TRV130 ( Oliceridine )
Catalog No: 51910
CAS Number: 1401031-39-7
Purity: ≧98.0%
TRV 130 Hcl is a novel -opioid receptor (MOR) G protein-biased ligand; elicits robust G protein signaling ( pEC50=8.1), with potency and efficacy similar to morphine, but with far less -arrestin recruitment and receptor internalization.
For research use only. We do not sell to patients.
Chemical Information
| Name | TRV130 ( Oliceridine ) |
|---|---|
| Iupac Chemical Name | (R)-N-((3-methoxythiophen-2-yl)methyl)-2-(9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl)ethanamine hydrochloride |
| Synonyms | TRV-130 ；TRV130 ；TRV 130 ；Oliceridine |
| Molecular Formula | 423.01 |
| Molecular Weight | C22H31ClN2O2S |
| Smile | COC1=C(CNCC[C@@](C2)(C3=NC=CC=C3)CCOC42CCCC4)SC=C1.[H]Cl |
| InChiKey | YIIWXYLJZRISQP-ZMBIFBSDSA-N |
| InChi | InChI=1S/C22H30N2O2S.ClH/c1-25-18-7-15-27-19(18)16-23-13-10-21(20-6-2-5-12-24-20)11-14-26-22(17-21)8-3-4-9-22;/h2,5-7,12,15,23H,3-4,8-11,13-14,16-17H2,1H3;1H/t21-;/m1./s1 |
| CAS Number | 1401031-39-7 |
| Related CAS | 1401031-39-7 (HCl) 1401028-24-7 (free base) |
Ordering Information
| Packaging | Price | Availability | Purity | Shipping Time |
|---|---|---|---|---|
| Bulk | Enquiry | Enquiry | Enquiry |
| Formulation | white solid |
|---|---|
| Purity | ≧98.0% |
| Storage | 3 years -20ºCpowder |
| Solubility | 5mg/ml in DMSO |
| Handling | Avoid inhalation, contact with eyes and skin. Avoid dust and aerosol formation. Use only in areas with appropriate exhaust ventilation. |
| Shipping Condition | Shipped under ambient temperature. |
| HS Code |
Coming soon.
| Targets | |
|---|---|
| Mechanism | |
| Cell study | |
| Animal study | |
| Clinical study |
Not available
Chemical Structure
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