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Inhibitors & Agonists

CATALOG NOPRODUCT NAMECASPURITYSTRUCTURE
51801UNC03791620401-82-298% 
UNC0379 is a selective, substrate competitive inhibitor ofN-lysine methyltransferase
51705Foretinib(GSK1363089)849217-64-798% 
Foretinib (GSK1363089) is an ATP-competitive inhibitor of HGFR and VEGFR, mostly forM
51606CH5424802 Hydrochloride1256589-74-898% 
CH5424802 Hcl (AF 802 Hcl; Alectinib Hcl) is a potent ALK inhibitor with IC50 of 1.9
52207BKM120(NVP-BKM120, Buparlisib)944396-07-098% 
BKM120(NVP-BKM120, Buparlisib) is an orally bioavailable specific oral inhibitor of t
52215GNE-3171394076-92-698% 
GNE-317 is a potent, brain-penetrantPI3Kinhibitor
52309LY294002154447-36-698% 
LY294002 is the first synthetic molecule known to inhibitPI3K//withIC50of 0.5 M/0.57
51612Filgotinib1206161-97-898% 
Filgotinib (GLPG0634) is a selective JAK1 inhibitor with IC50 of 10 nM, 28 nM, 810 nM
51805GSK5031346572-63-198% 
GSK-503 is a potent EZH2 inhibitor with potential anticancer activity. Reference: 1.
52208GSK1261346574-57-998% 
GSK126 is a potent, highly selectiveEZH2 methyltransferaseinhibitor withIC50of 9.9 nM
52113PFI-21627676-59-898% 
PFI-2 is a potent, selective, and cell-activelysine methyltransferase SETD7inhibitor
52311Torin 21223001-51-198% 
Torin 2 is a potent and selectivemTORinhibitor withIC50of 0.25 nM; 800-fold greater s
52402WH-4-023837422-57-898% 
WH-4-023 is a potent and orally activeLck/Srcinhibitor withIC50of 2 nM and 6 nM, resp