AGN 196996
Catalog No: 226191
CAS Number: 958295-17-5
Purity: ≧98.0%
AGN 196996 is a potent and selective RARα antagonist with Ki value of 2 nM; little binding affinity for RARβ(Ki=1087 nM) and RARγ(Ki=8523 nM).
For research use only. We do not sell to patients.
Chemical Information
| Name | AGN 196996 |
|---|---|
| Iupac Chemical Name | 4-(3-bromo-4-ethoxy-5-(4-methylbenzoyl)benzamido)benzoic acid |
| Synonyms | AGN 196996 ; AGN-196996 ; AGN196996 ; |
| Molecular Formula | C24H20BrNO5 |
| Molecular Weight | 482.33 |
| Smile | O=C(O)C1=CC=C(NC(C2=CC(C(C3=CC=C(C)C=C3)=O)=C(OCC)C(Br)=C2)=O)C=C1 |
| InChiKey | BUGXGZOGQGUTBC-UHFFFAOYSA-N |
| InChi | InChI=1S/C24H20BrNO5/c1-3-31-22-19(21(27)15-6-4-14(2)5-7-15)12-17(13-20(22)25)23(28)26-18-10-8-16(9-11-18)24(29)30/h4-13H,3H2,1-2H3,(H,26,28)(H,29,30) |
| CAS Number | 958295-17-5 |
| Related CAS | 958295-17-5 |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | Off-white solid to white powder |
|---|---|
| Purity | ≧98.0% |
| Storage | Dry, dark and at 0-4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
| Solubility | Soluble in CDCl3, MeOH etc. |
| Handling | Refer to MSDS operation |
| Shipping Condition | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
| HS Code | 2934200090 |
| Targets | RARα antagonist |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
