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TCS-OX2-29

Catalog No: 61117
CAS Number: 372523-75-6
Purity: 98% 

TCS-OX2-29 is a potent and selective OX2 receptor antagonist with IC50 of 40 nM. Displays >250-fold selectivity for OX2 over OX1. 

TCS-OX2-29 shows selectivity for ion channels, and transporters (<30% inhibition at 10 M), which includes G-protein coupled receptors associated with food intake including galanin and neuripeptide Y. 
TCS-OX2-29 Inhibits orexin A induced IP3 accumulation and ERK1/2 phosphorylation in CHO cells transfected with the OX2 receptor.

 

For research use only. We do not sell to patients.

Chemical Information

NameTCS-OX2-29
Iupac Chemical NameTCS-OX2-29 
SynonymsTCS OX2 29 
Molecular FormulaC23H31N3O3 
Molecular Weight397.51 
SmileCC(C)(C)[C@@H](C(=O)N1CCc2cc(c(cc2C1)OC)OC)NCc3ccncc3.Cl
InChiKeyNHKNHFJTMINMBP-ZMBIFBSDSA-N
InChiInChI=1S/C23H31N3O3.ClH/c1-23(2,3)21(25-14-16-6-9-24-10-7-16)22(27)26-11-8-17-12-19(28-4)20(29-5)13-18(17)15-26;/h6-7,9-10,12-13,21,25H,8,11,14-15H2,1-5H3;1H/t21-;/m1./s1
CAS Number372523-75-6
MDLMFCD12828766
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Ordering Information

PackagingPriceAvailabilityPurityShipping Time
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Formulationcrystalline solid 
Purity98% 
Storage3 years -20&ordm;Cpowder 
SolubilitySoluble in DMSO 
Handling
Shipping ConditionShipped under ambient temperature as non-hazardous chemical. 
HS Code
Coming soon.
Targets
Mechanism
Cell study
Animal study
Clinical study
Not available

Chemical Structure

61117 - TCS-OX2-29 | CAS 372523-75-6

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