 1 (IDH1) inhibitor.
24031GW-280264 ( GW-280264X )866924-39-2≧98.0%
GW-280264 ( GW-280264X ) is the mixedADAM10/TACE (ADAM17) metalloproteinasesinhibitor.
24108JHU-0831998725-11-3≧98.0%
JHU-083 selectively blocks glutaminase activity in brain CD11b+ cells and prevents de
24109CBR-5884681159-27-3≧98.0%
CBR 5884 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor which was able to inhi
25147MAT2A-IN-9 ( GSK4362676 )2439277-80-0≧98.0%
MAT2A-IN-9 ( GSK4362676 ), is a 2-oxoquinazoline derivative, is a potent MAT2A (methi
25150Ranosidenib2301974-60-5≧98.0%
Ranosidenib, also known as HMPL-306, is an isocitrate dehydrogenase (IDH) inhibitor.
25155PF-078535783036158-98-9≧98.0%
PF-07853578 is a Patatin-Like Phospholipase Domain-Containing 3 Protein (PNPLA3) modu
25178DS-1001b1898207-64-1≧98.0%
DS-1001 is an oral brain-penetrant mutant IDH1 selective inhibitor.