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Remibrutinib ( LOU064 )

Catalog No.: 2073103
Cas No.: 1787294-07-8
Purity : 98% Min.

Remibrutinib ( LOU064 ) is a Potent and Highly Selective Covalent Inhibitor of Bruton’s Tyrosine Kinase. Remibrutinib ( LOU064 ) exhibits an exquisite kinase selectivity due to binding to an inactive conformation of BTK and has the potential for a best-in-class covalent BTK inhibitor for the treatment of autoimmune diseases. It demonstrates potent in vivo target occupancy with an EC90 of 1.6 mg/kg and dose-dependent efficacy in rat collagen-induced arthritis. Remibrutinib ( LOU064 ) is currently being tested in phase 2 clinical studies for chronic spontaneous urticaria and Sjoegren’s syndrome.

For research use only. We do not sell to patients.

Chemical Information

NameRemibrutinib ( LOU064 )
Iupac Chemical NameN-(3-(6-amino-5-(2-(N-methylacrylamido)ethoxy)pyrimidin-4-yl)-5-fluoro-2-methylphenyl)-4-cyclopropyl-2-fluorobenzamide
SynonymsRemibrutinib ; LOU064 ; LOU 064 ; LOU-064
Molecular FormulaC27H27F2N5O3
Molecular Weight507.53
CAS Number1787294-07-8
Related CAS1787294-07-8

Ordering Information

PackagingPriceAvailabilityPurityShipping Time
Request Bulk Quote Download MSDS Tel : +86-27-65522453   Email : sales@sun-shinechem.com
FormulationOff-white solid to white solid
Purity98% Min.
StorageDry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).
SolubilitySoluble in DMSO
Shipping ConditionShipped under ambient temperature 
HS Code
Coming soon.
Cell study
Animal study
Clinical study
Not available

Chemical Structure

2073103 - Remibrutinib ( LOU064 ) | CAS 1787294-07-8

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