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Giredestrant tartrate

Catalog No: 20263
CAS Number: 2407529-33-1
Purity: ≧98.0%

Giredestrant tartrate (GDC-9545 tartrate), a non-steroidal ER ligand, is an orally active and selective estrogen receptor (ER) antagonist. Giredestrant tartrate potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain.

For research use only. We do not sell to patients.

Chemical Information

NameGiredestrant tartrate
Iupac Chemical Name3-((1R,3R)-1-(2,6-difluoro-4-((1-(3-fluoropropyl)azetidin-3-yl)amino)phenyl)-3-methyl-1,3,4,9-tetrahydro-2H-pyrido[3,4-b]indol-2-yl)-2,2-difluoropropan-1-ol (2R,3R)-2,3-dihydroxysuccinate
SynonymsGiredestrant tartrate ; GDC-9545 tartrate ; GDC9545 tartrate ; GDC 9545 tartrate ; RG6171 tartrate ; RG-6171 tartrate ; RG 6171 tartrate ; Giredestrant ;
Molecular FormulaC31H37F5N4O7
Molecular Weight672.64
SmileC[C@H](C1)N(CC(F)(F)CO)[C@H](C2=C(F)C=C(NC3CN(CCCF)C3)C=C2F)C4=C1C5=C(N4)C=CC=C5.OC([C@H](O)[C@@H](O)C(O)=O)=O
InChiKeyQZOTWXMHTSEIJY-WULFPPIKSA-N
InChiInChI=1S/C27H31F5N4O.C4H6O6/c1-16-9-20-19-5-2-3-6-23(19)34-25(20)26(36(16)14-27(31,32)15-37)24-21(29)10-17(11-22(24)30)33-18-12-35(13-18)8-4-7-28;5-1(3(7)8)2(6)4(9)10/h2-3,5-6,10-11,16,18,26,33-34,37H,4,7-9,12-15H2,1H3;1-2,5-6H,(H,7,8)(H,9,10)/t16-,26-;1-,2-/m11/s1
CAS Number2407529-33-1
Related CAS1953133-47-5

Ordering Information

PackagingPriceAvailabilityPurityShipping Time
BulkEnquiryEnquiryEnquiry
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Formulation黄色固体粉末
Purity≧98.0%
Storage短期(几天到几周)为0-4摄氏度,长期(几个月)为-20摄氏度
Solubility溶于DMSO
HandlingAvoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation.
Shipping Condition作为非危险化学品在环境温度下装运。这种产品在正常运输和海关工作期间可以稳定几周.
HS Code
Coming soon.
Targets
Mechanism
Cell study
Animal study
Clinical study
Not available

Chemical Structure

20263 - Giredestrant tartrate | CAS 2407529-33-1

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