Galunisertib(LY2157299)
Catalog No: 52017
CAS Number: 700874-72-2
Purity: 98%
Galunisertib (LY2157299) is selective TGF- receptor kinase inhibitor. Galunisertib was found to inhibit the growth in an in vitro clonogenic assay in 6.3% (5/79) of the examined PDX.
For research use only. We do not sell to patients.
Chemical Information
| Name | Galunisertib(LY2157299) |
|---|---|
| Iupac Chemical Name | 4-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinoline-6-carboxamide |
| Synonyms | Galunisertib,LY2157299,LY-2157299,LY 2157299 |
| Molecular Formula | C22H19N5O |
| Molecular Weight | 369.42 |
| Smile | CC1=CC=CC(=N1)C=1C(=C2N(N1)CCC2)C2=CC=NC1=CC=C(C=C21)C(=O)N |
| InChiKey | IVRXNBXKWIJUQB-UHFFFAOYSA-N |
| InChi | InChI=1S/C22H19N5O/c1-13-4-2-5-18(25-13)21-20(19-6-3-11-27(19)26-21)15-9-10-24-17-8-7-14(22(23)28)12-16(15)17/h2,4-5,7-10,12H,3,6,11H2,1H3,(H2,23,28) |
| CAS Number | 700874-72-2 |
| Related CAS |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | off-white solid |
|---|---|
| Purity | 98% |
| Storage | 3 years -20ºCpowder |
| Solubility | 5mg/ml in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
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