Timapiprant,又名OC000459,是一种强效、选择性和口服的CRTH2拮抗剂。OC000459减少了对花粉过敏的受试者的鼻和眼症状,这是一种随机、安慰剂对照、双盲试验。
For research use only. We do not sell to patients.
| Name | Timapiprant |
|---|---|
| Iupac Chemical Name | 2-(5-fluoro-2-methyl-3-(quinolin-2-ylmethyl)-1H-indol-1-yl)acetic acid |
| Synonyms | OC000459; OC-000459; OC 000459; Timapiprant. |
| Molecular Formula | C21H17FN2O2 |
| Molecular Weight | 348.3774 |
| Smile | O=C(O)CN1C(C)=C(CC2=NC3=CC=CC=C3C=C2)C4=C1C=CC(F)=C4 |
| InChiKey | FATGTHLOZSXOBC-UHFFFAOYSA-N |
| InChi | InChI=1S/C21H17FN2O2/c1-13-17(11-16-8-6-14-4-2-3-5-19(14)23-16)18-10-15(22)7-9-20(18)24(13)12-21(25)26/h2-10H,11-12H2,1H3,(H,25,26) |
| CAS Number | 851723-84-7 |
| Related CAS |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | 白色粉末 |
|---|---|
| Purity | >98% |
| Storage | 短期可在0-4度保存,数天至数月;长期可在-20度保存三年。 |
| Solubility | 可溶于DMSO |
| Handling | |
| Shipping Condition | 可在常温下运输 |
| HS Code |
| Targets | |
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| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |