Balipodect (TAK 063 ) is a novel PDE10A inhibitor. It has shown high inhibitory activity and selectivity for human recombinant PDE10A2 in vitro; the half-maximal inhibitory concentration was 0.30 nM, and selectivity over other phosphodiesterases (PDEs) was more than 15000-fold.
Balipodect (TAK 063 ), Bulk in stock,
For research use only. We do not sell to patients.
| Name | Balipodect ( TAK-063 ) |
|---|---|
| Iupac Chemical Name | 1-(2-fluoro-4-(1H-pyrazol-1-yl)phenyl)-5-methoxy-3-(1-phenyl-1H-pyrazol-5-yl)pyridazin-4(1H)-one |
| Synonyms | TAK063 ;TAK 063 ; Balipodect. |
| Molecular Formula | C23H17FN6O2 |
| Molecular Weight | 428.42 |
| Smile | O=C1C(C2=CC=NN2C3=CC=CC=C3)=NN(C4=CC=C(N5N=CC=C5)C=C4F)C=C1OC |
| InChiKey | KVHRYLNQDWXAGI-UHFFFAOYSA-N |
| InChi | InChI=1S/C23H17FN6O2/c1-32-21-15-29(19-9-8-17(14-18(19)24)28-13-5-11-25-28)27-22(23(21)31)20-10-12-26-30(20)16-6-3-2-4-7-16/h2-15H,1H3 |
| CAS Number | 1238697-26-1 |
| Related CAS | 1238697-26-1 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Light-yellow powder |
|---|---|
| Purity | 98% |
| Storage | -20 ºC for 3 years |
| Solubility | Soluble in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
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| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |