Lazertinib is a an orally available third-generation, selective inhibitor of certain forms of the epidermal growth factor receptor (EGFR) .
For research use only. We do not sell to patients.
| Name | Lazertinib mesylate |
|---|---|
| Iupac Chemical Name | N-(5-((4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yl)pyrimidin-2-yl)amino)-4-methoxy-2-morpholinophenyl)acrylamide methanesulfonate |
| Synonyms | lazertinib mesylate |
| Molecular Formula | C30H34N8O3*CH4O3S |
| Molecular Weight | 650.759 |
| Smile | C=CC(NC1=CC(NC2=NC=CC(N3N=C(C4=CC=CC=C4)C(CN(C)C)=C3)=N2)=C(OC)C=C1N5CCOCC5)=O.CS(=O)(O)=O |
| InChiKey | BXBUSQVSAAMGMR-UHFFFAOYSA-N |
| InChi | InChI=1S/C30H34N8O3.CH4O3S/c1-5-28(39)32-23-17-24(26(40-4)18-25(23)37-13-15-41-16-14-37)33-30-31-12-11-27(34-30)38-20-22(19-36(2)3)29(35-38)21-9-7-6-8-10-21;1-5(2,3)4/h5-12,17-18,20H,1,13-16,19H2,2-4H3,(H,32,39)(H,31,33,34);1H3,(H,2,3,4) |
| CAS Number | 2247995-37-3 |
| Related CAS | 2247995-37-3 ; 2867596-17-4 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Off-white solid |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
| Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
| Handling | Refer to MSDS |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |