Elinzanetant ( NT-814 )
编号: 20259
Cas号: 929046-33-3
纯度: ≧98.0%
Elinzanetant, previously known as NT-814 (45), is a dual NK1,3R antagonist and therefore has the potential to reduce GnRH pulsatility by blocking the endogenous effects of NKB and SP on the reproductive axis.
For research use only. We do not sell to patients.
化学信息
| 名称 | Elinzanetant ( NT-814 ) |
|---|---|
| Iupac 化学名称 | 2-[3,5-bis(trifluoromethyl)phenyl]-N-{4-(4-fluoro-2-methylphenyl)-6-[(7S,9aS)-7-(hydroxymethyl)hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl]pyridin-3-yl}-N,2-dimethylpropanamide |
| 同义词 | Elinzanetant ; GSK1144814A ; NT-814 ; NT 814 ; NT814 ; GSK-1144814A ; GSK 1144814A |
| 分子式 | C33H35F7N4O3 |
| 分子量 | 668.64 |
| Smile | CC(C)(C1=CC(C(F)(F)F)=CC(C(F)(F)F)=C1)C(N(C2=C(C3=CC=C(F)C=C3C)C=C(N4C[C@@]5([H])COCCN5C[C@H]4CO)N=C2)C)=O |
| InChiKey | DWRIJNIPBUFCQS-DQEYMECFSA-N |
| InChi | InChI=1S/C33H35F7N4O3/c1-19-9-23(34)5-6-26(19)27-13-29(44-16-25-18-47-8-7-43(25)15-24(44)17-45)41-14-28(27)42(4)30(46)31(2,3)20-10-21(32(35,36)37)12-22(11-20)33(38,39)40/h5-6,9-14,24-25,45H,7-8,15-18H2,1-4H3/t24-,25-/m0/s1 |
| Cas号 | 929046-33-3 |
| Related CAS | 929046-33-3 |
订购信息
| Packaging | 价格 | Availability | 纯度 | Shipping Time |
|---|---|---|---|---|
| Bulk | 询价 | 询价 | 询价 |
| Formulation | Off-white Solid |
|---|---|
| 纯度 | ≧98.0% |
| 存储 | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
| 可溶性 | Soluble in DMSO |
| Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| 运输条件 | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
