CVN-424 (Solengepras) is a first-in-class, small molecule GPR6 inverse agonist.
For research use only. We do not sell to patients.
| Name | CVN-424 ( Solangepras ) |
|---|---|
| Iupac Chemical Name | (R)-1-(2-(4-(2,4-difluorophenoxy)piperidin-1-yl)-3-((tetrahydrofuran-3-yl)amino)-7,8-dihydropyrido[3,4-b]pyrazin-6(5H)-yl)ethan-1-one |
| Synonyms | CVN-424 ; Solangepras ; CVN 424 ; CVN424 |
| Molecular Formula | C24H29F2N5O3 |
| Molecular Weight | 473.22 |
| Smile | CC(N1CCC2=NC(N3CCC(OC4=CC=C(F)C=C4F)CC3)=C(N[C@H]5COCC5)N=C2C1)=O |
| InChiKey | HSWVJQBEXRKOBZ-QGZVFWFLSA-N |
| InChi | InChI=1S/C24H29F2N5O3/c1-15(32)31-10-6-20-21(13-31)28-23(27-17-7-11-33-14-17)24(29-20)30-8-4-18(5-9-30)34-22-3-2-16(25)12-19(22)26/h2-3,12,17-18H,4-11,13-14H2,1H3,(H,27,28)/t17-/m1/s1 |
| CAS Number | 2254706-21-1 |
| Related CAS | 2254706-21-1 |
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Solid powder |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years). |
| Solubility | Soluble in DMSO (DMSO : ≥ 100 mg/mL) |
| Handling | Refer to MSDS |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
| Targets | GPR6 inverse agonist |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |