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Inhibitors & Agonists

CATALOG NOPRODUCT NAMECASPURITYSTRUCTURE
101205Temsirolimus162635-04-398% 
Temsirolimus is a recently developed mTOR inhibitor. with improved aqueous solubility
101207TP-0903(Dubermatinib)1341200-45-098% 
TP-0903 is a potent and selective Axl kinase inhibitor with IC50 of 27 nM.
101901SCR-1481B11174161-69-398% 
SCR-1481B1 is a potent and selective MET inhibitor. SCR-1481B1 inhibited MET kinase w
111016VPS34-IN11383716-33-398% by HPLC/HNMR 
VPS34-IN1 is a selective inhibitor of Vps34.
120101A661166227-08-298% 
A66 is a potent and specific p110 inhibitor with IC50 of 32 nM, >100 fold selectiv
120115GDC-0941957054-30-798% 
GDC-0941 is a potent inhibitor of PI3K/ with IC50 of 3 nM, with modest selectivity ag
121418PHA-665752 hydrate477575-56-798% 
PHA-665752 is a potent, selective and ATP-competitive c-Met inhibitor with IC50 of 9
121420Torkinib1092351-67-198% 
PP242 is a selective mTOR inhibitor with IC50 of 8 nM; targets both mTOR complexes wi
121421PKI-4021173204-81-398% 
PKI-402 is a potent dual pan-PI3K/mTOR inhibitor targeting PI3K/// and mTOR with IC50
121424Ku-0063794938440-64-398% 
KU-0063794 is a selective inhibitor of mammalian target of rapamycin (mTOR) (IC50 ~10
121426YM-201636371942-69-798% 
YM201636 is a selective PIKfyve inhibitor with IC50 of 33 nM, less potent to p110.
122908PI-3065955977-50-198% 
PI-3065 is a novel potent and selective PI3K p110 inhibitor with IC50 of 15 nM; exhib