Lemborexant(CAS 1369764-02-2)is a novel investigational small molecule that inhibits orexin signaling by binding competitively to both orexin receptor subtypes (orexin receptor 1 and 2).
Lemborexant (E-2006), Bulk in stock, contact us by email for the quotation. Kg scale intermediates are also be provided by custom synthesis.
For research use only. We do not sell to patients.
| Name | Lemborexant (E-2006) |
|---|---|
| Iupac Chemical Name | (1R,2S)-2-(((2,4-dimethylpyrimidin-5-yl)oxy)methyl)-2-(3-fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropanecarboxamide |
| Synonyms | E-2006; E 2006; E2006; Lemborexant ; Dayvigo |
| Molecular Formula | C22H20F2N4O2 |
| Molecular Weight | 410.1554 |
| Smile | FC1=CC=CC([C@@]2(COC3=CN=C(C)N=C3C)[C@H](C(NC4=CC=C(F)C=N4)=O)C2)=C1 |
| InChiKey | MUGXRYIUWFITCP-PGRDOPGGSA-N |
| InChi | InChI=1S/C22H20F2N4O2/c1-13-19(11-25-14(2)27-13)30-12-22(15-4-3-5-16(23)8-15)9-18(22)21(29)28-20-7-6-17(24)10-26-20/h3-8,10-11,18H,9,12H2,1-2H3,(H,26,28,29)/t18-,22+/m0/s1 |
| CAS Number | 1369764-02-2 |
| Related CAS |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Off-white solid |
|---|---|
| Purity | 98% Min. |
| Storage | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| Solubility | Soluble in DMSO, not in water |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
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| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |