SB-742457(Intepirdine) is a highly selective 5-HT6 receptor antagonist with pKi of 9.63; exhibits >100-fold selectivity over other receptors.
For research use only. We do not sell to patients.
| Name | SB-742457 ( Intepirdine ) |
|---|---|
| Iupac Chemical Name | 3-(benzenesulfonyl)-8-piperazin-1-ylquinoline |
| Synonyms | GSK-742457 ; RVT-101 ; Intepirdine ; SB-742457 ; SB742457 |
| Molecular Formula | C19H19N3O2S |
| Molecular Weight | 353.438 |
| Smile | C1CN(CCN1)C2=CC=CC3=CC(=CN=C32)S(=O)(=O)C4=CC=CC=C4 |
| InChiKey | JJZFWROHYSMCMU-UHFFFAOYSA-N |
| InChi | InChI=1S/C19H19N3O2S/c23-25(24,16-6-2-1-3-7-16)17-13-15-5-4-8-18(19(15)21-14-17)22-11-9-20-10-12-22/h1-8,13-14,20H,9-12H2 |
| CAS Number | 607742-69-8 |
| Related CAS | 607742-69-8 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Light-yellow solid |
|---|---|
| Purity | 98% |
| Storage | -20 ºC for 3 years |
| Solubility | Soluble in DMSO |
| Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |