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GDC-0810(Brilanestrant,ARN-810)

Catalog No.: 90731
Cas No.: 1365888-06-7
Purity : 98% by HPLC 
90731 - GDC-0810(Brilanestrant,ARN-810) | CAS 1365888-06-7

Catalog number : 90731

CAS number : 1365888-06-7

Molecular Formula : C26H20ClFN2O2 

Molecular Weight : 446.90 

Iupac Chemical Name : (E)-3-(4-((E)-2-(2-chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl)phenyl)acrylic acid 

Smile : O=C(O)/C=C/C1=CC=C(/C(C2=CC3=C(NN=C3)C=C2)=C(C4=CC=C(F)C=C4Cl)/CC)C=C1

InChiKey : BURHGPHDEVGCEZ-KJGLQBJMSA-N

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SynonymsBrilanestrant;GDC-0810;GDC 0810;GDC0810;ARN-810;ARN 810;ARN810 
Molecular FormulaC26H20ClFN2O2 
Molecular Weight446.90 
Appearancecrystalline solid 
Purity98% by HPLC 
SolubilitySoluble in DMSO 
Storage3 years -20ºCpowder 6 months-80ºCin solvent 
Shipping ConditionShipped under ambient temperature 
SmileO=C(O)/C=C/C1=CC=C(/C(C2=CC3=C(NN=C3)C=C2)=C(C4=CC=C(F)C=C4Cl)/CC)C=C1
InChiKeyBURHGPHDEVGCEZ-KJGLQBJMSA-N
InChiInChI=1S/C26H20ClFN2O2/c1-2-21(22-10-9-20(28)14-23(22)27)26(18-8-11-24-19(13-18)15-29-30-24)17-6-3-16(4-7-17)5-12-25(31)32/h3-15H,2H2,1H3,(H,29,30)(H,31,32)/b12-5+,26-21+
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GDC-0810 (Brilanestrant, ARN-810, RG6046) is a selective estrogen receptor degrader (SERD) that is designed to bind to the estrogen receptor to limit its function. In addition, when SERDs bind to the estrogen receptor, they may be able to change the shape of the receptor in such a way that the cell eliminates it by degradation.

Mechanism of Action / Target

Selective estrogen receptor degrader

 

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