Prifetrastat
Catalog No: 26A088
CAS Number: 2569008-99-5
Purity: ≧98.0%
Prifetrastat (also known as PF 07248144) is a small molecule KAT6A/B inhibitor.
For research use only. We do not sell to patients.
Chemical Information
| Name | Prifetrastat |
|---|---|
| Iupac Chemical Name | N-(6-((1H-pyrazol-1-yl)methyl)-4-methoxybenzo[d]isoxazol-3-yl)-2-methoxybenzenesulfonamide |
| Synonyms | Prifetrastat; PF-07248144; PF 07248144; PF07248144 |
| Molecular Formula | C19H18N4O5S |
| Molecular Weight | 414.44 |
| Smile | O=S(C1=CC=CC=C1OC)(NC2=NOC3=CC(CN4N=CC=C4)=CC(OC)=C23)=O |
| InChiKey | RCBWSTJGOASLEO-UHFFFAOYSA-N |
| InChi | InChI=1S/C19H18N4O5S/c1-26-14-6-3-4-7-17(14)29(24,25)22-19-18-15(27-2)10-13(11-16(18)28-21-19)12-23-9-5-8-20-23/h3-11H,12H2,1-2H3,(H,21,22) |
| CAS Number | 2569008-99-5 |
| Related CAS | 2569008-99-5 |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
| Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
| Handling | Refer to MSDS |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
Coming soon.
| Targets | KAT6A protein inhibitors |
|---|---|
| Mechanism | KAT6A protein inhibitors; KAT6B protein inhibitors |
| Cell study | |
| Animal study | |
| Clinical study | Phase III : HER2 negative breast cancer |
Not available
Chemical Structure
