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MLN-1117

Catalog No.: 17030101
Cas No.: 1268454-23-4
Purity : 98% 
17030101 - MLN-1117 | CAS 1268454-23-4

Catalog number : 17030101

CAS number : 1268454-23-4

Molecular Formula : C19H17N5O3 

Molecular Weight : 363.377 

Iupac Chemical Name : [6-(2-amino-5-benzoxazolyl)imidazo[1,2-a]pyridin-3-yl]-4-morpholinyl-methanone 

Smile : NC=1OC2=C(N1)C=C(C=C2)C=2C=CC=1N(C2)C(=CN1)C(=O)N1CCOCC1

InChiKey : BLGWHBSBBJNKJO-UHFFFAOYSA-N

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SynonymsINK1117; INK-1117; INK 1117; MLN1117; MLN 1117; MLN-1117; TAK-117; TAK 117; TAK117 
Molecular FormulaC19H17N5O3 
Molecular Weight363.377 
Appearanceoff-white solid 
Purity98% 
SolubilitySoluble in DMSO 
Storage3 years -20ºCpowder 
Shipping ConditionShipped under ambient temperature as non-hazardous chemical. 
SmileNC=1OC2=C(N1)C=C(C=C2)C=2C=CC=1N(C2)C(=CN1)C(=O)N1CCOCC1
InChiKeyBLGWHBSBBJNKJO-UHFFFAOYSA-N
InChiInChI=1S/C19H17N5O3/c20-19-22-14-9-12(1-3-16(14)27-19)13-2-4-17-21-10-15(24(17)11-13)18(25)23-5-7-26-8-6-23/h1-4,9-11H,5-8H2,(H2,20,22)
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Serabelisib (also known as MLN1117, INK1117, and TAK-117) is an orally bioavailable inhibitor of the class I phosphoinositide 3-kinase (PI3K) alpha isoform with potential antineoplastic activity. PI3K alpha inhibitor INK1117 selectively inhibits PI3K alpha kinase, including mutations of PIK3CA, in the PI3K/Akt/mTOR pathway, which may result in tumor cell apoptosis and growth inhibition in PI3K alpha-expressing tumor cells. By specifically targeting class I PI3K alpha, this agent may be more efficacious and less toxic than pan-PI3K inhibitors. 

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