GSK3787 is as a selective and irreversible antagonist of PPAR with pIC50 of 6.6, with no measurable affinity for hPPAR or hPPAR.
For research use only. We do not sell to patients.
| Name | GSK3787 |
|---|---|
| Iupac Chemical Name | Benzamide, 4-chloro-N-[2-[[5-(trifluoromethyl)-2-pyridinyl]sulfonyl]ethyl]- |
| Synonyms | N/A |
| Molecular Formula | C15H12ClF3N2O3S |
| Molecular Weight | 392.78 |
| Smile | ClC1=CC=C(C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)C=C1 |
| InChiKey | JFUIMTGOQCQTPF-UHFFFAOYSA-N |
| InChi | InChI=1S/C15H12ClF3N2O3S/c16-12-4-1-10(2-5-12)14(22)20-7-8-25(23,24)13-6-3-11(9-21-13)15(17,18)19/h1-6,9H,7-8H2,(H,20,22) |
| CAS Number | 188591-46-0 |
| Related CAS |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | off-white solid |
|---|---|
| Purity | 98% |
| Storage | 3 years -20ºCpowder |
| Solubility | 2mg/ml in DMSO |
| Handling | |
| Shipping Condition | Shipped under ambient temperature |
| HS Code |
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |