HUHS015
Catalog No: 16062902
CAS Number: 1453097-13-6
Purity: 98% by HPLC
HUHS015 is a potent PCA-1/ALKBH3 inhibitor both in vitro and in vivo. The bioavailability (BA) of HUHS015 was 7.2% in rats after oral administration. As expected, continuously administering HUHS015 significantly suppressed the growth of DU145 cells, which are human hormone-independent prostate cancer cells, in a mouse xenograft model without untoward effects.
For research use only. We do not sell to patients.
Chemical Information
| Name | HUHS015 |
|---|---|
| Iupac Chemical Name | 4-benzyl-3-methyl-1-(5-methyl-1H-benzo[d]imidazol-2-yl)-1H-pyrazol-5-ol |
| Synonyms | HUHS 015;HUHS-015 |
| Molecular Formula | C19H18N4O |
| Molecular Weight | 318.37242 |
| Smile | C(C1=CC=CC=C1)C=1C(=NN(C1O)C1=NC2=C(N1)C=CC(=C2)C)C |
| InChiKey | LFEFEOLVKXXVGD-UHFFFAOYSA-N |
| InChi | InChI=1S/C19H18N4O/c1-12-8-9-16-17(10-12)21-19(20-16)23-18(24)15(13(2)22-23)11-14-6-4-3-5-7-14/h3-10,24H,11H2,1-2H3,(H,20,21) |
| CAS Number | 1453097-13-6 |
| Related CAS |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | 98% by HPLC |
| Storage | -20 ºC for 3 years |
| Solubility | Soluble in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
