Oveporexton is an oral small molecule selective orexin type-2 receptor (OX2R) agonist.
For research use only. We do not sell to patients.
| Name | Oveporexton ( TAK-861 ) |
|---|---|
| Iupac Chemical Name | N-((2S,3R)-4,4-difluoro-1-(2-hydroxy-2-methylpropanoyl)-2-((2,3',5'-trifluoro-[1,1'-biphenyl]-3-yl)methyl)pyrrolidin-3-yl)ethanesulfonamide |
| Synonyms | Oveporexton ; TAK-861 ; TAK861 ; TAK 861 |
| Molecular Formula | C23H25F5N2O4S |
| Molecular Weight | 520.52 |
| Smile | CCS(=O)(N[C@@H]1[C@H](CC2=C(F)C(C3=CC(F)=CC(F)=C3)=CC=C2)N(C(C(C)(O)C)=O)CC1(F)F)=O |
| InChiKey | KVMGAIOTUIGROS-AZUAARDMSA-N |
| InChi | InChI=1S/C23H25F5N2O4S/c1-4-35(33,34)29-20-18(30(12-23(20,27)28)21(31)22(2,3)32)10-13-6-5-7-17(19(13)26)14-8-15(24)11-16(25)9-14/h5-9,11,18,20,29,32H,4,10,12H2,1-3H3/t18-,20+/m0/s1 |
| CAS Number | 2460722-04-5 |
| Related CAS | 2460722-04-5 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
| Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
| Handling | Refer to MSDS |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |